EA200702282A1 - Комбинация феррохина и производного артемизинина для лечения малярии - Google Patents

Комбинация феррохина и производного артемизинина для лечения малярии

Info

Publication number
EA200702282A1
EA200702282A1 EA200702282A EA200702282A EA200702282A1 EA 200702282 A1 EA200702282 A1 EA 200702282A1 EA 200702282 A EA200702282 A EA 200702282A EA 200702282 A EA200702282 A EA 200702282A EA 200702282 A1 EA200702282 A1 EA 200702282A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivative
malaria
combination
treatment
relates
Prior art date
Application number
EA200702282A
Other languages
English (en)
Other versions
EA012630B1 (ru
Inventor
Лоран Фрэсс
Даниэль Тер-Минассян
Original Assignee
Санофи-Авентис
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Санофи-Авентис filed Critical Санофи-Авентис
Publication of EA200702282A1 publication Critical patent/EA200702282A1/ru
Publication of EA012630B1 publication Critical patent/EA012630B1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/47064-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00Medicinal preparations containing inorganic active ingredients
    • A61K33/24Heavy metals; Compounds thereof
    • A61K33/26Iron; Compounds thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

Изобретение относится к комбинации, содержащей феррохин в виде свободного основания, соли, гидрата или сольвата и производное артемизинина. Изобретение относится также к фармацевтической композиции, содержащей феррохин в виде одной из его фармацевтически приемлемых солей, гидрата или сольвата и по меньшей мере одно производное артемизинина. Изобретение относится также к применению такой комбинации для получения лекарственного средства, предназначенного для лечения или профилактики малярии. Изобретение относится также к набору для лечения или профилактики малярии.
EA200702282A 2005-04-20 2006-04-18 Комбинация феррохина и производного артемизинина для лечения малярии EA012630B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0503932A FR2884715B1 (fr) 2005-04-20 2005-04-20 Association entre la ferroquine et un derive d'artemisinine pour le traitement du paludisme
PCT/FR2006/000842 WO2006111647A1 (fr) 2005-04-20 2006-04-18 Association entre la ferroquine et un derive d’artemisinine pour le traitement du paludisme

Publications (2)

Publication Number Publication Date
EA200702282A1 true EA200702282A1 (ru) 2008-02-28
EA012630B1 EA012630B1 (ru) 2009-10-30

Family

ID=35385843

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200702282A EA012630B1 (ru) 2005-04-20 2006-04-18 Комбинация феррохина и производного артемизинина для лечения малярии

Country Status (30)

Country Link
US (1) US20120258945A1 (ru)
EP (1) EP1874293A1 (ru)
JP (1) JP5148478B2 (ru)
KR (1) KR20080009088A (ru)
CN (2) CN102836163A (ru)
AP (1) AP2782A (ru)
AR (1) AR054253A1 (ru)
AU (1) AU2006238506B2 (ru)
BR (1) BRPI0610851A2 (ru)
CA (1) CA2605385A1 (ru)
CR (1) CR9425A (ru)
DO (1) DOP2006000092A (ru)
EA (1) EA012630B1 (ru)
FR (1) FR2884715B1 (ru)
GT (1) GT200600157A (ru)
HN (1) HN2006015130A (ru)
IL (1) IL186048A0 (ru)
MA (1) MA29451B1 (ru)
MX (1) MX2007012645A (ru)
MY (1) MY145581A (ru)
NO (1) NO20075920L (ru)
NZ (1) NZ562117A (ru)
PA (1) PA8669801A1 (ru)
PE (2) PE20061314A1 (ru)
SG (1) SG161270A1 (ru)
TN (1) TNSN07359A1 (ru)
TW (1) TWI387456B (ru)
UA (1) UA96414C2 (ru)
WO (1) WO2006111647A1 (ru)
ZA (1) ZA200708800B (ru)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2926993B1 (fr) * 2008-02-06 2011-03-11 Sanofi Aventis Association entre un sel de bis-thiazolium ou l'un de ses precurseurs et l'artemisinine ou l'un de ses derives pour le traitement du paludisme
FR2952823B1 (fr) * 2009-10-30 2012-04-20 Sanofi Aventis Utilisation de la ferroquine dans le traitement ou la prevention du paludisme
FR2951945B1 (fr) 2009-11-05 2013-08-09 Sanofi Aventis Composition pharmaceutique
FR2961209B1 (fr) * 2010-06-11 2013-03-01 Sanofi Aventis Procede de synthese de la ferroquine par amination reductrice convergente.
FR2989588A1 (fr) * 2012-04-19 2013-10-25 Centre Nat Rech Scient Composes pour la prevention ou le traitement des infections par des virus de la famille des flaviviridae
MX2016005959A (es) 2013-11-08 2016-10-14 Exthera Medical Corp Métodos para diagnosticar enfermedades infecciosas usando medio de adsorción.
CN105250295B (zh) * 2014-07-07 2018-12-25 广州中医药大学科技产业园有限公司 一种联合用药物及其作为免疫调节剂的应用
WO2017015344A1 (en) * 2015-07-20 2017-01-26 University Of Vermont And State Agricultural College Use of cymanquine compounds as antimalarial agents
CN107802755A (zh) * 2017-11-08 2018-03-16 江西龙卿堂科技有限公司 一种具有防蚊防疟作用的青蒿软膏
KR102073961B1 (ko) * 2018-11-16 2020-02-05 (주)프론트바이오 메트포르민 및 페로센계 화합물을 유효성분으로 함유하는 암 예방 또는 치료용 약학적 조성물
WO2022231238A1 (ko) * 2021-04-26 2022-11-03 심민보 아르테수네이트 또는 그의 염, 및 피로나리딘 또는 그의 염의 해열, 항염증, 항바이러스용, 또는 covid-19 예방 또는 치료용 약학적 조성물 및 이를 이용한 방법
CN113952360B (zh) * 2021-09-14 2023-03-10 上海交通大学 一种亚铁离子在治疗疟疾的药物中的应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN166154B (ru) * 1987-05-08 1990-03-24 Hoechst India
ZA200602031B (en) * 2003-09-04 2007-05-30 Cipla Ltd Antimalarial compositions and process thereof

Also Published As

Publication number Publication date
MX2007012645A (es) 2007-12-13
FR2884715A1 (fr) 2006-10-27
EA012630B1 (ru) 2009-10-30
PE20061314A1 (es) 2006-12-27
JP5148478B2 (ja) 2013-02-20
CN101163470A (zh) 2008-04-16
MY145581A (en) 2012-02-29
TW200716092A (en) 2007-05-01
PA8669801A1 (es) 2006-11-09
TWI387456B (zh) 2013-03-01
US20120258945A1 (en) 2012-10-11
NO20075920L (no) 2007-11-16
DOP2006000092A (es) 2006-11-15
NZ562117A (en) 2010-01-29
CA2605385A1 (fr) 2006-10-26
EP1874293A1 (fr) 2008-01-09
FR2884715B1 (fr) 2007-06-15
ZA200708800B (en) 2009-01-28
AR054253A1 (es) 2007-06-13
WO2006111647A1 (fr) 2006-10-26
AU2006238506B2 (en) 2012-03-01
JP2008536900A (ja) 2008-09-11
CN102836163A (zh) 2012-12-26
BRPI0610851A2 (pt) 2010-08-03
UA96414C2 (ru) 2011-11-10
HN2006015130A (es) 2010-08-19
PE20110119A1 (es) 2011-03-08
AU2006238506A1 (en) 2006-10-26
CR9425A (es) 2008-02-20
TNSN07359A1 (en) 2008-12-31
AP2782A (en) 2013-10-31
AP2007004211A0 (en) 2007-10-31
SG161270A1 (en) 2010-05-27
KR20080009088A (ko) 2008-01-24
GT200600157A (es) 2006-11-07
IL186048A0 (en) 2008-02-09
MA29451B1 (fr) 2008-05-02

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM

MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): RU