BG37527A3 - Method for preparing 1- etoxycarbonyloxyethylic esters of 6- (d- (-)- alpha- amino- alpha- phenylacetamido) penicillanic acid - Google Patents

Method for preparing 1- etoxycarbonyloxyethylic esters of 6- (d- (-)- alpha- amino- alpha- phenylacetamido) penicillanic acid

Info

Publication number: BG37527A3
Authority: BG; Bulgaria
Prior art keywords: alpha; phenylacetamido; preparing; etoxycarbonyloxyethylic; esters
Prior art date: 1982-06-29

Application number

BG061516A

Other languages

Bulgarian (bg)

English (en)

Inventor

Luigi Ratti

Derek Palmer

Robert Tyson

Original Assignee

Astra Laekemedel Aktiebolag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-06-29

Filing date

1983-06-28

Publication date

1985-06-14

1982-06-29 Priority claimed from IT22141/82A external-priority patent/IT1190897B/it

1983-01-07 Priority claimed from GB838300331A external-priority patent/GB8300331D0/en

1983-06-28 Application filed by Astra Laekemedel Aktiebolag filed Critical Astra Laekemedel Aktiebolag

1985-06-14 Publication of BG37527A3 publication Critical patent/BG37527A3/xx

Links

-1 d- (-)- alpha- amino- alpha- phenylacetamido Chemical group 0.000 title abstract 2
150000002148 esters Chemical class 0.000 title 1
RBKMMJSQKNKNEV-RITPCOANSA-N penicillanic acid Chemical compound OC(=O)[C@H]1C(C)(C)S[C@@H]2CC(=O)N21 RBKMMJSQKNKNEV-RITPCOANSA-N 0.000 title 1
239000002253 acid Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C68/00—Preparation of esters of carbonic or haloformic acids
- C07C68/02—Preparation of esters of carbonic or haloformic acids from phosgene or haloformates
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/96—Esters of carbonic or haloformic acids
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Plural Heterocyclic Compounds (AREA)

BG061516A 1982-06-29 1983-06-28 Method for preparing 1- etoxycarbonyloxyethylic esters of 6- (d- (-)- alpha- amino- alpha- phenylacetamido) penicillanic acid BG37527A3 (en)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
IT22141/82A IT1190897B (it)	1982-06-29	1982-06-29	Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
GB8226751		1982-09-20
GB8228622		1982-10-06
GB8232629		1982-11-16
GB838300331A GB8300331D0 (en)	1983-01-07	1983-01-07	Preparation of bromo carbonates

Publications (1)

Publication Number	Publication Date
BG37527A3 true BG37527A3 (en)	1985-06-14

Family

ID=27516485

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
BG061516A BG37527A3 (en)	1982-06-29	1983-06-28	Method for preparing 1- etoxycarbonyloxyethylic esters of 6- (d- (-)- alpha- amino- alpha- phenylacetamido) penicillanic acid
BG068053A BG38336A3 (en)	1982-06-29	1983-06-28	Method for preparing 1- etoxycarbonyloxyethylic ester of 6- (d (-)- alpha- amino- alpha- phenylacetate- amino)- penicillanic acid
BG068052A BG38335A3 (en)	1982-06-29	1983-06-28	Method for preparing 1- etoxycarbonyloxyethylic ester of penicillin g

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
BG068053A BG38336A3 (en)	1982-06-29	1983-06-28	Method for preparing 1- etoxycarbonyloxyethylic ester of 6- (d (-)- alpha- amino- alpha- phenylacetate- amino)- penicillanic acid
BG068052A BG38335A3 (en)	1982-06-29	1983-06-28	Method for preparing 1- etoxycarbonyloxyethylic ester of penicillin g

Country Status (23)

Country	Link
JP (2)	JPH0730082B2 (fi)
AT (1)	AT383128B (fi)
AU (1)	AU566803B2 (fi)
BG (3)	BG37527A3 (fi)
CH (2)	CH657620B (fi)
CY (2)	CY1520A (fi)
DD (1)	DD211561A5 (fi)
DE (2)	DE3322783A1 (fi)
DK (3)	DK160039C (fi)
FI (1)	FI79115C (fi)
FR (1)	FR2543957B1 (fi)
GB (3)	GB2168050A (fi)
GR (1)	GR78585B (fi)
HU (1)	HU191534B (fi)
IE (1)	IE56712B1 (fi)
IL (1)	IL68992A (fi)
IS (1)	IS1361B6 (fi)
NL (1)	NL194081C (fi)
NO (3)	NO157696C (fi)
NZ (1)	NZ204736A (fi)
PT (1)	PT76944B (fi)
SE (2)	SE454879B (fi)
YU (2)	YU43926B (fi)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2573756B1 (fr) *	1984-11-23	1987-01-16	Poudres & Explosifs Ste Nale	Procede de preparation des carbonates de bromo-1 ethyle et d'hydrocarbyle et nouveaux carbonates de bromo-1 ethyle et d'hydrocarbyle

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH516593A (de) *	1967-09-29	1971-12-15	Leo Pharm Prod Ltd	Verfahren zur Herstellung von neuen Estern von a-Aminobenzyl-penicillin
US3873521A (en) *	1970-09-17	1975-03-25	Astra Laekemedel Ab	Esters of {60 -amino penicillins
IE35648B1 (en) *	1970-09-25	1976-04-14	Beecham Group Ltd	Penicillins
DE2161420A1 (de) *	1970-12-30	1972-07-27	Toyama Chemical Co. Ltd., Tokio	Penicillinderivate und Verfahren zu deren Herstellung
DE2228670A1 (de) *	1971-06-15	1973-01-11	Yamanouchi Pharma Co Ltd	Neue oxymethylesterderivate von penicillin und cephalosporin
NZ169577A (en) *	1972-02-15	1984-09-28	Ayerst Mckenna & Harrison	Preparation of lh-and fsh-releasing hormone,intermediates,and pharmaceutical compositions
GB1426717A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
GB1426869A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
GB1425571A (en) *	1972-03-13	1976-02-18	Astra Laekemedel Ab	Penicillins and cephaosporins
SE397981B (sv) *	1973-02-19	1977-11-28	Astra Laekemedel Ab	Nya tetraalkylammoniumsalter av 6-aminopenicillansyra och av bensylpenicillin avsedda att anvendas som mellanprodukter vid framstellning av vissa estrar av 6-aminopenicillansyra och av bensylpenicillin
GB1565656A (en) *	1975-12-13	1980-04-23	Beecham Group Ltd	Preparation of substituted penicillin acid esters
GB1598568A (en) *	1977-04-19	1981-09-23	Glaxo Lab Ltd	Esters of(6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl)-2-methoxyiminoacetamido)-ceph-3-em-4-carboxylic acid
JPS5444694A (en) *	1977-09-06	1979-04-09	Kou Kamata	Aminobenzylpenicillin derivative
GB2123414B (en) *	1982-06-30	1985-12-04	Glaxo Group Ltd	Cephalosporin antibiotics
ATE43833T1 (de) *	1982-11-04	1989-06-15	Astra Laekemedel Ab	Verfahren zur herstellung des 1'ethoxycarbonyloxyethylestersvon benzylpenicillin.

1983
- 1983-06-15 SE SE8303414A patent/SE454879B/sv not_active IP Right Cessation
- 1983-06-15 IL IL68992A patent/IL68992A/xx not_active IP Right Cessation
- 1983-06-20 IE IE1445/83A patent/IE56712B1/en not_active IP Right Cessation
- 1983-06-24 DE DE3322783A patent/DE3322783A1/de active Granted
- 1983-06-24 DE DE3348299A patent/DE3348299C2/de not_active Expired - Lifetime
- 1983-06-27 GB GB08528958A patent/GB2168050A/en not_active Withdrawn
- 1983-06-28 NL NL8302286A patent/NL194081C/nl not_active IP Right Cessation
- 1983-06-28 AU AU16328/83A patent/AU566803B2/en not_active Expired
- 1983-06-28 HU HU832325A patent/HU191534B/hu unknown
- 1983-06-28 FI FI832363A patent/FI79115C/fi not_active IP Right Cessation
- 1983-06-28 BG BG061516A patent/BG37527A3/xx unknown
- 1983-06-28 CH CH527585A patent/CH657620B/de not_active IP Right Cessation
- 1983-06-28 GR GR71790A patent/GR78585B/el unknown
- 1983-06-28 NZ NZ204736A patent/NZ204736A/en unknown
- 1983-06-28 PT PT76944A patent/PT76944B/pt unknown
- 1983-06-28 BG BG068053A patent/BG38336A3/xx unknown
- 1983-06-28 CH CH3540/83A patent/CH656377A5/de not_active IP Right Cessation
- 1983-06-28 BG BG068052A patent/BG38335A3/xx unknown
- 1983-06-28 DK DK296683A patent/DK160039C/da not_active IP Right Cessation
- 1983-06-28 NO NO832351A patent/NO157696C/no not_active IP Right Cessation
- 1983-06-29 IS IS2825A patent/IS1361B6/is unknown
- 1983-06-29 AT AT0238483A patent/AT383128B/de not_active IP Right Cessation
- 1983-06-29 YU YU1415/83A patent/YU43926B/xx unknown
- 1983-06-29 DD DD83252531A patent/DD211561A5/de unknown
- 1983-12-30 FR FR8321138A patent/FR2543957B1/fr not_active Expired
1985
- 1985-03-28 NO NO851254A patent/NO851254L/no unknown
- 1985-03-28 NO NO851255A patent/NO851255L/no unknown
- 1985-09-16 GB GB08522826A patent/GB2168699B/en not_active Expired
- 1985-09-16 GB GB08522827A patent/GB2169287B/en not_active Expired
1986
- 1986-02-14 YU YU218/86A patent/YU43693B/xx unknown
1990
- 1990-04-30 DK DK106090A patent/DK167807B1/da not_active IP Right Cessation
- 1990-04-30 DK DK105990A patent/DK159821C/da not_active IP Right Cessation
- 1990-11-16 CY CY1520A patent/CY1520A/xx unknown
- 1990-11-16 CY CY1519A patent/CY1519A/xx unknown
1991
- 1991-02-26 SE SE9100548A patent/SE503843C2/xx not_active IP Right Cessation
- 1991-04-30 JP JP3124441A patent/JPH0730082B2/ja not_active Expired - Lifetime
- 1991-04-30 JP JP3124442A patent/JPH0819052B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
IL68992A (en)	1991-06-10
DK160039B (da)	1991-01-21
DE3322783C2 (fi)	1991-01-31
SE503843C2 (sv)	1996-09-16
NL8302286A (nl)	1984-01-16
DK106090A (da)	1990-04-30
NO832351L (no)	1983-12-30
JPH0819052B2 (ja)	1996-02-28
DD211561A5 (de)	1984-07-18
JPH0717918A (ja)	1995-01-20
DE3348299C2 (fi)	1990-12-20
NO851254L (no)	1983-12-30
PT76944A (en)	1983-07-01
GB2168699B (en)	1987-04-15
FI79115B (fi)	1989-07-31
IS1361B6 (is)	1989-05-25
IS2825A7 (is)	1984-07-08
SE8303414D0 (sv)	1983-06-15
PT76944B (en)	1986-04-09
GB8528958D0 (en)	1986-01-02
YU141583A (en)	1986-06-30
DK159821B (da)	1990-12-10
DK105990D0 (da)	1990-04-30
HU191534B (en)	1987-03-30
GB2169287A (en)	1986-07-09
DK167807B1 (da)	1993-12-20
FR2543957A1 (fr)	1984-10-12
IE831445L (en)	1983-12-29
NL194081B (nl)	2001-02-01
DK296683A (da)	1983-12-30
SE8303414L (sv)	1983-12-30
FI832363L (fi)	1983-12-30
NO851255L (no)	1983-12-30
SE9100548L (sv)	1991-02-26
CY1520A (en)	1990-11-16
FI832363A0 (fi)	1983-06-28
CH656377A5 (de)	1986-06-30
CH657620B (fi)	1986-09-15
SE9100548D0 (sv)	1991-02-26
FR2543957B1 (fr)	1986-10-24
JPH0730082B2 (ja)	1995-04-05
NO157696B (no)	1988-01-25
DK296683D0 (da)	1983-06-28
GB2168050A (en)	1986-06-11
GB8522827D0 (en)	1985-10-23
DE3322783A1 (de)	1984-02-09
YU43693B (en)	1989-10-31
BG38335A3 (en)	1985-11-15
YU21886A (en)	1987-10-31
GB2169287B (en)	1987-04-08
JPH0543583A (ja)	1993-02-23
SE454879B (sv)	1988-06-06
FI79115C (fi)	1989-11-10
NL194081C (nl)	2001-06-05
AU566803B2 (en)	1987-10-29
GB8522826D0 (en)	1985-10-23
AU1632883A (en)	1984-01-05
AT383128B (de)	1987-05-25
NZ204736A (en)	1986-11-12
NO157696C (no)	1988-05-04
DK106090D0 (da)	1990-04-30
DK160039C (da)	1991-06-10
YU43926B (en)	1989-12-31
ATA238483A (de)	1986-10-15
GB2168699A (en)	1986-06-25
IE56712B1 (en)	1991-11-20
DK159821C (da)	1991-04-29
CY1519A (en)	1990-11-16
GR78585B (fi)	1984-09-27
DK105990A (da)	1990-04-30
BG38336A3 (en)	1985-11-15

Publication	Publication Date	Title
BG38639A3 (en)	1986-01-15	Method for preparing ester derivatives of 6- beta- hydroxymethylpenicillanic acid
BG37526A3 (en)	1985-06-14	Method for preparing esters of malonic acid
BG35467A3 (en)	1984-04-15	Method for preparing diesters of methanediol
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BG36787A3 (en)	1985-01-15	Method for preparing monoester salts of phosphoric acid
BG34908A3 (en)	1983-12-15	Method for preparing d- 6- n- propylergolines
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BG28568A3 (bg)	1980-05-15	Метод за получаване на естери на оксаловата киселина
BG41821A3 (en)	1987-08-14	Method for preparing pyridyl derivatives
BG41126A3 (en)	1987-04-15	Method for preparing benzamides
BG35746A3 (en)	1984-06-15	Method for preparing 1- cyclohexenylmethylpyrolidines
BG40650A3 (en)	1986-01-15	Method for preparing ester of treo- 2- hydroxy- 3- (4- metoxyphenyl)- 3- (2- nitrophenylthio)- propionic acid
BG42352A3 (en)	1987-11-14	Method for preparing derivatives of cyclopropane- carbonic acid esters
BG38938A3 (en)	1986-03-14	Method for preparing chlormethylester of penicillanic acid derivatives
BG38939A3 (en)	1986-03-14	Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid
BG30628A3 (en)	1981-07-15	Method for obtaining of 3- exomethelenecefam sulphoxide esters
BG35749A3 (en)	1984-06-15	Method for preparing 20- dihydro- 20, 23- dideoxytilonolide
BG37527A3 (en)	1985-06-14	Method for preparing 1- etoxycarbonyloxyethylic esters of 6- (d- (-)- alpha- amino- alpha- phenylacetamido) penicillanic acid
BG40653A3 (en)	1986-01-15	Method for preparing amidothiocarbamate derivatives of carbon acid
BG39977A3 (en)	1986-09-15	Method for preparing derivatives of furyloxazolylacetic acid
GB2045746B (en)	1983-05-11	6-(azacycloalky-or azabicycloalkyl-methylimino)penicillanic acid esters
BG36345A3 (en)	1984-10-15	Method for preparing cyclopentenic derivatives
BG34460A3 (en)	1983-09-15	Method of obtaining derivatives of 7 beta-amino- thiazolylacetamido-3-cephem-4-carbonic acid
BG36633A3 (en)	1984-12-16	Method for preparing 3- hydroxycephalosporines
BG32857A3 (en)	1982-10-15	Method for obtaining of cephalosporint solvates