MX2020010556A - Inhibidores de cinasa de insercion proviral en linfomas murinos (pim) para el tratamiento de neoplasias mieloproliferativas y fibrosis asociadas con cancer. - Google Patents
Inhibidores de cinasa de insercion proviral en linfomas murinos (pim) para el tratamiento de neoplasias mieloproliferativas y fibrosis asociadas con cancer.Info
- Publication number
- MX2020010556A MX2020010556A MX2020010556A MX2020010556A MX2020010556A MX 2020010556 A MX2020010556 A MX 2020010556A MX 2020010556 A MX2020010556 A MX 2020010556A MX 2020010556 A MX2020010556 A MX 2020010556A MX 2020010556 A MX2020010556 A MX 2020010556A
- Authority
- MX
- Mexico
- Prior art keywords
- cancer
- treatment
- fibrosis associated
- myeloproliferative neoplasms
- kinase inhibitors
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Abstract
Se proporcionan métodos para el tratamiento de neoplasias mieloproliferativas y/o fibrosis asociadas con cáncer. Los métodos descritos comprenden administrar un inhibidor de cinasa PIM, y opcionalmente un inhibidor de cinasa JAK u otro agente terapéutico, a un mamífero que lo necesite.
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862657563P | 2018-04-13 | 2018-04-13 | |
US201862657540P | 2018-04-13 | 2018-04-13 | |
US201862743469P | 2018-10-09 | 2018-10-09 | |
US201862753025P | 2018-10-30 | 2018-10-30 | |
US201862753023P | 2018-10-30 | 2018-10-30 | |
PCT/US2019/027217 WO2019200254A1 (en) | 2018-04-13 | 2019-04-12 | Pim kinase inhibitors for treatment of myeloproliferative neoplasms and fibrosis associated with cancer |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2020010556A true MX2020010556A (es) | 2021-03-02 |
Family
ID=68164545
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2020010556A MX2020010556A (es) | 2018-04-13 | 2019-04-12 | Inhibidores de cinasa de insercion proviral en linfomas murinos (pim) para el tratamiento de neoplasias mieloproliferativas y fibrosis asociadas con cancer. |
MX2023001425A MX2023001425A (es) | 2018-04-13 | 2020-10-06 | Inhibidores de cinasa de insercion proviral en linfomas murinos (pim) para el tratamiento de neoplasias mieloproliferativas y fibrosis asociadas con cancer. |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2023001425A MX2023001425A (es) | 2018-04-13 | 2020-10-06 | Inhibidores de cinasa de insercion proviral en linfomas murinos (pim) para el tratamiento de neoplasias mieloproliferativas y fibrosis asociadas con cancer. |
Country Status (9)
Country | Link |
---|---|
US (1) | US20210113562A1 (es) |
EP (1) | EP3773560A4 (es) |
JP (2) | JP2021521170A (es) |
KR (1) | KR20200143454A (es) |
CN (2) | CN117838695A (es) |
AU (1) | AU2019252793A1 (es) |
CA (1) | CA3095580A1 (es) |
MX (2) | MX2020010556A (es) |
WO (1) | WO2019200254A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PL3409278T3 (pl) | 2011-07-21 | 2021-02-22 | Sumitomo Pharma Oncology, Inc. | Heterocykliczne inhibitory kinazy białkowej |
JP2022520361A (ja) | 2019-02-12 | 2022-03-30 | スミトモ ダイニッポン ファーマ オンコロジー, インコーポレイテッド | 複素環式タンパク質キナーゼ阻害剤を含む製剤 |
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-
2019
- 2019-04-12 MX MX2020010556A patent/MX2020010556A/es unknown
- 2019-04-12 CA CA3095580A patent/CA3095580A1/en active Pending
- 2019-04-12 US US17/047,383 patent/US20210113562A1/en active Pending
- 2019-04-12 CN CN202311324993.3A patent/CN117838695A/zh active Pending
- 2019-04-12 JP JP2020555451A patent/JP2021521170A/ja active Pending
- 2019-04-12 WO PCT/US2019/027217 patent/WO2019200254A1/en unknown
- 2019-04-12 AU AU2019252793A patent/AU2019252793A1/en active Pending
- 2019-04-12 CN CN201980037795.4A patent/CN112236139A/zh active Pending
- 2019-04-12 KR KR1020207032677A patent/KR20200143454A/ko unknown
- 2019-04-12 EP EP19785217.1A patent/EP3773560A4/en active Pending
-
2020
- 2020-10-06 MX MX2023001425A patent/MX2023001425A/es unknown
-
2024
- 2024-01-25 JP JP2024009550A patent/JP2024038485A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
MX2023001425A (es) | 2023-03-03 |
US20210113562A1 (en) | 2021-04-22 |
JP2024038485A (ja) | 2024-03-19 |
KR20200143454A (ko) | 2020-12-23 |
CN112236139A (zh) | 2021-01-15 |
JP2021521170A (ja) | 2021-08-26 |
EP3773560A1 (en) | 2021-02-17 |
WO2019200254A1 (en) | 2019-10-17 |
EP3773560A4 (en) | 2022-01-19 |
CN117838695A (zh) | 2024-04-09 |
CA3095580A1 (en) | 2019-10-17 |
AU2019252793A1 (en) | 2020-10-15 |
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