TR200002059T2 - Devamlı salınan bileşim, üretim yöntemi ve kullanımı. - Google Patents
Devamlı salınan bileşim, üretim yöntemi ve kullanımı.Info
- Publication number
- TR200002059T2 TR200002059T2 TR2000/02059T TR200002059T TR200002059T2 TR 200002059 T2 TR200002059 T2 TR 200002059T2 TR 2000/02059 T TR2000/02059 T TR 2000/02059T TR 200002059 T TR200002059 T TR 200002059T TR 200002059 T2 TR200002059 T2 TR 200002059T2
- Authority
- TR
- Turkey
- Prior art keywords
- release composition
- production method
- continuous release
- sustained release
- composition
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/24—Follicle-stimulating hormone [FSH]; Chorionic gonadotropins, e.g. HCG; Luteinising hormone [LH]; Thyroid-stimulating hormone [TSH]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
- A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Organic Chemistry (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Gastroenterology & Hepatology (AREA)
- Inorganic Chemistry (AREA)
- Zoology (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Abstract
Biyolojik olarak aktif bir maddenin bir hidroksinaftoik asit tuzunu ve bakterilerle ayrisabilen bir polimeri içeren, devamli salinan bir bilesim, bunun bir üretim yöntemi ve sözkonusu devamli salinan bilesimi içeren bir farmasötik bilesim.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP641298 | 1998-01-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200002059T2 true TR200002059T2 (tr) | 2001-01-22 |
Family
ID=11637664
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2000/02059T TR200002059T2 (tr) | 1998-01-16 | 1999-01-13 | Devamlı salınan bileşim, üretim yöntemi ve kullanımı. |
Country Status (19)
Country | Link |
---|---|
US (2) | US6740634B1 (tr) |
EP (1) | EP1048301A4 (tr) |
KR (1) | KR100577877B1 (tr) |
CN (1) | CN1199686C (tr) |
AU (1) | AU758596B2 (tr) |
BR (1) | BR9906903A (tr) |
CA (1) | CA2316273A1 (tr) |
HR (1) | HRP20000471A2 (tr) |
HU (1) | HUP0100221A3 (tr) |
IL (1) | IL136951A0 (tr) |
IS (1) | IS5560A (tr) |
NO (1) | NO20003530L (tr) |
NZ (1) | NZ505651A (tr) |
OA (1) | OA11446A (tr) |
PL (1) | PL341733A1 (tr) |
RU (1) | RU2230550C2 (tr) |
SK (1) | SK10272000A3 (tr) |
TR (1) | TR200002059T2 (tr) |
WO (1) | WO1999036099A1 (tr) |
Families Citing this family (120)
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1999
- 1999-01-13 RU RU2000121545/15A patent/RU2230550C2/ru not_active IP Right Cessation
- 1999-01-13 BR BR9906903-2A patent/BR9906903A/pt not_active IP Right Cessation
- 1999-01-13 CA CA002316273A patent/CA2316273A1/en not_active Abandoned
- 1999-01-13 SK SK1027-2000A patent/SK10272000A3/sk unknown
- 1999-01-13 IL IL13695199A patent/IL136951A0/xx not_active IP Right Cessation
- 1999-01-13 EP EP99900300A patent/EP1048301A4/en not_active Withdrawn
- 1999-01-13 TR TR2000/02059T patent/TR200002059T2/tr unknown
- 1999-01-13 HU HU0100221A patent/HUP0100221A3/hu unknown
- 1999-01-13 AU AU18897/99A patent/AU758596B2/en not_active Ceased
- 1999-01-13 WO PCT/JP1999/000086 patent/WO1999036099A1/ja not_active Application Discontinuation
- 1999-01-13 US US09/582,926 patent/US6740634B1/en not_active Expired - Fee Related
- 1999-01-13 NZ NZ505651A patent/NZ505651A/en unknown
- 1999-01-13 CN CNB998021148A patent/CN1199686C/zh not_active Expired - Fee Related
- 1999-01-13 PL PL99341733A patent/PL341733A1/xx unknown
- 1999-01-13 KR KR1020007007533A patent/KR100577877B1/ko not_active IP Right Cessation
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2000
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- 2000-07-11 IS IS5560A patent/IS5560A/is unknown
- 2000-07-13 HR HR20000471A patent/HRP20000471A2/hr not_active Application Discontinuation
- 2000-07-14 OA OA1200000208A patent/OA11446A/en unknown
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2004
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Publication number | Publication date |
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WO1999036099A8 (fr) | 1999-11-18 |
PL341733A1 (en) | 2001-05-07 |
CA2316273A1 (en) | 1999-07-22 |
AU1889799A (en) | 1999-08-02 |
CN1288387A (zh) | 2001-03-21 |
HUP0100221A3 (en) | 2002-11-28 |
WO1999036099A1 (fr) | 1999-07-22 |
US20050025826A1 (en) | 2005-02-03 |
NZ505651A (en) | 2003-08-29 |
EP1048301A4 (en) | 2005-03-09 |
AU758596B2 (en) | 2003-03-27 |
BR9906903A (pt) | 2000-12-12 |
IS5560A (is) | 2000-07-11 |
RU2230550C2 (ru) | 2004-06-20 |
KR20010033949A (ko) | 2001-04-25 |
NO20003530D0 (no) | 2000-07-07 |
CN1199686C (zh) | 2005-05-04 |
OA11446A (en) | 2004-04-30 |
SK10272000A3 (sk) | 2001-01-18 |
US6740634B1 (en) | 2004-05-25 |
IL136951A0 (en) | 2001-06-14 |
HRP20000471A2 (en) | 2000-12-31 |
EP1048301A1 (en) | 2000-11-02 |
US7388032B2 (en) | 2008-06-17 |
KR100577877B1 (ko) | 2006-05-09 |
NO20003530L (no) | 2000-09-14 |
HUP0100221A2 (hu) | 2001-06-28 |
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