CN101663303A - 杂芳族化合物、其制备方法以及其用途 - Google Patents

杂芳族化合物、其制备方法以及其用途 Download PDF

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Publication number
CN101663303A
CN101663303A CN200880012573A CN200880012573A CN101663303A CN 101663303 A CN101663303 A CN 101663303A CN 200880012573 A CN200880012573 A CN 200880012573A CN 200880012573 A CN200880012573 A CN 200880012573A CN 101663303 A CN101663303 A CN 101663303A
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mesyl
bases
amine
amino
compound
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CN101663303B (zh
Inventor
陈刚胜
刘圣
熊龙
杨宝海
冯瑞茂
何雷
吕爱锋
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Abstract

本发明涉及通式(I)的杂芳族化合物、其制备方法以及用途，通式(I)中，A、D、Y如说明书所定义。

Description

PCT国内申请，说明书已公开。

Claims (1)

  1. PCT国内申请，权利要求书已公开。
CN2008800125739A 2008-01-22 2008-12-23 杂芳族化合物、其制备方法以及其用途 Expired - Fee Related CN101663303B (zh)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN2008800125739A CN101663303B (zh) 2008-01-22 2008-12-23 杂芳族化合物、其制备方法以及其用途

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CNA2008100008154A CN101492445A (zh) 2008-01-22 2008-01-22 杂芳族化合物、其制备方法以及其用途
CN200810000815.4 2008-01-22
CN2008800125739A CN101663303B (zh) 2008-01-22 2008-12-23 杂芳族化合物、其制备方法以及其用途
PCT/CN2008/002046 WO2009094831A1 (fr) 2008-01-22 2008-12-23 Composés hétéroaromatiques, leur procédé de préparation et leur utilisation

Publications (2)

Publication Number Publication Date
CN101663303A true CN101663303A (zh) 2010-03-03
CN101663303B CN101663303B (zh) 2012-06-27

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CNA2008100008154A Pending CN101492445A (zh) 2008-01-22 2008-01-22 杂芳族化合物、其制备方法以及其用途
CN2008800125739A Expired - Fee Related CN101663303B (zh) 2008-01-22 2008-12-23 杂芳族化合物、其制备方法以及其用途

Family Applications Before (1)

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CNA2008100008154A Pending CN101492445A (zh) 2008-01-22 2008-01-22 杂芳族化合物、其制备方法以及其用途

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CN (2) CN101492445A (zh)
TW (1) TW201002704A (zh)
WO (1) WO2009094831A1 (zh)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101735200B (zh) * 2008-11-17 2013-01-02 岑均达 喹唑啉类化合物
CN101787017A (zh) * 2009-01-23 2010-07-28 岑均达 光学纯喹唑啉类化合物
CN102344445B (zh) * 2010-07-23 2015-11-25 岑均达 光学纯喹唑啉类化合物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL112249A (en) * 1994-01-25 2001-11-25 Warner Lambert Co Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds
RS49779B (sr) * 1998-01-12 2008-06-05 Glaxo Group Limited, Biciklična heteroaromatična jedinjenja kao inhibitori protein tirozin kinaze

Also Published As

Publication number Publication date
WO2009094831A1 (fr) 2009-08-06
TW201002704A (en) 2010-01-16
CN101492445A (zh) 2009-07-29
CN101663303B (zh) 2012-06-27

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Granted publication date: 20120627

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CF01 Termination of patent right due to non-payment of annual fee