UY31673A1 - "derivados heterocíclicos de urea y métodos de uso de los mismos-211" - Google Patents

"derivados heterocíclicos de urea y métodos de uso de los mismos-211"

Info

Publication number
UY31673A1
UY31673A1 UY031673A UY31673A UY31673A1 UY 31673 A1 UY31673 A1 UY 31673A1 UY 031673 A UY031673 A UY 031673A UY 31673 A UY31673 A UY 31673A UY 31673 A1 UY31673 A1 UY 31673A1
Authority
UY
Uruguay
Prior art keywords
methods
same
heterocyclic derivatives
urea
urea heterocyclic
Prior art date
Application number
UY031673A
Other languages
English (en)
Inventor
Shanta Bist
Sherer Brian
Dangel Brian
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40474753&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY31673(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of UY31673A1 publication Critical patent/UY31673A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Abstract

describe procesos para su preparación, composiciones farmacéuticas que los contienen, su uso como medicamentos y su uso en el tratamiento de infecciones bacterianas.
UY031673A 2008-02-26 2009-02-25 "derivados heterocíclicos de urea y métodos de uso de los mismos-211" UY31673A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US3162108P 2008-02-26 2008-02-26

Publications (1)

Publication Number Publication Date
UY31673A1 true UY31673A1 (es) 2009-09-30

Family

ID=40474753

Family Applications (1)

Application Number Title Priority Date Filing Date
UY031673A UY31673A1 (es) 2008-02-26 2009-02-25 "derivados heterocíclicos de urea y métodos de uso de los mismos-211"

Country Status (23)

Country Link
US (1) US20120101100A1 (es)
EP (1) EP2262801A1 (es)
JP (1) JP2011513216A (es)
KR (1) KR20100117681A (es)
CN (1) CN102015699A (es)
AR (1) AR070493A1 (es)
AU (1) AU2009219883A1 (es)
BR (1) BRPI0907562A2 (es)
CA (1) CA2716365A1 (es)
CL (1) CL2009000426A1 (es)
CO (1) CO6290656A2 (es)
CR (1) CR11641A (es)
DO (1) DOP2010000259A (es)
EA (1) EA201001368A1 (es)
EC (1) ECSP10010419A (es)
IL (1) IL207731A0 (es)
MX (1) MX2010009163A (es)
PE (1) PE20091573A1 (es)
SA (1) SA109300138B1 (es)
TW (1) TW200940537A (es)
UY (1) UY31673A1 (es)
WO (1) WO2009106885A1 (es)
ZA (1) ZA201005997B (es)

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RU2011123647A (ru) 2008-11-10 2012-12-20 Вертекс Фармасьютикалз Инкорпорейтед Соединения, полезные в качестве ингибиторов atr киназы
CN106496210B (zh) 2008-12-19 2020-06-09 沃泰克斯药物股份有限公司 用作atr激酶抑制剂的化合物
CA2750935A1 (en) 2009-01-30 2010-08-12 Millennium Pharmaceuticals, Inc. Heteroaryls and their use as pi3k inhibitors
US9090601B2 (en) * 2009-01-30 2015-07-28 Millennium Pharmaceuticals, Inc. Thiazole derivatives
US8796314B2 (en) 2009-01-30 2014-08-05 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
TW201102065A (en) 2009-05-29 2011-01-16 Astrazeneca Ab Heterocyclic urea derivatives and methods of use thereof
FR2953519B1 (fr) * 2009-12-08 2012-02-10 Commissariat Energie Atomique Nouveaux composes chimiques aptes a complexer au moins un element metallique et complexe de coordination a base de ces composes
US20130096119A1 (en) 2010-03-31 2013-04-18 Daniel Bur Isoquinolin-3-Ylurea Derivatives
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US9133123B2 (en) 2010-04-23 2015-09-15 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
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US8623869B2 (en) 2010-06-23 2014-01-07 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of ATR kinase
JP2013536193A (ja) 2010-08-11 2013-09-19 ミレニアム ファーマシューティカルズ， インコーポレイテッド ヘテロアリール類およびその使用
WO2012021615A1 (en) 2010-08-11 2012-02-16 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
WO2012021611A1 (en) 2010-08-11 2012-02-16 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
US9056832B2 (en) * 2010-09-17 2015-06-16 Purdue Pharma L.P. Pyridine compounds and the users thereof
WO2012051410A2 (en) 2010-10-13 2012-04-19 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
AR088729A1 (es) 2011-03-29 2014-07-02 Actelion Pharmaceuticals Ltd Derivados de 3-ureidoisoquinolin-8-ilo y una composicion farmaceutica
KR20140027974A (ko) 2011-04-05 2014-03-07 버텍스 파마슈티칼스 인코포레이티드 Ｔｒａ 키나제의 억제제로서 유용한 아미노피라진 화합물
US8822469B2 (en) 2011-06-22 2014-09-02 Vertex Pharmaceuticals Incorporated Pyrrolo[2,3-B]pyrazines useful as inhibitors of ATR kinase
US9096602B2 (en) 2011-06-22 2015-08-04 Vertex Pharmaceuticals Incorporated Substituted pyrrolo[2,3-B]pyrazines as ATR kinase inhibitors
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RU2014111321A (ru) * 2011-09-12 2015-10-20 Ф. Хоффманн-Ля Рош Аг Гидразиды 3-пиридинкарбоновых кислот в качестве агентов, повышающих содержание холестерина липопротеинов высокой плотности
MX2014003796A (es) 2011-09-30 2015-01-16 Vertex Pharma Compuestos utiles como inhibidores de la cinasa ataxia telangiectasia mutada y rad3 relacionados (atr).
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RU2677292C2 (ru) 2011-09-30 2019-01-16 Вертекс Фармасьютикалз Инкорпорейтед Способы получения соединений, которые можно использовать в качестве ингибиторов киназы atr
CA2850491C (en) 2011-09-30 2020-10-27 Vertex Pharmaceuticals Incorporated Treating pancreatic cancer and non-small cell lung cancer with atr inhibiors
US8853217B2 (en) 2011-09-30 2014-10-07 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of ATR kinase
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WO2013071093A1 (en) 2011-11-09 2013-05-16 Vertex Pharmaceuticals Incorporated Pyrazine compounds useful as inhibitors of atr kinase
WO2013071088A1 (en) 2011-11-09 2013-05-16 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
US8841449B2 (en) 2011-11-09 2014-09-23 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of ATR kinase
EP2776422A1 (en) 2011-11-09 2014-09-17 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
JP5957537B2 (ja) * 2011-12-21 2016-07-27 ビオタ ヨーロッパ リミテッドＢｉｏｔａ Ｅｕｒｏｐｅ Ｌｔｄ 複素環式ウレア化合物
WO2013152298A1 (en) 2012-04-05 2013-10-10 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase and combination therapies thereof
JP5977349B2 (ja) * 2012-06-15 2016-08-24 田辺三菱製薬株式会社 芳香族複素環化合物
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Also Published As

Publication number Publication date
US20120101100A1 (en) 2012-04-26
CN102015699A (zh) 2011-04-13
PE20091573A1 (es) 2009-11-12
ECSP10010419A (es) 2010-09-30
JP2011513216A (ja) 2011-04-28
CL2009000426A1 (es) 2011-02-11
CR11641A (es) 2010-10-05
WO2009106885A1 (en) 2009-09-03
CA2716365A1 (en) 2009-09-03
SA109300138B1 (ar) 2012-11-03
EP2262801A1 (en) 2010-12-22
DOP2010000259A (es) 2010-09-15
EA201001368A1 (ru) 2011-04-29
TW200940537A (en) 2009-10-01
IL207731A0 (en) 2010-12-30
AU2009219883A1 (en) 2009-09-03
AR070493A1 (es) 2010-04-07
ZA201005997B (en) 2013-01-30
KR20100117681A (ko) 2010-11-03
BRPI0907562A2 (pt) 2017-05-23
CO6290656A2 (es) 2011-06-20
MX2010009163A (es) 2010-09-14

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Effective date: 20180831