ECSP088763A - Nuevas combinaciones terapéuticas para el tratamiento de la depresión - Google Patents

Nuevas combinaciones terapéuticas para el tratamiento de la depresión

Info

Publication number
ECSP088763A
ECSP088763A EC2008008763A ECSP088763A ECSP088763A EC SP088763 A ECSP088763 A EC SP088763A EC 2008008763 A EC2008008763 A EC 2008008763A EC SP088763 A ECSP088763 A EC SP088763A EC SP088763 A ECSP088763 A EC SP088763A
Authority
EC
Ecuador
Prior art keywords
depression
treatment
therapeutic combinations
new therapeutic
combinations
Prior art date
Application number
EC2008008763A
Other languages
English (en)
Inventor
Sharon Joy Rosenzweig-Lipson
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ECSP088763A publication Critical patent/ECSP088763A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4525Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/55131,4-Benzodiazepines, e.g. diazepam or clozapine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/55131,4-Benzodiazepines, e.g. diazepam or clozapine
    • A61K31/55171,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Se proveen combinaciones terapéuticas útiles en el tratamiento o la prevención de la depresión y otros trastornos emocionales; composiciones farmacéuticas que contienen dichas combinaciones; y su uso en el tratamiento o la profilaxis de la depresión u otros trastornos emocionales. Dichos compuestos tienen la fórmula I: Io una de sus sales aceptables para uso farmacéutico, donde cada R1, R2, R3, R4, R5, R6, n y m son como se definen y se describen en esta solicitud.
EC2008008763A 2006-03-24 2008-09-23 Nuevas combinaciones terapéuticas para el tratamiento de la depresión ECSP088763A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US78545406P 2006-03-24 2006-03-24

Publications (1)

Publication Number Publication Date
ECSP088763A true ECSP088763A (es) 2008-10-31

Family

ID=38466269

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2008008763A ECSP088763A (es) 2006-03-24 2008-09-23 Nuevas combinaciones terapéuticas para el tratamiento de la depresión

Country Status (19)

Country Link
US (1) US20070225279A1 (es)
EP (1) EP1998773A2 (es)
JP (1) JP2009531435A (es)
KR (1) KR20080105104A (es)
CN (1) CN101410112A (es)
AR (1) AR060087A1 (es)
AU (1) AU2007231011A1 (es)
BR (1) BRPI0709159A2 (es)
CA (1) CA2644662A1 (es)
CR (1) CR10245A (es)
EC (1) ECSP088763A (es)
IL (1) IL193747A0 (es)
MX (1) MX2008012094A (es)
NO (1) NO20083758L (es)
PA (1) PA8720801A1 (es)
PE (1) PE20080010A1 (es)
RU (1) RU2008135326A (es)
TW (1) TW200806300A (es)
WO (1) WO2007112014A2 (es)

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Also Published As

Publication number Publication date
WO2007112014A3 (en) 2007-12-21
AR060087A1 (es) 2008-05-21
MX2008012094A (es) 2008-10-03
IL193747A0 (en) 2009-08-03
CR10245A (es) 2008-11-26
BRPI0709159A2 (pt) 2011-06-28
WO2007112014A2 (en) 2007-10-04
US20070225279A1 (en) 2007-09-27
CA2644662A1 (en) 2007-10-04
NO20083758L (no) 2008-10-21
JP2009531435A (ja) 2009-09-03
PE20080010A1 (es) 2008-03-10
RU2008135326A (ru) 2010-04-27
PA8720801A1 (es) 2008-11-19
TW200806300A (en) 2008-02-01
AU2007231011A1 (en) 2007-10-04
EP1998773A2 (en) 2008-12-10
KR20080105104A (ko) 2008-12-03
CN101410112A (zh) 2009-04-15

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