MX2009000333A - Pirrilopirimidinas para composiciones farmaceuticas. - Google Patents

Pirrilopirimidinas para composiciones farmaceuticas.

Info

Publication number
MX2009000333A
MX2009000333A MX2009000333A MX2009000333A MX2009000333A MX 2009000333 A MX2009000333 A MX 2009000333A MX 2009000333 A MX2009000333 A MX 2009000333A MX 2009000333 A MX2009000333 A MX 2009000333A MX 2009000333 A MX2009000333 A MX 2009000333A
Authority
MX
Mexico
Prior art keywords
pharmaceutical compositions
pyrrolopyrimidines
pyrrolopyrimidine compounds
relates
present
Prior art date
Application number
MX2009000333A
Other languages
English (en)
Inventor
Stefan Jaekel
Tanja Reuter
Stephen Murfin
Steven Taylor
Thomas Stephen Coulter
Original Assignee
Develogen Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Develogen Ag filed Critical Develogen Ag
Publication of MX2009000333A publication Critical patent/MX2009000333A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • A—HUMAN NECESSITIES
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    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
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    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
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    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
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    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
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    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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Abstract

La presente invención se refiere a nuevos compuestos de pirrolopirimidina y a composiciones farmacéuticas que comprenden dichos compuestos de pirrolopirimidina. Además, la presente invención se refiere al uso de los compuestos de pirrolopirimidina de la invención para la producción de composiciones farmacéuticas para la profilaxis y/o el tratamiento de enfermedades que pueden verse influenciadas por la inhibición de la actividad quinasa de Mnk1 y/o Mnk2 (Mnk2a o Mnk2b) y/o de variantes adicionales de las mismas.
MX2009000333A 2006-07-10 2007-07-10 Pirrilopirimidinas para composiciones farmaceuticas. MX2009000333A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06014297A EP1889847A1 (en) 2006-07-10 2006-07-10 Pyrrolopyrimidines for pharmaceutical compositions
PCT/EP2007/006109 WO2008006547A2 (en) 2006-07-10 2007-07-10 Pyrrolopyrimidines for pharmaceutical compositions

Publications (1)

Publication Number Publication Date
MX2009000333A true MX2009000333A (es) 2009-03-13

Family

ID=37496429

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009000333A MX2009000333A (es) 2006-07-10 2007-07-10 Pirrilopirimidinas para composiciones farmaceuticas.

Country Status (16)

Country Link
US (1) US8697713B2 (es)
EP (2) EP1889847A1 (es)
JP (1) JP5331951B2 (es)
KR (1) KR20090039757A (es)
CN (1) CN101511837A (es)
AT (1) ATE526331T1 (es)
AU (1) AU2007271928A1 (es)
BR (1) BRPI0712882A2 (es)
CA (1) CA2690277A1 (es)
CO (1) CO6150162A2 (es)
EA (1) EA200900136A1 (es)
IL (1) IL196391A0 (es)
MX (1) MX2009000333A (es)
NO (1) NO20090029L (es)
WO (1) WO2008006547A2 (es)
ZA (1) ZA200810785B (es)

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US20100105708A1 (en) 2010-04-29
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ATE526331T1 (de) 2011-10-15
CO6150162A2 (es) 2010-04-20
AU2007271928A1 (en) 2008-01-17
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