ZA200105580B - Ketolide antibiotics. - Google Patents
Ketolide antibiotics. Download PDFInfo
- Publication number
- ZA200105580B ZA200105580B ZA200105580A ZA200105580A ZA200105580B ZA 200105580 B ZA200105580 B ZA 200105580B ZA 200105580 A ZA200105580 A ZA 200105580A ZA 200105580 A ZA200105580 A ZA 200105580A ZA 200105580 B ZA200105580 B ZA 200105580B
- Authority
- ZA
- South Africa
- Prior art keywords
- alkyl
- aryl
- groups
- halo
- independently selected
- Prior art date
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- 239000003835 ketolide antibiotic agent Substances 0.000 title description 2
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
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- Health & Medical Sciences (AREA)
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- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US11734299P | 1999-01-27 | 1999-01-27 |
Publications (1)
Publication Number | Publication Date |
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ZA200105580B true ZA200105580B (en) | 2003-02-17 |
Family
ID=22372371
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA200105580A ZA200105580B (en) | 1999-01-27 | 2001-07-06 | Ketolide antibiotics. |
Country Status (39)
Country | Link |
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US (1) | US6833444B2 (hu) |
EP (1) | EP1147121B1 (hu) |
JP (1) | JP3947360B2 (hu) |
KR (1) | KR20020002380A (hu) |
CN (1) | CN1342163A (hu) |
AP (1) | AP2001002222A0 (hu) |
AT (1) | ATE256694T1 (hu) |
AU (1) | AU1675400A (hu) |
BG (1) | BG105730A (hu) |
BR (1) | BR9916969A (hu) |
CA (1) | CA2359708C (hu) |
CO (1) | CO5150229A1 (hu) |
CZ (1) | CZ20012675A3 (hu) |
DE (1) | DE69913738T2 (hu) |
DK (1) | DK1147121T3 (hu) |
DZ (1) | DZ3000A1 (hu) |
EA (1) | EA200100623A1 (hu) |
EE (1) | EE200100394A (hu) |
ES (1) | ES2212655T3 (hu) |
HK (1) | HK1042707A1 (hu) |
HN (1) | HN2000000003A (hu) |
HR (1) | HRP20010559A2 (hu) |
HU (1) | HUP0105190A3 (hu) |
ID (1) | ID30233A (hu) |
IL (1) | IL144178A0 (hu) |
IS (1) | IS5984A (hu) |
MA (1) | MA26717A1 (hu) |
NO (1) | NO20013680L (hu) |
OA (1) | OA11753A (hu) |
PA (1) | PA8489501A1 (hu) |
PE (1) | PE20001422A1 (hu) |
PT (1) | PT1147121E (hu) |
SI (1) | SI1147121T1 (hu) |
SK (1) | SK10172001A3 (hu) |
TN (1) | TNSN00007A1 (hu) |
TR (1) | TR200102128T2 (hu) |
UY (1) | UY25990A1 (hu) |
WO (1) | WO2000044761A2 (hu) |
ZA (1) | ZA200105580B (hu) |
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AP1060A (en) | 1998-01-02 | 2002-04-23 | Pfizer Prod Inc | Novel erythromycin derivatives. |
TR200102128T2 (tr) | 1999-01-27 | 2001-12-21 | Pfizer Products Inc. | Ketolid antibiyotikler |
ATE340183T1 (de) | 1999-04-16 | 2006-10-15 | Kosan Biosciences Inc | Antiinfektiƶse makrolidderivate |
US6451768B1 (en) | 1999-04-16 | 2002-09-17 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
AU4354900A (en) | 1999-04-16 | 2000-11-02 | Kosan Biosciences, Inc. | Ketolide antibacterials |
US6514944B2 (en) | 1999-04-16 | 2003-02-04 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
US6590083B1 (en) | 1999-04-16 | 2003-07-08 | Ortho-Mcneil Pharmaceutical, Inc. | Ketolide antibacterials |
US6939861B2 (en) | 1999-04-16 | 2005-09-06 | Kosan Biosciences, Inc. | Amido macrolides |
CA2373117C (en) | 1999-05-24 | 2006-02-28 | Pfizer Products Inc. | 13-methyl-erythromycin derivatives |
ATE271062T1 (de) | 2000-06-30 | 2004-07-15 | Pfizer Prod Inc | Makrolid-antibiotika |
US20020115621A1 (en) | 2000-08-07 | 2002-08-22 | Wei-Gu Su | Macrolide antibiotics |
AU2002217277B2 (en) * | 2000-12-21 | 2005-06-16 | Glaxo Group Limited | Macrolide antibiotics |
PE20030438A1 (es) * | 2001-09-05 | 2003-07-03 | Hokuriku Pharmaceutical | Medicamento que comprende un derivado de eritromicina como agente antituberculoso |
ES2552682T3 (es) | 2003-03-10 | 2015-12-01 | Merck Sharp & Dohme Corp. | Agentes antibacterianos novedosos |
BRPI0513903A (pt) * | 2004-07-28 | 2008-05-20 | Ranbaxy Lab Ltd | derivados de cetolƬdeos Ćŗteis como agentes antimicrobianos, seus processos de preparaĆ§Ć£o e composiƧƵes farmacĆŖuticas compreendendo os mesmos |
BRPI0519135A2 (pt) | 2004-12-21 | 2008-12-23 | Pfizer Prod Inc | macrolĆdeos |
RU2455308C2 (ru) * | 2006-05-01 | 2012-07-10 | Š¢Š°Š¹ŃŠ¾ Š¤Š°ŃŠ¼Š°ŃŃŃŃŠøŠŗŠ°Š» ŠŠ¾., ŠŃŠ“. | ŠŠ°ŠŗŃŠ¾Š»ŠøŠ“Š½ŃŠµ ŠæŃŠ¾ŠøŠ·Š²Š¾Š“Š½ŃŠµ |
CN105732745A (zh) | 2007-10-25 | 2016-07-06 | ę£®ę®ęå¶čÆå ¬åø | 大ēÆå é Æē±»ęčåēå¶å¤ę¹ę³ |
ES2565083T3 (es) | 2008-10-24 | 2016-03-31 | Cempra Pharmaceuticals, Inc. | Biodefensas usando macrĆ³lidos que contienen triazol |
US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
CN102724874B (zh) | 2009-09-10 | 2018-06-01 | ę£®ę®ęå¶čÆå ¬åø | ę²»ēēē¾ćē»ę øē åmacē¾ē ēę¹ę³ |
MY162411A (en) | 2010-03-22 | 2017-06-15 | Cempra Pharmaceuticals Inc | Crystalline forms of a macrolide, and uses therefor |
JP6184319B2 (ja) | 2010-05-20 | 2017-08-23 | ć»ć³ćć© ćć”ć¼ćć·ć„ć¼ćć£ć«ć«ćŗļ¼ć¤ć³ć³ć¼ćć¬ć¤ććć | ććÆćć©ć¤ćé”ććć³ć±ćć©ć¤ćé”ćŖćć³ć«ćć®äøéä½ćčŖæč£½ććććć®å·„ēØ |
EP2613630A4 (en) | 2010-09-10 | 2014-01-15 | Cempra Pharmaceuticals Inc | FLUOROCETOLIDES FORMING HYDROGEN LINKS TO TREAT DISEASES |
KR20140139083A (ko) | 2012-03-27 | 2014-12-04 | ģ ķė¼ ķė§ģķ°ģ»¬ģ¤, ģøķ¬. | ė§ķ¬ė”¤ė¼ģ“ėź³ ķģģ ė„¼ ķ¬ģ¬ķźø° ģķ ė¹ź²½źµ¬ ģ ģ |
JP6426696B2 (ja) | 2013-03-14 | 2018-11-21 | ć»ć³ćć© ćć”ć¼ćć·ć„ć¼ćć£ć«ć«ćŗļ¼ć¤ć³ć³ć¼ćć¬ć¤ććć | å¼åøåØē¾ę£ć®ę²»ēć®ććć®ę¹ę³ććć³č£½å¤ |
WO2014145210A1 (en) | 2013-03-15 | 2014-09-18 | Cempra Pharmaceuticals, Inc. | Convergent processes for preparing macrolide antibacterial agents |
WO2014156549A1 (ja) | 2013-03-28 | 2014-10-02 | äøäŗč£½ę²¹ę Ŗå¼ä¼ē¤¾ | ē·č±čē½ć²ć«ē¶ēµęē©åć³ćć¼ćŗę§é£å |
CN106518939B (zh) * | 2015-09-14 | 2019-12-31 | ę±čå„„čµåŗ·čÆäøęéå ¬åø | äøē§å¶å¤Solithromycinååē©ēę¹ę³ |
WO2018067663A2 (en) * | 2016-10-04 | 2018-04-12 | Biopharmati Sa | Ketolides having antibacterial activity |
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YU43006B (en) | 1981-03-06 | 1989-02-28 | Pliva Pharm & Chem Works | Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof |
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FR2697524B1 (fr) | 1992-11-05 | 1994-12-23 | Roussel Uclaf | Nouveaux dƩrivƩs de l'Ʃrythromycine, leur procƩdƩ de prƩparation et leur application comme mƩdicaments. |
FR2719587B1 (fr) * | 1994-05-03 | 1996-07-12 | Roussel Uclaf | Nouveaux dƩrivƩs de l'Ʃrythromycine, leur procƩdƩ de prƩparation et leur application comme mƩdicaments. |
FR2727969B1 (fr) * | 1994-12-09 | 1997-01-17 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
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FR2789392B1 (fr) * | 1999-02-04 | 2001-10-05 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
AU4354900A (en) | 1999-04-16 | 2000-11-02 | Kosan Biosciences, Inc. | Ketolide antibacterials |
ATE340183T1 (de) | 1999-04-16 | 2006-10-15 | Kosan Biosciences Inc | Antiinfektiƶse makrolidderivate |
US6355620B1 (en) | 1999-05-14 | 2002-03-12 | Abbott Laboratories | C-2 modified erythromycin derivatives |
CA2373117C (en) | 1999-05-24 | 2006-02-28 | Pfizer Products Inc. | 13-methyl-erythromycin derivatives |
EP1114826A3 (en) | 1999-12-29 | 2001-10-31 | Pfizer Products Inc. | Novel antibacterial and prokinetic macrolides |
EP1122261A3 (en) | 2000-01-31 | 2001-09-26 | Pfizer Products Inc. | 13 and 14-membered antibacterial macrolides |
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ATE271062T1 (de) | 2000-06-30 | 2004-07-15 | Pfizer Prod Inc | Makrolid-antibiotika |
-
1999
- 1999-12-28 TR TR2001/02128T patent/TR200102128T2/xx unknown
- 1999-12-28 EA EA200100623A patent/EA200100623A1/ru unknown
- 1999-12-28 WO PCT/IB1999/002051 patent/WO2000044761A2/en active IP Right Grant
- 1999-12-28 CN CN99815909A patent/CN1342163A/zh active Pending
- 1999-12-28 AU AU16754/00A patent/AU1675400A/en not_active Abandoned
- 1999-12-28 EP EP99959627A patent/EP1147121B1/en not_active Expired - Lifetime
- 1999-12-28 JP JP2000596017A patent/JP3947360B2/ja not_active Expired - Fee Related
- 1999-12-28 OA OA1200100191A patent/OA11753A/en unknown
- 1999-12-28 KR KR1020017009382A patent/KR20020002380A/ko not_active Application Discontinuation
- 1999-12-28 BR BR9916969-0A patent/BR9916969A/pt not_active Application Discontinuation
- 1999-12-28 HU HU0105190A patent/HUP0105190A3/hu unknown
- 1999-12-28 CZ CZ20012675A patent/CZ20012675A3/cs unknown
- 1999-12-28 ES ES99959627T patent/ES2212655T3/es not_active Expired - Lifetime
- 1999-12-28 ID IDW00200101637A patent/ID30233A/id unknown
- 1999-12-28 EE EEP200100394A patent/EE200100394A/xx unknown
- 1999-12-28 DK DK99959627T patent/DK1147121T3/da active
- 1999-12-28 IL IL14417899A patent/IL144178A0/xx unknown
- 1999-12-28 PT PT99959627T patent/PT1147121E/pt unknown
- 1999-12-28 SI SI9930486T patent/SI1147121T1/xx unknown
- 1999-12-28 SK SK1017-2001A patent/SK10172001A3/sk unknown
- 1999-12-28 CA CA002359708A patent/CA2359708C/en not_active Expired - Fee Related
- 1999-12-28 DE DE69913738T patent/DE69913738T2/de not_active Expired - Lifetime
- 1999-12-28 AP APAP/P/2001/002222A patent/AP2001002222A0/en unknown
- 1999-12-28 AT AT99959627T patent/ATE256694T1/de not_active IP Right Cessation
-
2000
- 2000-01-05 TN TNTNSN00007A patent/TNSN00007A1/fr unknown
- 2000-01-05 DZ DZ000002A patent/DZ3000A1/xx active
- 2000-01-06 PA PA20008489501A patent/PA8489501A1/es unknown
- 2000-01-06 HN HN2000000003A patent/HN2000000003A/es unknown
- 2000-01-06 PE PE2000000013A patent/PE20001422A1/es not_active Application Discontinuation
- 2000-01-06 MA MA25883A patent/MA26717A1/fr unknown
- 2000-01-21 CO CO00003460A patent/CO5150229A1/es unknown
- 2000-01-27 UY UY25990A patent/UY25990A1/es unknown
-
2001
- 2001-06-28 IS IS5984A patent/IS5984A/is unknown
- 2001-07-06 ZA ZA200105580A patent/ZA200105580B/en unknown
- 2001-07-25 BG BG105730A patent/BG105730A/xx unknown
- 2001-07-25 HR HR20010559A patent/HRP20010559A2/hr not_active Application Discontinuation
- 2001-07-26 NO NO20013680A patent/NO20013680L/no not_active Application Discontinuation
-
2002
- 2002-04-05 US US10/116,969 patent/US6833444B2/en not_active Expired - Fee Related
- 2002-05-31 HK HK02104131.0A patent/HK1042707A1/zh unknown
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