CY1109629T1 - Συνθεσεις ρυθμιστη υποδοχεα 5ht2c και μεθοδοι χρησης - Google Patents

Συνθεσεις ρυθμιστη υποδοχεα 5ht2c και μεθοδοι χρησης

Info

Publication number
CY1109629T1
CY1109629T1 CY20091101197T CY091101197T CY1109629T1 CY 1109629 T1 CY1109629 T1 CY 1109629T1 CY 20091101197 T CY20091101197 T CY 20091101197T CY 091101197 T CY091101197 T CY 091101197T CY 1109629 T1 CY1109629 T1 CY 1109629T1
Authority
CY
Cyprus
Prior art keywords
methods
5ht2c receptor
compositions
receptor receiver
receiver compositions
Prior art date
Application number
CY20091101197T
Other languages
English (en)
Inventor
Dominic P Behan
Brian M Smith
Christina Bjenning
Original Assignee
Arena Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharmaceuticals, Inc. filed Critical Arena Pharmaceuticals, Inc.
Publication of CY1109629T1 publication Critical patent/CY1109629T1/el

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Liquid Crystal Substances (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cosmetics (AREA)
  • Steroid Compounds (AREA)
  • Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)

Abstract

Η παρούσα εφεύρεση αφορά μια σύνθεση περιλαμβάνουσα φαιντερμίνη και εκλεκτικό αγωνιστή υποδοχέα 5HT-2C. Επιπλέον η εφεύρεση αφορά σύνθεση περιλαμβάνουσα φαιντερμίνη και εκλεκτικό αγωνιστή υποδοχέα 5HT-2C που έχει τον Τύπο (I): ή φαρμακευτικώς αποδεκτό άλας, διαλύτωμα ή υδρίτη αυτού. Αυτές οι συνθέσεις είναι χρήσιμες σε φαρμακευτικές συνθέσεις, των οποίων η χρήση περιλαμβάνει τη θεραπεία παχυσαρκίας.
CY20091101197T 2004-12-23 2009-11-12 Συνθεσεις ρυθμιστη υποδοχεα 5ht2c και μεθοδοι χρησης CY1109629T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US63866704P 2004-12-23 2004-12-23
US68890105P 2005-06-08 2005-06-08
EP05855247A EP1833473B1 (en) 2004-12-23 2005-12-21 5ht2c receptor modulator compositions and methods of use

Publications (1)

Publication Number Publication Date
CY1109629T1 true CY1109629T1 (el) 2014-08-13

Family

ID=36615431

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20091101197T CY1109629T1 (el) 2004-12-23 2009-11-12 Συνθεσεις ρυθμιστη υποδοχεα 5ht2c και μεθοδοι χρησης

Country Status (25)

Country Link
US (4) US8153621B2 (el)
EP (3) EP1833473B1 (el)
JP (1) JP4886700B2 (el)
KR (3) KR101519441B1 (el)
CN (3) CN102627607A (el)
AT (1) ATE442135T1 (el)
AU (1) AU2005322183B2 (el)
BR (1) BRPI0515862A2 (el)
CA (1) CA2588941A1 (el)
CY (1) CY1109629T1 (el)
DE (1) DE602005016601D1 (el)
DK (1) DK1833473T3 (el)
EA (2) EA201100129A1 (el)
ES (1) ES2331656T3 (el)
HK (1) HK1102766A1 (el)
HR (1) HRP20090641T1 (el)
IL (2) IL183565A0 (el)
NZ (2) NZ589951A (el)
PL (1) PL1833473T3 (el)
PT (1) PT1833473E (el)
RS (1) RS50997B (el)
SG (1) SG158168A1 (el)
SI (1) SI1833473T1 (el)
WO (1) WO2006071740A2 (el)
ZA (1) ZA200705165B (el)

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ATE442135T1 (de) 2009-09-15
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NZ589951A (en) 2012-11-30
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