BR9906903A - Composição com liberação sustentada, processos para produzir a mesma, para suprimir a brusca liberação inicial da susbtância bioativa de uma composição com liberação sustentada e para aumentar a eficiência da inclusão da substância bioativa em uma composição com liberação sustentada, produto farmacêutico, agente para prevenir ou tratar câncer prostático, hipertrofia prostática, endometriose, histeromioma, metrofibroma, puberdade precoce, dismenorréia, ou câncer do seio, ou um contraceptivo, e, composto - Google Patents
Composição com liberação sustentada, processos para produzir a mesma, para suprimir a brusca liberação inicial da susbtância bioativa de uma composição com liberação sustentada e para aumentar a eficiência da inclusão da substância bioativa em uma composição com liberação sustentada, produto farmacêutico, agente para prevenir ou tratar câncer prostático, hipertrofia prostática, endometriose, histeromioma, metrofibroma, puberdade precoce, dismenorréia, ou câncer do seio, ou um contraceptivo, e, compostoInfo
- Publication number
- BR9906903A BR9906903A BR9906903-2A BR9906903A BR9906903A BR 9906903 A BR9906903 A BR 9906903A BR 9906903 A BR9906903 A BR 9906903A BR 9906903 A BR9906903 A BR 9906903A
- Authority
- BR
- Brazil
- Prior art keywords
- composition
- sustained release
- bioactive substance
- release
- metrofibroma
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/24—Follicle-stimulating hormone [FSH]; Chorionic gonadotropins, e.g. HCG; Luteinising hormone [LH]; Thyroid-stimulating hormone [TSH]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
- A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Organic Chemistry (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Gastroenterology & Hepatology (AREA)
- Inorganic Chemistry (AREA)
- Zoology (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Abstract
"COMPOSIçãO COM LIBERAçãO SUSTENTADA, PROCESSOS PARA PRODUZIR A MESMA, PARA SUPRIMIR A BRUSCA LIBERAçãO INICIAL DA SUBSTâNCIA BIOATIVA DE UMA COMPOSIçãO COM LIBERAçãO SUSTENTADA E PARA AUMENTAR EFICIêNCIA DA INCLUSãO DA SUBSTâNCIA BIOATIVA EM UMA COMPOSIçãO COM LIBERAçãO SUSTENTADA, PRODUTO FARMACêUTICO, AGENTE PARA PREVENIR OU TRATAR CâNCER PROSTáTICO, HIPERTROFIA PROSTáTICA, ENDOMETRIOSE, HISTEROMIOMA, METROFIBROMA, PUBERDADE PRECOCE, DISMENORRéIA, OU CâNCER DO SEIO, OU UM CONTRACEPTIVO, E, COMPOSTO" Composição com liberação sustentada contendo um sal de ácido hidroxinaftóico de uma substância biologicamente ativa e um polímero biodegradável, uma processo para sua produção, e uma composição farmacêutica contendo a mencionada composição com liberação sustentada.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP641298 | 1998-01-16 | ||
PCT/JP1999/000086 WO1999036099A1 (fr) | 1998-01-16 | 1999-01-13 | Compositions a liberation controlee, leur procede de fabrication et leur utilisation |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9906903A true BR9906903A (pt) | 2000-12-12 |
Family
ID=11637664
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9906903-2A BR9906903A (pt) | 1998-01-16 | 1999-01-13 | Composição com liberação sustentada, processos para produzir a mesma, para suprimir a brusca liberação inicial da susbtância bioativa de uma composição com liberação sustentada e para aumentar a eficiência da inclusão da substância bioativa em uma composição com liberação sustentada, produto farmacêutico, agente para prevenir ou tratar câncer prostático, hipertrofia prostática, endometriose, histeromioma, metrofibroma, puberdade precoce, dismenorréia, ou câncer do seio, ou um contraceptivo, e, composto |
Country Status (19)
Country | Link |
---|---|
US (2) | US6740634B1 (pt) |
EP (1) | EP1048301A4 (pt) |
KR (1) | KR100577877B1 (pt) |
CN (1) | CN1199686C (pt) |
AU (1) | AU758596B2 (pt) |
BR (1) | BR9906903A (pt) |
CA (1) | CA2316273A1 (pt) |
HR (1) | HRP20000471A2 (pt) |
HU (1) | HUP0100221A3 (pt) |
IL (1) | IL136951A0 (pt) |
IS (1) | IS5560A (pt) |
NO (1) | NO20003530L (pt) |
NZ (1) | NZ505651A (pt) |
OA (1) | OA11446A (pt) |
PL (1) | PL341733A1 (pt) |
RU (1) | RU2230550C2 (pt) |
SK (1) | SK10272000A3 (pt) |
TR (1) | TR200002059T2 (pt) |
WO (1) | WO1999036099A1 (pt) |
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1999
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- 1999-01-13 BR BR9906903-2A patent/BR9906903A/pt not_active IP Right Cessation
- 1999-01-13 CA CA002316273A patent/CA2316273A1/en not_active Abandoned
- 1999-01-13 SK SK1027-2000A patent/SK10272000A3/sk unknown
- 1999-01-13 IL IL13695199A patent/IL136951A0/xx not_active IP Right Cessation
- 1999-01-13 EP EP99900300A patent/EP1048301A4/en not_active Withdrawn
- 1999-01-13 TR TR2000/02059T patent/TR200002059T2/xx unknown
- 1999-01-13 HU HU0100221A patent/HUP0100221A3/hu unknown
- 1999-01-13 AU AU18897/99A patent/AU758596B2/en not_active Ceased
- 1999-01-13 WO PCT/JP1999/000086 patent/WO1999036099A1/ja not_active Application Discontinuation
- 1999-01-13 US US09/582,926 patent/US6740634B1/en not_active Expired - Fee Related
- 1999-01-13 NZ NZ505651A patent/NZ505651A/en unknown
- 1999-01-13 CN CNB998021148A patent/CN1199686C/zh not_active Expired - Fee Related
- 1999-01-13 PL PL99341733A patent/PL341733A1/xx unknown
- 1999-01-13 KR KR1020007007533A patent/KR100577877B1/ko not_active IP Right Cessation
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2000
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- 2000-07-14 OA OA1200000208A patent/OA11446A/en unknown
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2004
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WO1999036099A8 (fr) | 1999-11-18 |
PL341733A1 (en) | 2001-05-07 |
CA2316273A1 (en) | 1999-07-22 |
AU1889799A (en) | 1999-08-02 |
CN1288387A (zh) | 2001-03-21 |
HUP0100221A3 (en) | 2002-11-28 |
WO1999036099A1 (fr) | 1999-07-22 |
US20050025826A1 (en) | 2005-02-03 |
NZ505651A (en) | 2003-08-29 |
EP1048301A4 (en) | 2005-03-09 |
AU758596B2 (en) | 2003-03-27 |
IS5560A (is) | 2000-07-11 |
RU2230550C2 (ru) | 2004-06-20 |
KR20010033949A (ko) | 2001-04-25 |
NO20003530D0 (no) | 2000-07-07 |
CN1199686C (zh) | 2005-05-04 |
OA11446A (en) | 2004-04-30 |
SK10272000A3 (sk) | 2001-01-18 |
US6740634B1 (en) | 2004-05-25 |
IL136951A0 (en) | 2001-06-14 |
HRP20000471A2 (en) | 2000-12-31 |
EP1048301A1 (en) | 2000-11-02 |
US7388032B2 (en) | 2008-06-17 |
KR100577877B1 (ko) | 2006-05-09 |
NO20003530L (no) | 2000-09-14 |
TR200002059T2 (tr) | 2001-01-22 |
HUP0100221A2 (hu) | 2001-06-28 |
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