EA200970746A1 - Конденсированные циклические соединения в качестве частичных агонистов ppar-гамма - Google Patents

Конденсированные циклические соединения в качестве частичных агонистов ppar-гамма

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Publication number
EA200970746A1
EA200970746A1 EA200970746A EA200970746A EA200970746A1 EA 200970746 A1 EA200970746 A1 EA 200970746A1 EA 200970746 A EA200970746 A EA 200970746A EA 200970746 A EA200970746 A EA 200970746A EA 200970746 A1 EA200970746 A1 EA 200970746A1
Authority
EA
Eurasian Patent Office
Prior art keywords
cyclic compounds
condensed cyclic
gamma agonists
partial ppar
diabetes
Prior art date
Application number
EA200970746A
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English (en)
Inventor
Таисуке Тавараиси
Хироси Имото
Нобуо То
Original Assignee
Такеда Фармасьютикал Компани Лимитед
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39523585&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200970746(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Такеда Фармасьютикал Компани Лимитед filed Critical Такеда Фармасьютикал Компани Лимитед
Publication of EA200970746A1 publication Critical patent/EA200970746A1/ru

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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
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Abstract

Настоящее изобретение относится к средству для профилактики или лечения диабета, которое обладает превосходным гипогликемическим действием и вызывает меньшее число побочных эффектов, таких как увеличение массы тела и тому подобные. Настоящее изобретение относится к средству для профилактики или лечения диабета, которое включает соединение, выраженное формулойгде все символы имеют значения, указанные в описании изобретения, его соль или пролекарство.
EA200970746A 2007-02-09 2008-02-05 Конденсированные циклические соединения в качестве частичных агонистов ppar-гамма EA200970746A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007031221 2007-02-09
PCT/JP2008/052217 WO2008099794A1 (en) 2007-02-09 2008-02-05 Fused ring compounds as partial agonists of ppar-gamma

Publications (1)

Publication Number Publication Date
EA200970746A1 true EA200970746A1 (ru) 2010-02-26

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EA200970746A EA200970746A1 (ru) 2007-02-09 2008-02-05 Конденсированные циклические соединения в качестве частичных агонистов ppar-гамма

Country Status (21)

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US (2) US20110009384A1 (ru)
EP (1) EP2118066A1 (ru)
JP (1) JP2010517935A (ru)
KR (1) KR20090106660A (ru)
CN (1) CN101646653A (ru)
AR (1) AR065206A1 (ru)
AU (1) AU2008215490A1 (ru)
BR (1) BRPI0807014A2 (ru)
CA (1) CA2677736A1 (ru)
CL (1) CL2008000377A1 (ru)
CR (1) CR10991A (ru)
DO (1) DOP2009000202A (ru)
EA (1) EA200970746A1 (ru)
EC (1) ECSP099618A (ru)
IL (1) IL200114A0 (ru)
MA (1) MA31189B1 (ru)
MX (1) MX2009008103A (ru)
PE (1) PE20090068A1 (ru)
TN (1) TN2009000312A1 (ru)
TW (1) TW200838515A (ru)
WO (1) WO2008099794A1 (ru)

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