AR015940A1 - Derivados de rapamicina que contiene tetrazol con vidas medias acortadas y su uso para la manufactura de un medicamento - Google Patents

Derivados de rapamicina que contiene tetrazol con vidas medias acortadas y su uso para la manufactura de un medicamento

Info

Publication number
AR015940A1
AR015940A1 ARP980104798A ARP980104798A AR015940A1 AR 015940 A1 AR015940 A1 AR 015940A1 AR P980104798 A ARP980104798 A AR P980104798A AR P980104798 A ARP980104798 A AR P980104798A AR 015940 A1 AR015940 A1 AR 015940A1
Authority
AR
Argentina
Prior art keywords
manufacture
tetrazol
lives
medicinal product
derivatives containing
Prior art date
Application number
ARP980104798A
Other languages
English (en)
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25470968&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR015940(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of AR015940A1 publication Critical patent/AR015940A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Análogo de rapamicina que tiene la formula (I) o una sal o prodroga del mismo farmacéuticamente aceptable que es un agente inmunomodulador y esutil en el tratamiento de restenosis, enfermedades inmunes y autoinmunes, e inhibe cáncer, desarrolofungal , y el rechazo a los tejidos de post-transplante;y su uso para la manufactura de un medicamento.
ARP980104798A 1997-09-26 1998-09-25 Derivados de rapamicina que contiene tetrazol con vidas medias acortadas y su uso para la manufactura de un medicamento AR015940A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US93814497A 1997-09-26 1997-09-26

Publications (1)

Publication Number Publication Date
AR015940A1 true AR015940A1 (es) 2001-05-30

Family

ID=25470968

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP980104798A AR015940A1 (es) 1997-09-26 1998-09-25 Derivados de rapamicina que contiene tetrazol con vidas medias acortadas y su uso para la manufactura de un medicamento

Country Status (28)

Country Link
EP (1) EP1015459B9 (es)
JP (1) JP3790424B2 (es)
KR (3) KR100803639B1 (es)
CN (1) CN1161360C (es)
AR (1) AR015940A1 (es)
AT (1) ATE297398T1 (es)
AU (1) AU745576B2 (es)
BG (1) BG64955B1 (es)
BR (1) BR9812305A (es)
CA (1) CA2303934C (es)
CO (1) CO5070656A1 (es)
CZ (1) CZ299365B6 (es)
DE (1) DE69830502T2 (es)
DK (1) DK1015459T3 (es)
ES (1) ES2244087T3 (es)
HK (1) HK1030771A1 (es)
HU (1) HU228368B1 (es)
IL (2) IL134607A0 (es)
NO (1) NO325813B1 (es)
NZ (2) NZ502896A (es)
PL (1) PL191212B1 (es)
PT (1) PT1015459E (es)
SI (1) SI1015459T1 (es)
SK (1) SK285408B6 (es)
TR (1) TR200000778T2 (es)
TW (1) TW557297B (es)
WO (1) WO1999015530A1 (es)
ZA (1) ZA988750B (es)

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Also Published As

Publication number Publication date
BG64955B1 (bg) 2006-10-31
DE69830502D1 (de) 2005-07-14
BR9812305A (pt) 2000-09-05
KR20060071092A (ko) 2006-06-26
EP1015459B1 (en) 2005-06-08
SI1015459T1 (en) 2005-10-31
PL191212B1 (pl) 2006-03-31
CA2303934A1 (en) 1999-04-01
ZA988750B (en) 1999-04-01
TR200000778T2 (tr) 2000-07-21
KR20010024298A (ko) 2001-03-26
HK1030771A1 (en) 2001-05-18
PT1015459E (pt) 2005-09-30
AU745576B2 (en) 2002-03-21
HU228368B1 (en) 2013-03-28
SK4172000A3 (en) 2000-08-14
HUP0004556A2 (hu) 2001-10-28
DK1015459T3 (da) 2005-10-10
HUP0004556A3 (en) 2001-12-28
ES2244087T3 (es) 2005-12-01
CO5070656A1 (es) 2001-08-28
WO1999015530A1 (en) 1999-04-01
DE69830502T2 (de) 2006-05-11
CZ299365B6 (cs) 2008-07-02
PL339455A1 (en) 2000-12-18
KR100803639B1 (ko) 2008-02-19
NO325813B1 (no) 2008-07-21
CA2303934C (en) 2010-01-26
CZ20001014A3 (cs) 2000-07-12
CN1161360C (zh) 2004-08-11
KR100700319B1 (ko) 2007-03-29
NO20001438L (no) 2000-05-26
EP1015459A1 (en) 2000-07-05
SK285408B6 (sk) 2007-01-04
NO20001438D0 (no) 2000-03-20
EP1015459B9 (en) 2005-10-12
ATE297398T1 (de) 2005-06-15
KR100833812B1 (ko) 2008-05-30
JP2001517671A (ja) 2001-10-09
AU9581998A (en) 1999-04-12
JP3790424B2 (ja) 2006-06-28
BG104316A (en) 2000-12-29
CN1271361A (zh) 2000-10-25
KR20070086925A (ko) 2007-08-27
IL134607A0 (en) 2001-04-30
IL134607A (en) 2006-04-10
NZ514778A (en) 2005-01-28
TW557297B (en) 2003-10-11
NZ502896A (en) 2001-12-21

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