BR112017004613A2 - processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina - Google Patents

processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina

Info

Publication number
BR112017004613A2
BR112017004613A2 BR112017004613A BR112017004613A BR112017004613A2 BR 112017004613 A2 BR112017004613 A2 BR 112017004613A2 BR 112017004613 A BR112017004613 A BR 112017004613A BR 112017004613 A BR112017004613 A BR 112017004613A BR 112017004613 A2 BR112017004613 A2 BR 112017004613A2
Authority
BR
Brazil
Prior art keywords
pyrazol
chloro
pyridine
preparation
pyridin
Prior art date
Application number
BR112017004613A
Other languages
English (en)
Inventor
Lorsbach Beth
Yang Qiang
Li Xiaoyong
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of BR112017004613A2 publication Critical patent/BR112017004613A2/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

a presente invenção refere-se ao campo de preparação de 3-(3-cloro-1h)-pirazol-1-il)piridina e intermediários do mesmo. estes intermediários são úteis na preparação de determinados (3-halo-1-(piridin-3-il)-1h-pirazol-4-il)amidas e carbamatos e seu uso como pesticidas. é fornecido aqui um processo alternativo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina (5b) por ciclização de dicloridrato de 3-hidrazino piridina com um alquilmetacrilato para fornecer 4-metil-1-(piridin-3-il)pirazolidin-3-ona (1), por cloração de (1) para fornecer 3-(3-cloro-4-metil-4,5-di-hidro-1h-pirazol-1-il)piridina (2), por oxidação de (2) para fornecer 3-(3-cloro-4-metil-1h-pirazol-1-il)piridina (3), também por oxidação de (3) para fornecer ácido 3-cloro-1-(piridin-3-il)-1h-pirazol-4-carboxílico (4), e por descarboxilação de (4) para fornecer 3-(3-cloro-1h-pirazol-1-il)piridina (5b).
BR112017004613A 2014-09-12 2014-10-17 processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina BR112017004613A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462049537P 2014-09-12 2014-09-12
PCT/US2014/061030 WO2016039781A1 (en) 2014-09-12 2014-10-17 Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine

Publications (1)

Publication Number Publication Date
BR112017004613A2 true BR112017004613A2 (pt) 2017-12-05

Family

ID=53540075

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112017004613A BR112017004613A2 (pt) 2014-09-12 2014-10-17 processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina

Country Status (11)

Country Link
US (6) US9085552B1 (pt)
EP (1) EP3191455A4 (pt)
JP (1) JP2017528469A (pt)
KR (1) KR20170058388A (pt)
CN (1) CN107074775A (pt)
AR (1) AR098113A1 (pt)
BR (1) BR112017004613A2 (pt)
CA (1) CA2960985A1 (pt)
IL (1) IL250984A0 (pt)
TW (1) TW201613893A (pt)
WO (1) WO2016039781A1 (pt)

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Publication number Priority date Publication date Assignee Title
CA2925914A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
BR112016008070B8 (pt) 2013-10-17 2022-08-23 Dow Agrosciences Llc Compostos pesticidas, e seus processos de preparação
CA2925952A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
CN105636443A (zh) 2013-10-17 2016-06-01 美国陶氏益农公司 制备杀虫化合物的方法
JP2016539092A (ja) 2013-10-17 2016-12-15 ダウ アグロサイエンシィズ エルエルシー 有害生物防除性化合物の製造方法
WO2015058021A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
WO2015058026A1 (en) 2013-10-17 2015-04-23 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
US9249122B1 (en) 2014-07-31 2016-02-02 Dow Agrosciences Llc Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine
KR20170038785A (ko) 2014-07-31 2017-04-07 다우 아그로사이언시즈 엘엘씨 3-(3-클로로-1h-피라졸-1-일)피리딘의 제조 방법
JP2017523168A (ja) 2014-07-31 2017-08-17 ダウ アグロサイエンシィズ エルエルシー ３−（３−クロロ−１ｈ−ピラゾール−１−イル）ピリジンの製造方法
JP2017525703A (ja) 2014-08-19 2017-09-07 ダウ アグロサイエンシィズ エルエルシー ３−（３−クロロ−１ｈ−ピラゾール−１−イル）ピリジンの調製方法
BR112017004613A2 (pt) 2014-09-12 2017-12-05 Dow Agrosciences Llc processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina
CN110325036B (zh) 2016-12-29 2021-10-26 美国陶氏益农公司 用于制备杀虫化合物的方法
JP2020503336A (ja) * 2016-12-29 2020-01-30 ダウ アグロサイエンシィズ エルエルシー 殺有害生物化合物の調製方法

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