BR0014214A - Imidazoquinolinas substituìdas com amida - Google Patents

Imidazoquinolinas substituìdas com amida

Info

Publication number
BR0014214A
BR0014214A BR0014214-0A BR0014214A BR0014214A BR 0014214 A BR0014214 A BR 0014214A BR 0014214 A BR0014214 A BR 0014214A BR 0014214 A BR0014214 A BR 0014214A
Authority
BR
Brazil
Prior art keywords
amide substituted
useful
compounds
substituted imidazoquinolines
amide
Prior art date
Application number
BR0014214-0A
Other languages
English (en)
Inventor
Stephen L Crooks
Bryon A Merrill
Michael J Rice
Original Assignee
3M Innovative Properties Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 3M Innovative Properties Co filed Critical 3M Innovative Properties Co
Publication of BR0014214A publication Critical patent/BR0014214A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

"IMIDAZOQUINOLINAS SUBSTITUìDAS COM AMIDA". Compostos de imidazoquinolina e tetrahidroimidazoquinolina que contêm funcionalidade uréia, tiouréia, aciluréia ou sulfoniluréia na posição 1 são úteis como modificadores da resposta imunológica. Os compostos e composições da invenção podem induzir a biossíntese de várias citocinas e são úteis no tratamento de uma variedade de condições que incluem doenças virais e doenças neoplásticas.
BR0014214-0A 1999-06-10 2000-06-08 Imidazoquinolinas substituìdas com amida BR0014214A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US13836599P 1999-06-10 1999-06-10
US09/589,236 US6541485B1 (en) 1999-06-10 2000-06-07 Urea substituted imidazoquinolines
PCT/US2000/015656 WO2000076518A1 (en) 1999-06-10 2000-06-08 Urea substituted imidazoquinolines

Publications (1)

Publication Number Publication Date
BR0014214A true BR0014214A (pt) 2004-09-08

Family

ID=26836140

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0014214-0A BR0014214A (pt) 1999-06-10 2000-06-08 Imidazoquinolinas substituìdas com amida

Country Status (26)

Country Link
US (2) US6541485B1 (pt)
EP (1) EP1198232B1 (pt)
JP (1) JP2003501473A (pt)
KR (1) KR20020008223A (pt)
CN (1) CN1181070C (pt)
AT (1) ATE337007T1 (pt)
AU (1) AU766565B2 (pt)
BR (1) BR0014214A (pt)
CA (1) CA2376296A1 (pt)
DE (1) DE60030293T2 (pt)
DK (1) DK1198232T3 (pt)
EE (1) EE05065B1 (pt)
ES (1) ES2270839T3 (pt)
HK (1) HK1047224A1 (pt)
HR (1) HRP20010889A2 (pt)
HU (1) HUP0201664A2 (pt)
IL (1) IL146572A0 (pt)
MX (1) MXPA01012598A (pt)
NO (1) NO320853B1 (pt)
NZ (1) NZ515968A (pt)
PL (1) PL352257A1 (pt)
PT (1) PT1198232E (pt)
RU (1) RU2265020C2 (pt)
SK (1) SK17972001A3 (pt)
TR (1) TR200103576T2 (pt)
WO (1) WO2000076518A1 (pt)

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