ZA983257B - 5-Aryl--3-[8-azabicyclo(3.2.1)oct-3-yl]-1,3,4-oxadiazol-2(3H)-one dericatives their preparation and their therapeutic application - Google Patents

5-Aryl--3-[8-azabicyclo(3.2.1)oct-3-yl]-1,3,4-oxadiazol-2(3H)-one dericatives their preparation and their therapeutic application

Info

Publication number
ZA983257B
ZA983257B ZA983257A ZA983257A ZA983257B ZA 983257 B ZA983257 B ZA 983257B ZA 983257 A ZA983257 A ZA 983257A ZA 983257 A ZA983257 A ZA 983257A ZA 983257 B ZA983257 B ZA 983257B
Authority
ZA
South Africa
Prior art keywords
dericatives
oxadiazol
azabicyclo
oct
aryl
Prior art date
Application number
ZA983257A
Other languages
English (en)
Inventor
Samir Jegham
Alistair Lochead
Frederic Galli
Alain Nedelec
Axelle Samson
Thierry Gallet
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of ZA983257B publication Critical patent/ZA983257B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
ZA983257A 1997-04-18 1998-04-17 5-Aryl--3-[8-azabicyclo(3.2.1)oct-3-yl]-1,3,4-oxadiazol-2(3H)-one dericatives their preparation and their therapeutic application ZA983257B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9704802A FR2762316B1 (fr) 1997-04-18 1997-04-18 Derives de 5-aryl-3-(8-azabicyclo[3.2.1] octan-3-yl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
ZA983257B true ZA983257B (en) 1998-10-19

Family

ID=9506076

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA983257A ZA983257B (en) 1997-04-18 1998-04-17 5-Aryl--3-[8-azabicyclo(3.2.1)oct-3-yl]-1,3,4-oxadiazol-2(3H)-one dericatives their preparation and their therapeutic application

Country Status (32)

Country Link
US (1) US6255319B1 (xx)
EP (1) EP0975631B1 (xx)
JP (1) JP2001521542A (xx)
KR (1) KR20010006452A (xx)
CN (1) CN1260794A (xx)
AR (1) AR012458A1 (xx)
AT (1) ATE206424T1 (xx)
AU (1) AU742666B2 (xx)
BG (1) BG64053B1 (xx)
BR (1) BR9808926A (xx)
CA (1) CA2286106A1 (xx)
CO (1) CO4750656A1 (xx)
CZ (1) CZ289154B6 (xx)
DE (1) DE69801905T2 (xx)
DK (1) DK0975631T3 (xx)
EE (1) EE03769B1 (xx)
ES (1) ES2165162T3 (xx)
FR (1) FR2762316B1 (xx)
HU (1) HUP0002456A3 (xx)
IL (1) IL132352A0 (xx)
NO (1) NO995040L (xx)
NZ (1) NZ500396A (xx)
PL (1) PL186894B1 (xx)
PT (1) PT975631E (xx)
RU (1) RU2186066C2 (xx)
SI (1) SI0975631T1 (xx)
SK (1) SK283441B6 (xx)
TR (1) TR199902600T2 (xx)
TW (1) TW502005B (xx)
UA (1) UA57071C2 (xx)
WO (1) WO1998047898A1 (xx)
ZA (1) ZA983257B (xx)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0211230D0 (en) * 2002-05-16 2002-06-26 Medinnova Sf Treatment of heart failure
EP1610789B1 (en) * 2003-03-26 2010-07-21 Merck Sharp & Dohme Corp. Bicyclic piperidine derivatives as melanocortin-4 receptor agonists
CA2545513C (en) * 2003-11-18 2013-01-08 Boehringer Ingelheim International Gmbh Solid pharmaceutical preparation form
US7737163B2 (en) 2004-06-15 2010-06-15 Pfizer Inc. Benzimidazolone carboxylic acid derivatives
MXPA06014486A (es) 2004-06-15 2007-03-01 Pfizer Derivados de acido carboxilico de bencimidazolona.
SE532388C2 (sv) * 2008-03-14 2010-01-12 Tetra Laval Holdings & Finance Förpackningslaminat och -behållare med två separata gasbarriärskikt samt metod för deras framställning
JP6348568B2 (ja) 2013-03-15 2018-06-27 モンサント テクノロジー エルエルシー 線虫害虫防除のためのｎ−，ｃ−二置換アゾール
GB201814151D0 (en) 2018-08-31 2018-10-17 Ucl Business Plc Compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE182591T1 (de) * 1991-09-12 1999-08-15 Smithkline Beecham Plc 5-ht4 rezeptor antagonisten
PH31171A (en) * 1992-02-04 1998-03-20 Esai Co Ltd Aminobenzonic acid derivatives useful for treatinggastrointestinal conditions.
NZ246915A (en) * 1992-02-06 1996-05-28 Smithkline Beecham Plc Benzopyran, benzothiopyran and benzofuran derivatives, preparation and pharmaceutical compositions thereof
JP3235913B2 (ja) * 1993-07-30 2001-12-04 エーザイ株式会社 アミノ安息香酸誘導体
PL186204B1 (pl) * 1995-11-09 2003-11-28 Sanofi Synthelabo Pochodne 5-fenylo-3-(piperydyn-4-ylo)-1,3,4-oksadiazol-2(3H)-onu do stosowania jako ligandy receptora 5-HT lub H

Also Published As

Publication number Publication date
FR2762316A1 (fr) 1998-10-23
BG103810A (en) 2000-06-30
EE03769B1 (et) 2002-06-17
EE9900487A (et) 2000-06-15
CO4750656A1 (es) 1999-03-31
KR20010006452A (ko) 2001-01-26
SK142699A3 (en) 2000-05-16
EP0975631A1 (fr) 2000-02-02
EP0975631B1 (fr) 2001-10-04
AU742666B2 (en) 2002-01-10
SI0975631T1 (en) 2002-06-30
CZ364199A3 (cs) 2000-03-15
AR012458A1 (es) 2000-10-18
DE69801905T2 (de) 2002-07-04
FR2762316B1 (fr) 1999-12-17
PL186894B1 (pl) 2004-03-31
ATE206424T1 (de) 2001-10-15
SK283441B6 (sk) 2003-07-01
WO1998047898A1 (fr) 1998-10-29
PL336315A1 (en) 2000-06-19
JP2001521542A (ja) 2001-11-06
PT975631E (pt) 2002-03-28
NO995040L (no) 1999-12-16
NZ500396A (en) 2001-04-27
DK0975631T3 (da) 2002-01-28
TW502005B (en) 2002-09-11
BG64053B1 (bg) 2003-11-28
CA2286106A1 (en) 1998-10-29
AU7341598A (en) 1998-11-13
DE69801905D1 (de) 2001-11-08
IL132352A0 (en) 2001-03-19
BR9808926A (pt) 2000-08-01
ES2165162T3 (es) 2002-03-01
US6255319B1 (en) 2001-07-03
HUP0002456A3 (en) 2001-03-28
NO995040D0 (no) 1999-10-15
CZ289154B6 (cs) 2001-11-14
RU2186066C2 (ru) 2002-07-27
CN1260794A (zh) 2000-07-19
UA57071C2 (uk) 2003-06-16
HUP0002456A2 (hu) 2000-12-28
TR199902600T2 (xx) 2000-03-21

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