NO20014242L - Alkenyl- og alkynyl-inneholdende metalloprotease inhibitorer - Google Patents

Alkenyl- og alkynyl-inneholdende metalloprotease inhibitorer

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Publication number
NO20014242L
NO20014242L NO20014242A NO20014242A NO20014242L NO 20014242 L NO20014242 L NO 20014242L NO 20014242 A NO20014242 A NO 20014242A NO 20014242 A NO20014242 A NO 20014242A NO 20014242 L NO20014242 L NO 20014242L
Authority
NO
Norway
Prior art keywords
alkynyl
alkenyl
metalloprotease inhibitors
containing metalloprotease
inhibitors
Prior art date
Application number
NO20014242A
Other languages
English (en)
Norwegian (no)
Other versions
NO20014242D0 (no
Inventor
Menyan Cheng
Neil Gregory Almstead
Michael George Natchus
Stanislaw Pikul
Biswanath De
Roger Gunnard Bookland
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of NO20014242D0 publication Critical patent/NO20014242D0/no
Publication of NO20014242L publication Critical patent/NO20014242L/no

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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/337—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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    • C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
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    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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NO20014242A 1999-03-03 2001-08-31 Alkenyl- og alkynyl-inneholdende metalloprotease inhibitorer NO20014242L (no)

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PE20001565A1 (es) 2001-02-02
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IL145089A0 (en) 2002-06-30
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WO2000051975A1 (en) 2000-09-08
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CA2364878A1 (en) 2000-09-08
BR0008716A (pt) 2002-09-24
CZ20013176A3 (cs) 2002-04-17
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HK1044754A1 (zh) 2002-11-01
ZA200106967B (en) 2002-03-13
EP1165501A1 (en) 2002-01-02
TR200102523T2 (tr) 2002-02-21
US6197770B1 (en) 2001-03-06
CN1349498A (zh) 2002-05-15
NO20014242D0 (no) 2001-08-31

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