IL132352A0 - 5-Aryl-3-(8-azabicyclo (3.2.2) oct-3yl) -1,3,4-oxadiazol 22 (3h) - one derivatives as 5-ht4 receptor ligands - Google Patents

5-Aryl-3-(8-azabicyclo (3.2.2) oct-3yl) -1,3,4-oxadiazol 22 (3h) - one derivatives as 5-ht4 receptor ligands

Info

Publication number: IL132352A0
Authority: IL; Israel
Prior art keywords: oxadiazol; azabicyclo; oct; aryl; derivatives
Prior art date: 1997-04-18

Application number

IL13235298A

Other languages

English (en)

Original Assignee

Sanofi Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-04-18

Filing date

1998-04-15

Publication date

2001-03-19

1998-04-15 Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo

2001-03-19 Publication of IL132352A0 publication Critical patent/IL132352A0/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

IL13235298A 1997-04-18 1998-04-15 5-Aryl-3-(8-azabicyclo (3.2.2) oct-3yl) -1,3,4-oxadiazol 22 (3h) - one derivatives as 5-ht4 receptor ligands IL132352A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9704802A FR2762316B1 (fr)	1997-04-18	1997-04-18	Derives de 5-aryl-3-(8-azabicyclo[3.2.1] octan-3-yl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique
PCT/FR1998/000754 WO1998047898A1 (fr)	1997-04-18	1998-04-15	Derives de 5-aryl-3-(8-azabicyclo(3.2.2)oct-3-yl)-1,3,4-oxadiazol-2(3h)-one en tant que ligands des recepteurs 5-ht4

Publications (1)

Publication Number	Publication Date
IL132352A0 true IL132352A0 (en)	2001-03-19

Family

ID=9506076

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL13235298A IL132352A0 (en)	1997-04-18	1998-04-15	5-Aryl-3-(8-azabicyclo (3.2.2) oct-3yl) -1,3,4-oxadiazol 22 (3h) - one derivatives as 5-ht4 receptor ligands

Country Status (32)

Country	Link
US (1)	US6255319B1 (xx)
EP (1)	EP0975631B1 (xx)
JP (1)	JP2001521542A (xx)
KR (1)	KR20010006452A (xx)
CN (1)	CN1260794A (xx)
AR (1)	AR012458A1 (xx)
AT (1)	ATE206424T1 (xx)
AU (1)	AU742666B2 (xx)
BG (1)	BG64053B1 (xx)
BR (1)	BR9808926A (xx)
CA (1)	CA2286106A1 (xx)
CO (1)	CO4750656A1 (xx)
CZ (1)	CZ289154B6 (xx)
DE (1)	DE69801905T2 (xx)
DK (1)	DK0975631T3 (xx)
EE (1)	EE03769B1 (xx)
ES (1)	ES2165162T3 (xx)
FR (1)	FR2762316B1 (xx)
HU (1)	HUP0002456A3 (xx)
IL (1)	IL132352A0 (xx)
NO (1)	NO995040L (xx)
NZ (1)	NZ500396A (xx)
PL (1)	PL186894B1 (xx)
PT (1)	PT975631E (xx)
RU (1)	RU2186066C2 (xx)
SI (1)	SI0975631T1 (xx)
SK (1)	SK283441B6 (xx)
TR (1)	TR199902600T2 (xx)
TW (1)	TW502005B (xx)
UA (1)	UA57071C2 (xx)
WO (1)	WO1998047898A1 (xx)
ZA (1)	ZA983257B (xx)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0211230D0 (en) *	2002-05-16	2002-06-26	Medinnova Sf	Treatment of heart failure
EP1610789B1 (en) *	2003-03-26	2010-07-21	Merck Sharp & Dohme Corp.	Bicyclic piperidine derivatives as melanocortin-4 receptor agonists
CA2545513C (en) *	2003-11-18	2013-01-08	Boehringer Ingelheim International Gmbh	Solid pharmaceutical preparation form
US7737163B2 (en)	2004-06-15	2010-06-15	Pfizer Inc.	Benzimidazolone carboxylic acid derivatives
MXPA06014486A (es)	2004-06-15	2007-03-01	Pfizer	Derivados de acido carboxilico de bencimidazolona.
SE532388C2 (sv) *	2008-03-14	2010-01-12	Tetra Laval Holdings & Finance	Förpackningslaminat och -behållare med två separata gasbarriärskikt samt metod för deras framställning
JP6348568B2 (ja)	2013-03-15	2018-06-27	モンサントテクノロジーエルエルシー	線虫害虫防除のためのｎ−，ｃ−二置換アゾール
GB201814151D0 (en)	2018-08-31	2018-10-17	Ucl Business Plc	Compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ATE182591T1 (de) *	1991-09-12	1999-08-15	Smithkline Beecham Plc	5-ht4 rezeptor antagonisten
PH31171A (en) *	1992-02-04	1998-03-20	Esai Co Ltd	Aminobenzonic acid derivatives useful for treatinggastrointestinal conditions.
NZ246915A (en) *	1992-02-06	1996-05-28	Smithkline Beecham Plc	Benzopyran, benzothiopyran and benzofuran derivatives, preparation and pharmaceutical compositions thereof
JP3235913B2 (ja) *	1993-07-30	2001-12-04	エーザイ株式会社	アミノ安息香酸誘導体
PL186204B1 (pl) *	1995-11-09	2003-11-28	Sanofi Synthelabo	Pochodne 5-fenylo-3-(piperydyn-4-ylo)-1,3,4-oksadiazol-2(3H)-onu do stosowania jako ligandy receptora 5-HT lub H

1997
- 1997-04-18 FR FR9704802A patent/FR2762316B1/fr not_active Expired - Fee Related
1998
- 1998-04-15 HU HU0002456A patent/HUP0002456A3/hu unknown
- 1998-04-15 NZ NZ500396A patent/NZ500396A/en unknown
- 1998-04-15 EP EP98920622A patent/EP0975631B1/fr not_active Expired - Lifetime
- 1998-04-15 TR TR1999/02600T patent/TR199902600T2/xx unknown
- 1998-04-15 CN CN98806195A patent/CN1260794A/zh active Pending
- 1998-04-15 BR BR9808926-9A patent/BR9808926A/pt not_active IP Right Cessation
- 1998-04-15 UA UA99105665A patent/UA57071C2/uk unknown
- 1998-04-15 ES ES98920622T patent/ES2165162T3/es not_active Expired - Lifetime
- 1998-04-15 SI SI9830088T patent/SI0975631T1/xx unknown
- 1998-04-15 US US09/403,003 patent/US6255319B1/en not_active Expired - Fee Related
- 1998-04-15 RU RU99123933/04A patent/RU2186066C2/ru not_active IP Right Cessation
- 1998-04-15 DK DK98920622T patent/DK0975631T3/da active
- 1998-04-15 IL IL13235298A patent/IL132352A0/xx unknown
- 1998-04-15 DE DE69801905T patent/DE69801905T2/de not_active Expired - Fee Related
- 1998-04-15 EE EEP199900487A patent/EE03769B1/xx not_active IP Right Cessation
- 1998-04-15 CZ CZ19993641A patent/CZ289154B6/cs not_active IP Right Cessation
- 1998-04-15 PL PL98336315A patent/PL186894B1/pl not_active IP Right Cessation
- 1998-04-15 KR KR1019997009542A patent/KR20010006452A/ko not_active Application Discontinuation
- 1998-04-15 SK SK1426-99A patent/SK283441B6/sk unknown
- 1998-04-15 WO PCT/FR1998/000754 patent/WO1998047898A1/fr not_active Application Discontinuation
- 1998-04-15 AU AU73415/98A patent/AU742666B2/en not_active Ceased
- 1998-04-15 AT AT98920622T patent/ATE206424T1/de not_active IP Right Cessation
- 1998-04-15 PT PT98920622T patent/PT975631E/pt unknown
- 1998-04-15 CA CA002286106A patent/CA2286106A1/en not_active Abandoned
- 1998-04-15 JP JP54514298A patent/JP2001521542A/ja active Pending
- 1998-04-17 TW TW087105892A patent/TW502005B/zh not_active IP Right Cessation
- 1998-04-17 AR ARP980101772A patent/AR012458A1/es not_active Application Discontinuation
- 1998-04-17 ZA ZA983257A patent/ZA983257B/xx unknown
- 1998-04-17 CO CO98021244A patent/CO4750656A1/es unknown
1999
- 1999-10-15 BG BG103810A patent/BG64053B1/bg unknown
- 1999-10-15 NO NO995040A patent/NO995040L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
FR2762316A1 (fr)	1998-10-23
BG103810A (en)	2000-06-30
EE03769B1 (et)	2002-06-17
EE9900487A (et)	2000-06-15
CO4750656A1 (es)	1999-03-31
KR20010006452A (ko)	2001-01-26
SK142699A3 (en)	2000-05-16
EP0975631A1 (fr)	2000-02-02
EP0975631B1 (fr)	2001-10-04
AU742666B2 (en)	2002-01-10
SI0975631T1 (en)	2002-06-30
CZ364199A3 (cs)	2000-03-15
AR012458A1 (es)	2000-10-18
DE69801905T2 (de)	2002-07-04
FR2762316B1 (fr)	1999-12-17
PL186894B1 (pl)	2004-03-31
ATE206424T1 (de)	2001-10-15
SK283441B6 (sk)	2003-07-01
WO1998047898A1 (fr)	1998-10-29
PL336315A1 (en)	2000-06-19
JP2001521542A (ja)	2001-11-06
PT975631E (pt)	2002-03-28
NO995040L (no)	1999-12-16
NZ500396A (en)	2001-04-27
DK0975631T3 (da)	2002-01-28
TW502005B (en)	2002-09-11
BG64053B1 (bg)	2003-11-28
CA2286106A1 (en)	1998-10-29
AU7341598A (en)	1998-11-13
DE69801905D1 (de)	2001-11-08
ZA983257B (en)	1998-10-19
BR9808926A (pt)	2000-08-01
ES2165162T3 (es)	2002-03-01
US6255319B1 (en)	2001-07-03
HUP0002456A3 (en)	2001-03-28
NO995040D0 (no)	1999-10-15
CZ289154B6 (cs)	2001-11-14
RU2186066C2 (ru)	2002-07-27
CN1260794A (zh)	2000-07-19
UA57071C2 (uk)	2003-06-16
HUP0002456A2 (hu)	2000-12-28
TR199902600T2 (xx)	2000-03-21

Publication	Publication Date	Title
HK1016165A1 (en)	1999-10-29	5-Phenyl-3-(peperidin-4-yl)-1,3,4-oxadiazol-2(3h)-one derivatives for use as 5-ht4 or h3 receptor ligands
ZA988078B (en)	2000-03-22	Substituted oxindole derivatives.
SG71077A1 (en)	2000-03-21	8-Substituted-1,3, 8-triaza-spiro (4.5)decan-4-on derivatives
AP9701077A0 (en)	1997-10-31	Substituted 6,5-hetero bicyclic derivatives
AP9701076A0 (en)	1997-10-31	Substituted 6,6-hetero bicyclic derivatives
ZA200203581B (en)	2004-02-25	Bicyclic imidazo-3-yl-amine derivatives.
ZA9811339B (en)	1999-07-08	Benzamidine derivatives.
AU5640299A (en)	2000-03-27	4-quinolinemethanol derivatives as purine receptor antagonists.(ii)
ZA989204B (en)	2000-04-10	Halogen substituted tetracyclic tetrahydrofuran derivatives.
ZA987304B (en)	2000-02-14	2-(4-aryl or heteroaryl-piperazin-1-ylmethyl)-1H-indole derivatives.
HK1028399A1 (en)	2001-02-16	Cyclopentene derivatives useful as antagonists of the motilin receptor.
IL132352A0 (en)	2001-03-19	5-Aryl-3-(8-azabicyclo (3.2.2) oct-3yl) -1,3,4-oxadiazol 22 (3h) - one derivatives as 5-ht4 receptor ligands
ZA982436B (en)	1999-09-23	Thiazolimine derivatives.
ZA975626B (en)	1998-01-30	Antineurodegenerative ergoline derivatives.
AU7658798A (en)	1998-11-27	5-phenyl-1,3,4-oxadiazol-2(3h)-one derivatives and their use as 5-ht4 ligands
AU1449997A (en)	1997-08-22	Diazabicyclo-octane derivatives as 5-ht receptor ligands
ZA9710062B (en)	1998-05-08	Heterocyclic derivatives.
ZA981307B (en)	1999-08-17	4-aminoethoxyindazole derivatives.
ZA9600758D (en)	1997-09-30	Idole derivatives as 5-ht receptor antagonist.
IL135923A0 (en)	2001-05-20	Process for the preparation of 8-azabicyclo (3.2.1) octane derivatives
ZA926890B (en)	1993-06-14	5-HT4 receptor antagonists.
GB9719193D0 (en)	1997-11-12	Aryloxyalkylamines as selective 5-ht receptor ligands
ZA978806B (en)	1998-07-23	Indole-2,3-dione-3-oxime derivatives
DK1133494T3 (da)	2004-06-14	8-Azabicyclo[3.2.1]oct-2-en-derivater
TW334917U (en)	1998-06-21	Adjustable multi-spindle drills seat