ZA200108481B - 8A- and 9A-15-membered lactams. - Google Patents

8A- and 9A-15-membered lactams.

Info

Publication number: ZA200108481B
Authority: ZA; South Africa
Prior art keywords: membered lactams; lactams; membered
Prior art date: 1999-04-20

Application number

ZA200108481A

Other languages

English (en)

Inventor

Gorjana Lazarevski

Sulejman Alihodzic

Gabrijela Kobrehel

Stjepan Mutak

Original Assignee

Pliva Pharm & Chem Works

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-04-20

Filing date

2001-10-16

Publication date

2003-03-26

2001-10-16 Application filed by Pliva Pharm & Chem Works filed Critical Pliva Pharm & Chem Works

2003-03-26 Publication of ZA200108481B publication Critical patent/ZA200108481B/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Biochemistry (AREA)
Engineering & Computer Science (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Cephalosporin Compounds (AREA)
Hydrogenated Pyridines (AREA)
Steroid Compounds (AREA)

ZA200108481A 1999-04-20 2001-10-16 8A- and 9A-15-membered lactams. ZA200108481B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
HR990116A HRP990116B1 (en)	1999-04-20	1999-04-20	NOVEL 8a AND 9a- 15-MEMBERED LACTAMES

Publications (1)

Publication Number	Publication Date
ZA200108481B true ZA200108481B (en)	2003-03-26

Family

ID=10946907

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200108481A ZA200108481B (en)	1999-04-20	2001-10-16	8A- and 9A-15-membered lactams.

Country Status (33)

Country	Link
US (1)	US6593360B1 (xx)
EP (1)	EP1181298B1 (xx)
JP (1)	JP2002542254A (xx)
KR (1)	KR20020007379A (xx)
CN (1)	CN1246327C (xx)
AR (1)	AR028823A1 (xx)
AT (1)	ATE333461T1 (xx)
AU (1)	AU772272B2 (xx)
BG (1)	BG65281B1 (xx)
BR (1)	BR0009943A (xx)
CA (1)	CA2370273A1 (xx)
CZ (1)	CZ20013730A3 (xx)
DE (1)	DE60029439T2 (xx)
DK (1)	DK1181298T3 (xx)
EA (1)	EA003928B1 (xx)
EE (1)	EE04553B1 (xx)
ES (1)	ES2267519T3 (xx)
GE (1)	GEP20032929B (xx)
HK (1)	HK1049842B (xx)
HR (1)	HRP990116B1 (xx)
HU (1)	HUP0200868A3 (xx)
IL (1)	IL145990A0 (xx)
IS (1)	IS6110A (xx)
MX (1)	MXPA01010627A (xx)
NO (1)	NO320704B1 (xx)
NZ (1)	NZ515279A (xx)
PL (1)	PL351523A1 (xx)
PT (1)	PT1181298E (xx)
SK (1)	SK14942001A3 (xx)
TR (1)	TR200103019T2 (xx)
UA (1)	UA72246C2 (xx)
WO (1)	WO2000063223A1 (xx)
ZA (1)	ZA200108481B (xx)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0025688D0 (en)	2000-10-19	2000-12-06	Glaxo Group Ltd	Macrolides
HRP20020779A2 (en)	2002-09-27	2005-02-28	Pliva-Istra�iva�ki institut d.o.o.	NEW 3-DECLADINOSYL DERIVATIVES OF 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMICIN A 9a, 11-CYCLIC CARBAMATES
US7435805B2 (en) *	2003-05-30	2008-10-14	Glaxpsmithkline Istrazivacki	O-alkyl macrolide and azalide derivatives and regioselective process for their preparation
EP1879903A1 (en)	2005-05-10	2008-01-23	GlaxoSmithKline istrazivacki centar Zagreb d.o.o.	Ether linked macrolides useful for the treatment of microbial infections
EP2988597B1 (en)	2013-04-04	2022-06-08	President and Fellows of Harvard College	Macrolides and methods of their preparation and use
JP2017531663A (ja)	2014-10-08	2017-10-26	プレジデントアンドフェローズオブハーバードカレッジ	１４員ケトライドならびにそれらの調製および使用の方法
WO2016154591A1 (en)	2015-03-25	2016-09-29	President And Fellows Of Harvard College	Macrolides with modified desosamine sugars and uses thereof
GB201608236D0 (en)	2016-05-11	2016-06-22	Fidelta D O O	Seco macrolide compounds

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SI7910768A8 (en) *	1979-04-02	1996-06-30	Pliva Pharm & Chem Works	Process for pripering 11-aza-4-0-cladinosyl-6-0-desosaminyl-15-ethyl- 7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl- oxacyclopentadecane-2-one and their derivatives
SI9011409A (en) *	1990-07-18	1995-10-31	Pliva Pharm & Chem Works	O-methyl azitromycin derivates, methods and intermediates for their preparation and methods for preparation of pharmaceuticals products which comprise them
IL99995A (en) *	1990-11-21	1997-11-20	Roussel Uclaf	Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
US5527780A (en) *	1992-11-05	1996-06-18	Roussel Uclaf	Erythromycin derivatives
WO1997042204A1 (en) *	1996-05-07	1997-11-13	Abbott Laboratories	6-o-substituted erythromycins and method for making them
AU1082599A (en) *	1997-10-16	1999-05-03	Merck & Co., Inc.	8a-azalides, compositions containing such compounds and methods of treatment
HRP980189B1 (en) *	1998-04-06	2004-04-30	Pliva Pharm & Chem Works	Novel 15-membered lactams ketolides

1999
- 1999-04-20 HR HR990116A patent/HRP990116B1/xx not_active IP Right Cessation
2000
- 2000-04-19 UA UA2001117855A patent/UA72246C2/uk unknown
- 2000-04-19 TR TR2001/03019T patent/TR200103019T2/xx unknown
- 2000-04-19 BR BR0009943-0A patent/BR0009943A/pt not_active IP Right Cessation
- 2000-04-19 DK DK00920937T patent/DK1181298T3/da active
- 2000-04-19 CZ CZ20013730A patent/CZ20013730A3/cs unknown
- 2000-04-19 HU HU0200868A patent/HUP0200868A3/hu unknown
- 2000-04-19 EP EP00920937A patent/EP1181298B1/en not_active Expired - Lifetime
- 2000-04-19 PL PL00351523A patent/PL351523A1/xx unknown
- 2000-04-19 CN CNB008078238A patent/CN1246327C/zh not_active Expired - Fee Related
- 2000-04-19 AT AT00920937T patent/ATE333461T1/de not_active IP Right Cessation
- 2000-04-19 NZ NZ515279A patent/NZ515279A/xx unknown
- 2000-04-19 CA CA002370273A patent/CA2370273A1/en not_active Abandoned
- 2000-04-19 WO PCT/HR2000/000009 patent/WO2000063223A1/en active IP Right Grant
- 2000-04-19 GE GEAP20006202A patent/GEP20032929B/en unknown
- 2000-04-19 JP JP2000612313A patent/JP2002542254A/ja active Pending
- 2000-04-19 ES ES00920937T patent/ES2267519T3/es not_active Expired - Lifetime
- 2000-04-19 AU AU41347/00A patent/AU772272B2/en not_active Ceased
- 2000-04-19 SK SK1494-2001A patent/SK14942001A3/sk unknown
- 2000-04-19 DE DE60029439T patent/DE60029439T2/de not_active Expired - Fee Related
- 2000-04-19 PT PT00920937T patent/PT1181298E/pt unknown
- 2000-04-19 IL IL14599000A patent/IL145990A0/xx unknown
- 2000-04-19 EE EEP200100544A patent/EE04553B1/xx not_active IP Right Cessation
- 2000-04-19 MX MXPA01010627A patent/MXPA01010627A/es active IP Right Grant
- 2000-04-19 US US09/959,204 patent/US6593360B1/en not_active Expired - Fee Related
- 2000-04-19 KR KR1020017013433A patent/KR20020007379A/ko not_active Application Discontinuation
- 2000-04-19 EA EA200101103A patent/EA003928B1/ru not_active IP Right Cessation
- 2000-04-24 AR ARP000101906A patent/AR028823A1/es unknown
2001
- 2001-10-16 ZA ZA200108481A patent/ZA200108481B/xx unknown
- 2001-10-16 IS IS6110A patent/IS6110A/is unknown
- 2001-10-18 NO NO20015068A patent/NO320704B1/no unknown
- 2001-11-20 BG BG106117A patent/BG65281B1/bg unknown
2003
- 2003-01-23 HK HK03100592.9A patent/HK1049842B/zh not_active IP Right Cessation

Also Published As

Publication number	Publication date
CZ20013730A3 (cs)	2002-04-17
HUP0200868A2 (hu)	2002-07-29
CA2370273A1 (en)	2000-10-26
CN1362964A (zh)	2002-08-07
HK1049842A1 (en)	2003-05-30
CN1246327C (zh)	2006-03-22
WO2000063223A1 (en)	2000-10-26
AU772272B2 (en)	2004-04-22
HK1049842B (zh)	2006-09-22
TR200103019T2 (tr)	2002-01-21
NO20015068L (no)	2001-12-13
DK1181298T3 (da)	2006-11-13
IS6110A (is)	2001-10-16
ATE333461T1 (de)	2006-08-15
BR0009943A (pt)	2002-01-08
AR028823A1 (es)	2003-05-28
DE60029439T2 (de)	2007-02-01
HRP990116A2 (en)	2001-10-31
ES2267519T3 (es)	2007-03-16
EE200100544A (et)	2003-02-17
MXPA01010627A (es)	2002-06-04
US6593360B1 (en)	2003-07-15
NZ515279A (en)	2003-04-29
NO320704B1 (no)	2006-01-16
EP1181298B1 (en)	2006-07-19
EA003928B1 (ru)	2003-10-30
NO20015068D0 (no)	2001-10-18
BG65281B1 (bg)	2007-11-30
EP1181298A1 (en)	2002-02-27
DE60029439D1 (de)	2006-08-31
UA72246C2 (uk)	2005-02-15
JP2002542254A (ja)	2002-12-10
PT1181298E (pt)	2006-11-30
GEP20032929B (en)	2003-03-25
HUP0200868A3 (en)	2003-03-28
EA200101103A1 (ru)	2002-04-25
AU4134700A (en)	2000-11-02
SK14942001A3 (sk)	2002-08-06
KR20020007379A (ko)	2002-01-26
HRP990116B1 (en)	2007-10-31
BG106117A (en)	2002-07-31
PL351523A1 (en)	2003-05-05
IL145990A0 (en)	2002-07-25
EE04553B1 (et)	2005-10-17

Publication	Publication Date	Title
MXPA01013362A (es)	2003-09-04	Anticuerpos de humano, anti-alfavbeta3 recombinantes, °cidos nucleicos que codifican a los mismos y metodos de uso.
EG24361A (en)	2009-03-04	4-pyrimiding1-n-acy1.l.phenlalanines
ZA200200477B (en)	2003-06-25	2-pyrazolin-5-ones.
ZA200000894B (en)	2000-08-24	4-Phenyl-pyridine derivatives.
ZA200201055B (en)	2003-07-30	Amino-triazolopyridine derivatives.
ZA200201269B (en)	2003-02-14	Toothbrush.
HK1042488A1 (en)	2002-08-16	1-Heterocycle substituted diarylamines.
HK1052037A1 (en)	2003-08-29	Structural member.
MXPA03004292A (es)	2004-02-12	Compuesto de lactama.
ZA200203768B (en)	2003-08-11	Toothbrush.
ZA200202537B (en)	2003-09-23	Pour-on-formulations.
ZA200109595B (en)	2003-05-28	13-methyl-erythromycin derivatives.
HK1053470A1 (en)	2003-10-24	4-Pyridinyln-acyl-l-phenylalanines.
ZA200201829B (en)	2003-08-27	New phenylpiperazines.
HK1046411A1 (en)	2003-01-10	5-Phenyl-pyrimidine derivatives.
HK1029502A1 (en)	2001-04-06	Slider-pull-assembling unit.
HK1054848A1 (en)	2003-12-19	Toothbrush.
MXPA03004250A (es)	2003-09-22	Compuesto de lactama.
MXPA01012681A (es)	2003-09-04	Recipiente.
ZA200108481B (en)	2003-03-26	8A- and 9A-15-membered lactams.
ZA200201276B (en)	2003-07-30	3-Amino-2-phenyl-propane derivatives.
MXPA02000261A (es)	2003-08-20	Aminoindanos novedosos.
HK1054382A1 (en)	2003-11-28	Substituted pyrroles.
GB0029720D0 (en)	2001-01-17	I.S machine7544232001
MXPA01011285A (es)	2003-09-04	Derivados de tio-oxindol.