LV12686B - Diabeta arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas - Google Patents

Diabeta arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas

Info

Publication number
LV12686B
LV12686B LV010057A LV010057A LV12686B LV 12686 B LV12686 B LV 12686B LV 010057 A LV010057 A LV 010057A LV 010057 A LV010057 A LV 010057A LV 12686 B LV12686 B LV 12686B
Authority
LV
Latvia
Prior art keywords
combination
inhibitor
content
diabetes treatment
pravastatin
Prior art date
Application number
LV010057A
Other languages
English (en)
Other versions
LV12686A (lv
Inventor
Jeffrey Robl
Rex A Parker
Scott A Biller
Haris Jamil
Bruce L Jacobson
Krishna Kodukula
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22280975&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LV12686(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of LV12686A publication Critical patent/LV12686A/lv
Publication of LV12686B publication Critical patent/LV12686B/lv

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Electrical Discharge Machining, Electrochemical Machining, And Combined Machining (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
LV010057A 1998-09-17 2001-04-12 Diabeta arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas LV12686B (lv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10067798P 1998-09-17 1998-09-17
PCT/US1999/020946 WO2000015229A1 (en) 1998-09-17 1999-09-13 METHOD FOR TREATING DIABETES EMPLOYING AN aP2 INHIBITOR AND COMBINATION

Publications (2)

Publication Number Publication Date
LV12686A LV12686A (lv) 2001-07-20
LV12686B true LV12686B (lv) 2001-10-20

Family

ID=22280975

Family Applications (2)

Application Number Title Priority Date Filing Date
LV010058A LV12687B (lv) 1998-09-17 2001-04-12 Aterosklerozes arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas
LV010057A LV12686B (lv) 1998-09-17 2001-04-12 Diabeta arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas

Family Applications Before (1)

Application Number Title Priority Date Filing Date
LV010058A LV12687B (lv) 1998-09-17 2001-04-12 Aterosklerozes arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas

Country Status (30)

Country Link
US (1) US20020035064A1 (lv)
EP (2) EP1121129B1 (lv)
JP (2) JP2002524517A (lv)
KR (2) KR20010079842A (lv)
CN (2) CN1317970A (lv)
AT (1) ATE406898T1 (lv)
AU (2) AU754488B2 (lv)
BG (2) BG105432A (lv)
BR (2) BR9913831A (lv)
CA (2) CA2344300A1 (lv)
CO (2) CO5130026A1 (lv)
CZ (2) CZ2001964A3 (lv)
DE (1) DE69939481D1 (lv)
EE (2) EE200100155A (lv)
ES (1) ES2311306T3 (lv)
GE (2) GEP20033045B (lv)
HU (2) HUP0104108A2 (lv)
ID (2) ID28450A (lv)
IL (2) IL141785A0 (lv)
LT (2) LT4871B (lv)
LV (2) LV12687B (lv)
NO (2) NO20011351L (lv)
NZ (2) NZ510207A (lv)
PE (2) PE20001047A1 (lv)
PL (2) PL346660A1 (lv)
SK (1) SK3202001A3 (lv)
TR (2) TR200100774T2 (lv)
UY (2) UY25714A1 (lv)
WO (2) WO2000015229A1 (lv)
ZA (2) ZA200207433B (lv)

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US6586438B2 (en) 1999-11-03 2003-07-01 Bristol-Myers Squibb Co. Antidiabetic formulation and method
AU3294701A (en) 2000-01-28 2001-08-07 Bristol-Myers Squibb Company Tetrahydropyrimidone inhibitors of fatty acid binding protein and method
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JP6514282B2 (ja) * 2014-03-24 2019-05-15 花王株式会社 Ｇｉｐ上昇抑制剤の評価又は選択方法
JP6223376B2 (ja) * 2014-03-24 2017-11-01 花王株式会社 Ｇｉｐ上昇抑制剤の評価又は選択方法
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Also Published As

Publication number Publication date
PL346661A1 (en) 2002-02-25
LV12687A (lv) 2001-07-20
CN1319012A (zh) 2001-10-24
NO20011352L (no) 2001-05-11
IL141785A0 (en) 2002-03-10
EP1121129A1 (en) 2001-08-08
JP2002524518A (ja) 2002-08-06
EE200100155A (et) 2002-08-15
IL141786A0 (en) 2002-03-10
CZ2001964A3 (cs) 2002-01-16
LT4871B (lt) 2001-12-27
DE69939481D1 (de) 2008-10-16
HUP0104108A2 (hu) 2002-03-28
ES2311306T3 (es) 2009-02-01
HUP0104240A2 (hu) 2002-03-28
PE20001056A1 (es) 2000-12-24
NZ510207A (en) 2003-08-29
ZA200207430B (en) 2003-09-16
EE200100154A (et) 2002-12-16
NZ510209A (en) 2003-07-25
EE04356B1 (et) 2004-10-15
ZA200207433B (en) 2003-10-27
ID27833A (id) 2001-04-26
CA2344300A1 (en) 2000-03-23
EP1113801A4 (en) 2002-10-02
ID28450A (id) 2001-05-24
SK3202001A3 (en) 2002-04-04
JP2002524517A (ja) 2002-08-06
AU6143799A (en) 2000-04-03
EP1121129B1 (en) 2008-09-03
AU754488B2 (en) 2002-11-14
EP1121129A4 (en) 2002-10-16
CO5130025A1 (es) 2002-02-27
WO2000015229A1 (en) 2000-03-23
LT2001022A (en) 2001-08-27
LV12687B (lv) 2001-10-20
EP1113801A1 (en) 2001-07-11
LT2001023A (en) 2001-08-27
CN1317970A (zh) 2001-10-17
NO20011351L (no) 2001-05-11
BR9913831A (pt) 2001-05-29
KR20010079842A (ko) 2001-08-22
BR9913833A (pt) 2001-05-29
TR200100773T2 (tr) 2001-07-23
UY25713A1 (es) 2001-08-27
LV12686A (lv) 2001-07-20
GEP20033044B (en) 2003-08-25
UY25714A1 (es) 2001-08-27
ATE406898T1 (de) 2008-09-15
WO2000015230A1 (en) 2000-03-23
LT4870B (lt) 2001-12-27
CA2344309A1 (en) 2000-03-23
NO20011352D0 (no) 2001-03-16
TR200100774T2 (tr) 2001-12-21
US20020035064A1 (en) 2002-03-21
PL346660A1 (en) 2002-02-25
CO5130026A1 (es) 2002-02-27
AU755563B2 (en) 2002-12-12
NO20011351D0 (no) 2001-03-16
GEP20033045B (en) 2003-08-25
KR20010075150A (ko) 2001-08-09
PE20001047A1 (es) 2000-12-24
CZ2001965A3 (cs) 2002-02-13
BG105432A (en) 2001-12-29
BG105431A (en) 2001-12-29
AU6387799A (en) 2000-04-03

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