NO20053498L - Derivater av aryl-quinaolin/aryl-2-amino-fenylmetanon som fremmer frigivelse av paratyroidhormon - Google Patents

Derivater av aryl-quinaolin/aryl-2-amino-fenylmetanon som fremmer frigivelse av paratyroidhormon

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Publication number
NO20053498L
NO20053498L NO20053498A NO20053498A NO20053498L NO 20053498 L NO20053498 L NO 20053498L NO 20053498 A NO20053498 A NO 20053498A NO 20053498 A NO20053498 A NO 20053498A NO 20053498 L NO20053498 L NO 20053498L
Authority
NO
Norway
Prior art keywords
aryl
parathyroid hormone
quinaolin
phenylmethanone
derivatives
Prior art date
Application number
NO20053498A
Other languages
English (en)
Other versions
NO331845B1 (no
Inventor
Leo Widler
Eva Altmann
Marc Gerspacher
Renee Beerli
Johanne Renaud
Original Assignee
Novartis Ag
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9950319&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20053498(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO20053498L publication Critical patent/NO20053498L/no
Publication of NO331845B1 publication Critical patent/NO331845B1/no

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    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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Abstract

Forbindelse med formel I hvori Rl, R2, R3 og Y er som definert heri, eller en farmasøytisk akseptabel og spaltbar ester, eller syreaddisjonssalt derav, anvendelig for å fremme frigivelse av paratyroidhormon, for eksempel for å hindre eller behandle bentilstander som er assosiert med kalsiumutmagring eller resorpsjon eller hvori stimulering av bendannelse og kalsiumfiksering i benet er ønskelig.
NO20053498A 2002-12-23 2005-07-18 Nye forbindelser, anvendelse derav for a forebygge eller behandle bentilstander, og farmasoytiske sammensetninger med slike forbindelser NO331845B1 (no)

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GBGB0230015.0A GB0230015D0 (en) 2002-12-23 2002-12-23 Organic compounds
PCT/EP2003/014741 WO2004056365A2 (en) 2002-12-23 2003-12-22 Derivatives of aryl-quinazoline/aryl-2amino-phenyl methanone which promote the release of parathyroid hormone

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NO331845B1 NO331845B1 (no) 2012-04-23

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NO331845B1 (no) 2012-04-23
US7696216B2 (en) 2010-04-13
PE20040971A1 (es) 2005-01-12
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MY152921A (en) 2014-12-15
KR20050094822A (ko) 2005-09-28
PT1585521E (pt) 2008-09-30
US20100063075A1 (en) 2010-03-11
EP1844780A3 (en) 2008-03-05
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EP1585521B8 (en) 2009-03-25
WO2004056365A2 (en) 2004-07-08
EP1844780A2 (en) 2007-10-17
PL378916A1 (pl) 2006-05-29
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CA2509151A1 (en) 2004-07-08
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