EA200970447A1 - Соединения и композиции в качестве ингибиторов протеинкиназы - Google Patents

Соединения и композиции в качестве ингибиторов протеинкиназы

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Publication number
EA200970447A1
EA200970447A1 EA200970447A EA200970447A EA200970447A1 EA 200970447 A1 EA200970447 A1 EA 200970447A1 EA 200970447 A EA200970447 A EA 200970447A EA 200970447 A EA200970447 A EA 200970447A EA 200970447 A1 EA200970447 A1 EA 200970447A1
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EA
Eurasian Patent Office
Prior art keywords
compounds
compositions
proteinkinase inhibitors
proteinkinase
inhibitors
Prior art date
Application number
EA200970447A
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English (en)
Inventor
Донателла Кьянелли
Сяолинь ЛИ
Сяодун Лю
Джон Лорен
Валентина Мольтени
Джульет Набакка
Ласло Ревес
Лоренс Б. Перес
Клинтон Брукс
Войцех Врона
Пол В. Мэнли
Вернер Брайтенштайн
Original Assignee
АйАрЭм ЭлЭлСи
Новартис Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by АйАрЭм ЭлЭлСи, Новартис Аг filed Critical АйАрЭм ЭлЭлСи
Publication of EA200970447A1 publication Critical patent/EA200970447A1/ru

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Abstract

Изобретение обеспечивает новый класс соединений, фармацевтических композиций, включающих такие соединения, и способов применения таких соединений для лечения или предупреждения заболеваний или расстройств, связанных с аномальной или нерегулируемой киназной активностью, в частности, заболеваний или расстройств, которые включают аномальную активацию c-kit, PDGFRα и PDGFRβ киназ. Формула (I)
EA200970447A 2006-11-03 2007-11-02 Соединения и композиции в качестве ингибиторов протеинкиназы EA200970447A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86437806P 2006-11-03 2006-11-03
PCT/US2007/083543 WO2008058037A1 (en) 2006-11-03 2007-11-02 Compounds and compositions as protein kinase inhibitors

Publications (1)

Publication Number Publication Date
EA200970447A1 true EA200970447A1 (ru) 2009-10-30

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
EA200970447A EA200970447A1 (ru) 2006-11-03 2007-11-02 Соединения и композиции в качестве ингибиторов протеинкиназы

Country Status (20)

Country Link
US (1) US20100048539A1 (ru)
EP (1) EP2079729A1 (ru)
JP (1) JP2010509349A (ru)
KR (2) KR20120049397A (ru)
CN (1) CN101622244A (ru)
AU (1) AU2007317349B2 (ru)
BR (1) BRPI0718677A2 (ru)
CA (1) CA2668190A1 (ru)
CO (1) CO6241115A2 (ru)
CR (1) CR10755A (ru)
EA (1) EA200970447A1 (ru)
EC (1) ECSP099378A (ru)
IL (1) IL198315A0 (ru)
MA (1) MA30906B1 (ru)
MX (1) MX2009004716A (ru)
NO (1) NO20092138L (ru)
RU (1) RU2009120882A (ru)
SM (1) SMAP200900031A (ru)
TN (1) TN2009000163A1 (ru)
WO (1) WO2008058037A1 (ru)

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