DE602007009272D1 - Adenosinderivate als agonisten am a2a-rezeptor - Google Patents

Adenosinderivate als agonisten am a2a-rezeptor

Info

Publication number
DE602007009272D1
DE602007009272D1 DE602007009272T DE602007009272T DE602007009272D1 DE 602007009272 D1 DE602007009272 D1 DE 602007009272D1 DE 602007009272 T DE602007009272 T DE 602007009272T DE 602007009272 T DE602007009272 T DE 602007009272T DE 602007009272 D1 DE602007009272 D1 DE 602007009272D1
Authority
DE
Germany
Prior art keywords
agonists
receptor
adenosine derivatives
adenosine
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602007009272T
Other languages
English (en)
Inventor
Robin Alec Fairhurst
Roger John Taylor
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis AG filed Critical Novartis AG
Publication of DE602007009272D1 publication Critical patent/DE602007009272D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/16—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
DE602007009272T 2006-09-14 2007-09-13 Adenosinderivate als agonisten am a2a-rezeptor Active DE602007009272D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06120706A EP1903044A1 (de) 2006-09-14 2006-09-14 Adenosinderivate als Agonisten des A2A-Rezeptors
PCT/EP2007/059666 WO2008031875A1 (en) 2006-09-14 2007-09-13 Adenosine derivatives as a2a receptor agonists

Publications (1)

Publication Number Publication Date
DE602007009272D1 true DE602007009272D1 (de) 2010-10-28

Family

ID=37622170

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602007009272T Active DE602007009272D1 (de) 2006-09-14 2007-09-13 Adenosinderivate als agonisten am a2a-rezeptor

Country Status (31)

Country Link
US (1) US8188100B2 (de)
EP (2) EP1903044A1 (de)
JP (1) JP2010503639A (de)
KR (1) KR20090040386A (de)
CN (1) CN101511831B (de)
AR (1) AR062768A1 (de)
AT (1) ATE481404T1 (de)
AU (1) AU2007296227A1 (de)
BR (1) BRPI0716936A2 (de)
CA (1) CA2662104A1 (de)
CL (1) CL2007002658A1 (de)
CR (1) CR10621A (de)
CY (1) CY1110990T1 (de)
DE (1) DE602007009272D1 (de)
DK (1) DK2066669T3 (de)
ES (1) ES2353141T3 (de)
HK (1) HK1131392A1 (de)
HR (1) HRP20100694T1 (de)
IL (1) IL197153A0 (de)
MA (1) MA30722B1 (de)
MX (1) MX2009002811A (de)
NO (1) NO20091244L (de)
PE (1) PE20081151A1 (de)
PL (1) PL2066669T3 (de)
PT (1) PT2066669E (de)
RU (1) RU2009113668A (de)
SI (1) SI2066669T1 (de)
TN (1) TN2009000084A1 (de)
TW (1) TW200821324A (de)
WO (1) WO2008031875A1 (de)
ZA (1) ZA200901036B (de)

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US8188100B2 (en) 2012-05-29
TW200821324A (en) 2008-05-16
CR10621A (es) 2009-03-27
ZA200901036B (en) 2010-01-27
CN101511831B (zh) 2012-04-25
AR062768A1 (es) 2008-12-03
HRP20100694T1 (hr) 2011-01-31
EP2066669A1 (de) 2009-06-10
DK2066669T3 (da) 2011-01-10
NO20091244L (no) 2009-04-07
WO2008031875A1 (en) 2008-03-20
PT2066669E (pt) 2010-12-17
IL197153A0 (en) 2009-11-18
RU2009113668A (ru) 2010-10-20
ES2353141T3 (es) 2011-02-25
JP2010503639A (ja) 2010-02-04
PL2066669T3 (pl) 2011-03-31
AU2007296227A1 (en) 2008-03-20
MX2009002811A (es) 2009-03-31
TN2009000084A1 (en) 2010-08-19
HK1131392A1 (en) 2010-01-22
US20090325967A1 (en) 2009-12-31
PE20081151A1 (es) 2008-10-06
CA2662104A1 (en) 2008-03-20
CN101511831A (zh) 2009-08-19
KR20090040386A (ko) 2009-04-23
EP2066669B1 (de) 2010-09-15
ATE481404T1 (de) 2010-10-15
EP1903044A1 (de) 2008-03-26
CL2007002658A1 (es) 2008-08-08
SI2066669T1 (sl) 2011-01-31

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