BR112021026899A2 - Compostos heterocíclicos - Google Patents
Compostos heterocíclicosInfo
- Publication number
- BR112021026899A2 BR112021026899A2 BR112021026899A BR112021026899A BR112021026899A2 BR 112021026899 A2 BR112021026899 A2 BR 112021026899A2 BR 112021026899 A BR112021026899 A BR 112021026899A BR 112021026899 A BR112021026899 A BR 112021026899A BR 112021026899 A2 BR112021026899 A2 BR 112021026899A2
- Authority
- BR
- Brazil
- Prior art keywords
- compounds
- heterocyclic compounds
- heterocyclic
- processes
- making
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Abstract
compostos heterocíclicos. a presente invenção refere-se a novos compostos heterocíclicos possuindo a fórmula geral (i), em que r1, r2, x, e y são como definidos neste documento, composições incluindo os compostos, processos de fabricação dos compostos e métodos de uso dos compostos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP19185088 | 2019-07-09 | ||
PCT/EP2020/069074 WO2021005034A1 (en) | 2019-07-09 | 2020-07-07 | New heterocyclic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112021026899A2 true BR112021026899A2 (pt) | 2022-05-10 |
Family
ID=67220669
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112021026899A BR112021026899A2 (pt) | 2019-07-09 | 2020-07-07 | Compostos heterocíclicos |
Country Status (18)
Country | Link |
---|---|
US (1) | US20220242876A1 (pt) |
EP (1) | EP3997096A1 (pt) |
JP (1) | JP2022539604A (pt) |
KR (1) | KR20220034104A (pt) |
CN (1) | CN114096545A (pt) |
AR (1) | AR119376A1 (pt) |
AU (1) | AU2020311584A1 (pt) |
BR (1) | BR112021026899A2 (pt) |
CA (1) | CA3145338A1 (pt) |
CL (1) | CL2022000019A1 (pt) |
CO (1) | CO2022000186A2 (pt) |
CR (1) | CR20220004A (pt) |
IL (1) | IL288987A (pt) |
MX (1) | MX2022000243A (pt) |
PE (1) | PE20220515A1 (pt) |
TW (1) | TW202116781A (pt) |
WO (1) | WO2021005034A1 (pt) |
ZA (1) | ZA202110352B (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2019134985A1 (en) | 2018-01-08 | 2019-07-11 | F. Hoffmann-La Roche Ag | Octahydropyrido[1,2-alpha]pyrazines as magl inhibitors |
EP3837263A1 (en) | 2018-08-13 | 2021-06-23 | F. Hoffmann-La Roche AG | New heterocyclic compounds as monoacylglycerol lipase inhibitors |
EP4028403B1 (en) | 2019-09-12 | 2023-11-22 | F. Hoffmann-La Roche AG | 4,4a,5,7,8,8a-hexapyrido[4,3-b][1,4]oxazin-3-one compounds as magl inhibitors |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2014110401A (ru) * | 2011-08-19 | 2015-09-27 | Мерк Шарп И Доум Корп. | Ингибиторы внешнего медуллярного калиевого канала почек |
EP2934533B1 (en) * | 2012-12-19 | 2017-11-15 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
US10323038B2 (en) * | 2015-11-20 | 2019-06-18 | Abide Therapeutics, Inc. | Pyrazole compounds and methods of making and using same |
BR112019014099A2 (pt) * | 2017-01-23 | 2020-02-11 | Pfizer Inc. | Compostos espiro-heterocíclico como inibidores de magl |
JOP20190267A1 (ar) * | 2017-05-23 | 2019-11-18 | Lundbeck La Jolla Research Center Inc | مثبطات بيرازول magl |
-
2020
- 2020-07-07 CA CA3145338A patent/CA3145338A1/en active Pending
- 2020-07-07 BR BR112021026899A patent/BR112021026899A2/pt unknown
- 2020-07-07 JP JP2022500908A patent/JP2022539604A/ja active Pending
- 2020-07-07 CN CN202080050165.3A patent/CN114096545A/zh active Pending
- 2020-07-07 AU AU2020311584A patent/AU2020311584A1/en active Pending
- 2020-07-07 KR KR1020227000611A patent/KR20220034104A/ko active Search and Examination
- 2020-07-07 MX MX2022000243A patent/MX2022000243A/es unknown
- 2020-07-07 EP EP20740259.5A patent/EP3997096A1/en active Pending
- 2020-07-07 CR CR20220004A patent/CR20220004A/es unknown
- 2020-07-07 PE PE2021002265A patent/PE20220515A1/es unknown
- 2020-07-07 WO PCT/EP2020/069074 patent/WO2021005034A1/en unknown
- 2020-07-08 AR ARP200101928A patent/AR119376A1/es unknown
- 2020-07-08 TW TW109123050A patent/TW202116781A/zh unknown
-
2021
- 2021-12-13 ZA ZA2021/10352A patent/ZA202110352B/en unknown
- 2021-12-14 IL IL288987A patent/IL288987A/en unknown
-
2022
- 2022-01-04 CL CL2022000019A patent/CL2022000019A1/es unknown
- 2022-01-06 US US17/569,749 patent/US20220242876A1/en active Pending
- 2022-01-13 CO CONC2022/0000186A patent/CO2022000186A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
CR20220004A (es) | 2022-01-31 |
CN114096545A (zh) | 2022-02-25 |
JP2022539604A (ja) | 2022-09-12 |
AU2020311584A1 (en) | 2022-01-20 |
MX2022000243A (es) | 2022-02-03 |
EP3997096A1 (en) | 2022-05-18 |
KR20220034104A (ko) | 2022-03-17 |
PE20220515A1 (es) | 2022-04-07 |
IL288987A (en) | 2022-02-01 |
TW202116781A (zh) | 2021-05-01 |
AR119376A1 (es) | 2021-12-15 |
CO2022000186A2 (es) | 2022-01-17 |
US20220242876A1 (en) | 2022-08-04 |
WO2021005034A1 (en) | 2021-01-14 |
ZA202110352B (en) | 2022-08-31 |
CL2022000019A1 (es) | 2022-10-21 |
CA3145338A1 (en) | 2021-01-14 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CL2021001330A1 (es) | Nuevos compuestos heterocíclicos | |
CO2021002382A2 (es) | Nuevos compuestos heterocíclicos como inhibidores de la monoacilglicerol lipasa | |
BR112019006571A2 (pt) | derivados de éter de isoxazolila como gaba a alfa5 pam | |
BR112021026899A2 (pt) | Compostos heterocíclicos | |
CO2019009373A2 (es) | Compuestos heterocíclicos útiles como inhibidores duales de atx/ca. | |
CL2020002423A1 (es) | Nuevos compuestos heterocíclicos | |
BR112015022804A2 (pt) | novos derivados de octahidro-pirrol [3,4-c]-pirrol e seus análogos como inibidores de autotaxina | |
BR112018006080A2 (pt) | novos compostos bicíclicos como inibidores de dupla ação de atx/ca | |
BR112018006034A2 (pt) | compostos bicíclicos como inibidores de atx | |
BR112022003982A2 (pt) | Compostos heterocíclicos | |
BR112015004111A2 (pt) | novos derivados bicíclicos | |
BR112014010644A2 (pt) | novos derivados de aril-quinolina | |
BR112013018732A2 (pt) | novos derivados de amida de aril-benzocicloalquila | |
BR112017026682A2 (pt) | novos compostos bicíclicos como inibidores de dupla ação de atx/ca | |
CO2022002000A2 (es) | Nuevos inhibidores heterocíclicos de monoacilglicerol lipasa (magl) | |
BR112022002375A2 (pt) | Compostos de 4,4a,5,7,8,8a-hexapirido[4,3-b][1,4]oxazin-3-ona como inibidores de magl | |
UY36473A (es) | Composiciones con efecto inhibidor de la ureasa mejorado que comprenden triamida del ácido (tio)fosfórico y otros compuestos, tales como aminas y colorantes | |
BR112022003704A2 (pt) | Compostos de 4,4a,5,7,8,8a-hexapirido[4,3-b][1,4]oxazin-3-ona como inibidores de magl | |
BR112016002638A2 (pt) | novos aza-oxo-indóis para o tratamento e profilaxia de infecção pelo virus sincicial respiratório | |
BR112022003357A2 (pt) | Compostos heterocíclicos | |
BR112023003580A2 (pt) | Compostos heterocíclicos | |
BR112015024109A2 (pt) | derivados de ureia e seu uso como inibidores de proteína de ligação de ácidos graxos (fabp) | |
BR112022018828A2 (pt) | Derivados de benzodiazepina como gaba a gamma1 pams | |
UY38941A (es) | Nuevas sulfiliminas o sulfoximinas que contienen compuestos heterocíclicos fungicidas | |
BR112023023527A2 (pt) | Inibidores de nlrp3 |