ZA200701950B - 6H-[1]benzopyrano[4,3-b]quinolines and their use as estrogenic agents - Google Patents

6H-[1]benzopyrano[4,3-b]quinolines and their use as estrogenic agents

Info

Publication number
ZA200701950B
ZA200701950B ZA200701950A ZA200701950A ZA200701950B ZA 200701950 B ZA200701950 B ZA 200701950B ZA 200701950 A ZA200701950 A ZA 200701950A ZA 200701950 A ZA200701950 A ZA 200701950A ZA 200701950 B ZA200701950 B ZA 200701950B
Authority
ZA
South Africa
Prior art keywords
benzopyrano
quinolines
estrogenic agents
estrogenic
agents
Prior art date
Application number
ZA200701950A
Other languages
English (en)
Inventor
An-Thien Vu
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ZA200701950B publication Critical patent/ZA200701950B/xx

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • A61P11/06Antiasthmatics
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    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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    • A61P13/12Drugs for disorders of the urinary system of the kidneys
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    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • AHUMAN NECESSITIES
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    • A61P35/00Antineoplastic agents
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    • A61P35/02Antineoplastic agents specific for leukemia
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    • A61P37/02Immunomodulators
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

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  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
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  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Reproductive Health (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Vascular Medicine (AREA)
ZA200701950A 2004-09-07 2007-03-06 6H-[1]benzopyrano[4,3-b]quinolines and their use as estrogenic agents ZA200701950B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US60776604P 2004-09-07 2004-09-07

Publications (1)

Publication Number Publication Date
ZA200701950B true ZA200701950B (en) 2009-11-25

Family

ID=35677606

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200701950A ZA200701950B (en) 2004-09-07 2007-03-06 6H-[1]benzopyrano[4,3-b]quinolines and their use as estrogenic agents

Country Status (15)

Country Link
US (1) US7354927B2 (ja)
EP (1) EP1789420A2 (ja)
JP (1) JP2008512458A (ja)
KR (1) KR20070061536A (ja)
CN (1) CN101052641A (ja)
AU (1) AU2005282554A1 (ja)
BR (1) BRPI0514974A (ja)
CA (1) CA2578164A1 (ja)
EC (1) ECSP077302A (ja)
IL (1) IL181514A0 (ja)
MX (1) MX2007002789A (ja)
NO (1) NO20071364L (ja)
RU (1) RU2007106870A (ja)
WO (1) WO2006029146A2 (ja)
ZA (1) ZA200701950B (ja)

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