AU506340B2 - Benzodiazepine derivatives - Google Patents

Benzodiazepine derivatives

Info

Publication number: AU506340B2
Authority: AU; Australia
Prior art keywords: benzodiazepine derivatives; benzodiazepine; derivatives
Prior art date: 1974-11-26
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

AU86858/75A

Other languages

English (en)

Other versions

AU8685875A (en

Inventor

J. K. and Tupper D. E Chakrabarti

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Lilly Industries Ltd

Original Assignee

Lilly Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1974-11-26

Filing date

1975-11-21

Publication date

1979-12-20

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10459213&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU506340(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1975-11-21 Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd

1977-05-26 Publication of AU8685875A publication Critical patent/AU8685875A/en

1979-12-20 Application granted granted Critical

1979-12-20 Publication of AU506340B2 publication Critical patent/AU506340B2/en

Status Expired legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

AU86858/75A 1974-11-26 1975-11-21 Benzodiazepine derivatives Expired AU506340B2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB51240/74		1974-11-26
GB51240/74A GB1533235A (en)	1974-11-26	1974-11-26	Benzodiazepine derivatives

Publications (2)

Publication Number	Publication Date
AU8685875A AU8685875A (en)	1977-05-26
AU506340B2 true AU506340B2 (en)	1979-12-20

Family

ID=10459213

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU86858/75A Expired AU506340B2 (en)	1974-11-26	1975-11-21	Benzodiazepine derivatives

Country Status (30)

Country	Link
JP (1)	JPS6044314B2 (cs)
AR (1)	AR221203A1 (cs)
AT (1)	AT351547B (cs)
AU (1)	AU506340B2 (cs)
BE (1)	BE835932A (cs)
BG (1)	BG29573A3 (cs)
CA (1)	CA1075687A (cs)
CH (2)	CH613454A5 (cs)
CS (1)	CS236753B2 (cs)
DD (1)	DD123343A5 (cs)
DE (1)	DE2552403C2 (cs)
DK (1)	DK146887C (cs)
ES (1)	ES443011A1 (cs)
FR (1)	FR2292479A1 (cs)
GB (1)	GB1533235A (cs)
HK (1)	HK58681A (cs)
HU (1)	HU172493B (cs)
IE (1)	IE42564B1 (cs)
IL (1)	IL48502A (cs)
KE (1)	KE3163A (cs)
MY (1)	MY8200149A (cs)
NL (1)	NL186088C (cs)
NZ (1)	NZ179335A (cs)
PH (2)	PH11669A (cs)
PL (1)	PL100135B1 (cs)
RO (1)	RO69912A (cs)
SE (2)	SE421209B (cs)
SU (2)	SU629879A3 (cs)
YU (1)	YU298375A (cs)
ZA (1)	ZA757344B (cs)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL62792A (en) *	1980-05-07	1985-02-28	Byk Gulden Lomberg Chem Fab	Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them
GB8819059D0 (en) *	1988-08-11	1988-09-14	Lilly Industries Ltd	Benzodiazepine compounds & their use as pharmaceuticals
GB9009229D0 (en)	1990-04-25	1990-06-20	Lilly Industries Ltd	Pharmaceutical compounds
ES2153373T3 (es) *	1992-05-29	2001-03-01	Lilly Co Eli	Derivados de tienobenzodiazepina para el tratamiento de trastornos del sistema nervioso central.
AU700078B2 (en) *	1995-11-01	1998-12-17	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
US6043358A (en)	1995-11-01	2000-03-28	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
CA2302409A1 (en)	1997-09-02	1999-03-11	Hiroshi Yasumatsu	Condensed thiophene compounds and pharmaceutical use thereof
PL199016B1 (pl) *	2002-06-20	2008-08-29	Adamed Sp Z Oo	Sposób wytwarzania olanzapiny
SI21270A (sl)	2002-07-15	2004-02-29	Krka, Tovarna Zdravil, D.D., Novo Mesto	Kristalne oblike olanzapina in postopki za njihovo pripravo
DE10301923B3 (de) *	2003-01-17	2004-09-16	Krka Tovarna Zdravil, D.D.	Verfahren und Zwischenprodukte zur Herstellung von Olanzapin
AR047460A1 (es) *	2004-01-27	2006-01-18	Synthon Bv	Proceso para la fabricacion de acetato de 2-metil-4-(4-metil-1-piperazinil)-10h-tieno[2,3-b][1,5]benzodiazepina (acetato de olanzapina)
AR048272A1 (es)	2004-03-18	2006-04-12	Lek Pharmaceuticals	Sintesis de 2 metil - 4- (4- metil -1- piperazinil) - 10 h- tieno ( 2,3-b) (1,5) benzodiazepina y sus sales, metodos para su preparacion, composiciones farmaceuticas que la contienen y su uso en la fabricacion de medicamentos para el tratamiento de enfermedades mentales.
CA2565683C (en) *	2004-06-30	2013-04-02	Athersys, Inc.	Substituted azepine derivatives as serotonin receptor modulators
EP2292624A1 (en)	2009-07-20	2011-03-09	LEK Pharmaceuticals d.d.	Process for the purification of olanzapine

1974
- 1974-11-25 SU SU742191705A patent/SU629879A3/ru active
- 1974-11-26 GB GB51240/74A patent/GB1533235A/en not_active Expired
1975
- 1975-11-20 DK DK524175A patent/DK146887C/da active
- 1975-11-20 CA CA240,082A patent/CA1075687A/en not_active Expired
- 1975-11-20 IL IL48502A patent/IL48502A/xx unknown
- 1975-11-21 PH PH17788A patent/PH11669A/en unknown
- 1975-11-21 AU AU86858/75A patent/AU506340B2/en not_active Expired
- 1975-11-22 DE DE2552403A patent/DE2552403C2/de not_active Expired
- 1975-11-24 NZ NZ179335A patent/NZ179335A/xx unknown
- 1975-11-24 SE SE7513185A patent/SE421209B/xx not_active IP Right Cessation
- 1975-11-24 CH CH1517275A patent/CH613454A5/xx not_active IP Right Cessation
- 1975-11-24 CH CH604478A patent/CH613455A5/xx not_active IP Right Cessation
- 1975-11-24 ZA ZA757344A patent/ZA757344B/xx unknown
- 1975-11-25 RO RO7584018A patent/RO69912A/ro unknown
- 1975-11-25 FR FR7535900A patent/FR2292479A1/fr active Granted
- 1975-11-25 YU YU02983/75A patent/YU298375A/xx unknown
- 1975-11-25 AR AR261340A patent/AR221203A1/es active
- 1975-11-25 JP JP50141080A patent/JPS6044314B2/ja not_active Expired
- 1975-11-25 DD DD189666A patent/DD123343A5/xx unknown
- 1975-11-25 BE BE6045266A patent/BE835932A/xx not_active IP Right Cessation
- 1975-11-25 IE IE2565/75A patent/IE42564B1/en unknown
- 1975-11-26 AT AT898275A patent/AT351547B/de not_active IP Right Cessation
- 1975-11-26 HU HU75LI00000284A patent/HU172493B/hu unknown
- 1975-11-26 CS CS757991A patent/CS236753B2/cs unknown
- 1975-11-26 PL PL1975184991A patent/PL100135B1/pl unknown
- 1975-11-26 BG BG031601A patent/BG29573A3/xx unknown
- 1975-11-26 ES ES443011A patent/ES443011A1/es not_active Expired
- 1975-11-26 NL NLAANVRAGE7513833,A patent/NL186088C/xx not_active IP Right Cessation
1976
- 1976-10-07 SU SU762406250A patent/SU626702A3/ru active
1977
- 1977-02-22 PH PH19480A patent/PH24534A/en unknown
1978
- 1978-11-27 SE SE7812194A patent/SE429045B/sv not_active IP Right Cessation
1981
- 1981-09-24 KE KE3163A patent/KE3163A/xx unknown
- 1981-11-26 HK HK586/81A patent/HK58681A/xx unknown
1982
- 1982-12-30 MY MY149/82A patent/MY8200149A/xx unknown

Also Published As

Publication number	Publication date
DE2552403A1 (de)	1976-08-12
AU8685875A (en)	1977-05-26
JPS5176296A (en)	1976-07-01
NL186088B (nl)	1990-04-17
GB1533235A (en)	1978-11-22
ES443011A1 (es)	1977-07-01
BE835932A (fr)	1976-05-25
AR221203A1 (es)	1981-01-15
CH613455A5 (en)	1979-09-28
DE2552403C2 (de)	1986-06-19
DD123343A5 (cs)	1976-12-12
YU298375A (en)	1982-10-31
MY8200149A (en)	1982-12-31
IL48502A (en)	1980-01-31
KE3163A (en)	1981-10-16
PL100135B1 (pl)	1978-09-30
ATA898275A (de)	1979-01-15
RO69912A (ro)	1980-08-15
SU629879A3 (ru)	1978-10-25
SE421209B (sv)	1981-12-07
CH613454A5 (en)	1979-09-28
IE42564B1 (en)	1980-09-10
NZ179335A (en)	1978-11-13
DK524175A (da)	1976-05-27
SE7812194L (sv)	1978-11-27
PH11669A (en)	1978-05-19
BG29573A3 (en)	1980-12-12
SE7513185L (sv)	1976-05-27
IL48502A0 (en)	1976-01-30
FR2292479A1 (fr)	1976-06-25
DK146887C (da)	1984-07-09
CA1075687A (en)	1980-04-15
AT351547B (de)	1979-07-25
CS236753B2 (en)	1985-05-15
SU626702A3 (ru)	1978-09-30
DK146887B (da)	1984-01-30
ZA757344B (en)	1976-11-24
NL186088C (nl)	1990-09-17
JPS6044314B2 (ja)	1985-10-02
IE42564L (en)	1976-05-26
NL7513833A (nl)	1976-05-31
PH24534A (en)	1990-08-03
FR2292479B1 (cs)	1978-07-28
HK58681A (en)	1981-12-04
HU172493B (hu)	1978-09-28
SE429045B (sv)	1983-08-08

Publication	Publication Date	Title
AU500910B2 (en)	1979-06-07	Benzimidazolinone derivatives
AU505998B2 (en)	1979-12-13	Diazepine derivative
AU506340B2 (en)	1979-12-20	Benzodiazepine derivatives
AU498132B2 (en)	1979-02-15	5 - nitro - pyrimidine derivatives
AU470711B2 (en)	1976-03-25	Oxacyclohexane derivatives
AU502405B2 (en)	1979-07-26	Benzodiazepine derivatives
AU501915B2 (en)	1979-07-05	Phenyl-pyridylamine derivatives
AU503060B2 (en)	1979-08-23	Ergopeptine derivatives
AU499054B2 (en)	1979-04-05	Benzodiazepine derivatives
AU472498B2 (en)	1976-05-27	Aminomethylarylmethlpenicillin derivatives
AU500509B2 (en)	1979-05-24	Diazepine derivatives
KE3004A (en)	1979-12-14	Benzodiazepine derivatives
GB1482503A (en)	1977-08-10	Benzodiazepine derivatives
AU490569B2 (en)	1976-11-18	Benzodiazepine derivatives
AU530519B2 (en)	1983-07-21	Diazepine derivatives
AU527906B2 (en)	1983-03-31	Diazepine derivatives
AU471140B2 (en)	1976-04-08	Benzodiazepin derivatives
AU493074B2 (en)	1976-08-26	Thiepino- and oxepino - pyrrole derivatives
AU488080B2 (en)	1976-02-05	Cyclopentate derivatives
AU491184B2 (en)	1977-06-16	Benzenedisulphonamide derivatives
AU475893B2 (en)	1976-09-09	Triazapentadiene derivatives
AU489669B2 (en)	1976-10-28	3-piperazino-isoquinoline derivatives
AU480360B2 (en)	1975-08-21	2-aminomethyl-phenol derivatives
AU488651B2 (en)	1976-03-18	2-cyclopropyl-4-phenylprrolidine derivatives
AU488164B2 (en)	1976-11-04	Pyrimidincl derivatives