YU43585B - Process for making 1,1-dioxopenicilano-iloximethyl-6-(2-amino-2-phenylacetamido) penicilanate - Google Patents

Process for making 1,1-dioxopenicilano-iloximethyl-6-(2-amino-2-phenylacetamido) penicilanate

Info

Publication number: YU43585B
Authority: YU; Yugoslavia
Prior art keywords: iloximethyl; dioxopenicilano; penicilanate; phenylacetamido; amino
Prior art date: 1981-03-23

Application number

YU1810/84A

Other languages

English (en)

Other versions

YU181084A (en

Inventor

V J Jasys

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-03-23

Filing date

1984-10-23

Publication date

1989-08-31

1984-10-23 Application filed by Pfizer filed Critical Pfizer

1987-06-30 Publication of YU181084A publication Critical patent/YU181084A/xx

1989-08-31 Publication of YU43585B publication Critical patent/YU43585B/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
- C07D499/32—Esters
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Cephalosporin Compounds (AREA)

YU1810/84A 1981-03-23 1984-10-23 Process for making 1,1-dioxopenicilano-iloximethyl-6-(2-amino-2-phenylacetamido) penicilanate YU43585B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US24645681A	1981-03-23	1981-03-23

Publications (2)

Publication Number	Publication Date
YU181084A YU181084A (en)	1987-06-30
YU43585B true YU43585B (en)	1989-08-31

Family

ID=22930766

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
YU619/82A YU42761B (en)	1981-03-23	1982-03-22	Process for obtaining 6-halogenated 1,1-dioxo-penicillanoyloxy-methyl-6-(2-amino-2-phenylacetamido)penicillanate
YU1810/84A YU43585B (en)	1981-03-23	1984-10-23	Process for making 1,1-dioxopenicilano-iloximethyl-6-(2-amino-2-phenylacetamido) penicilanate

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
YU619/82A YU42761B (en)	1981-03-23	1982-03-22	Process for obtaining 6-halogenated 1,1-dioxo-penicillanoyloxy-methyl-6-(2-amino-2-phenylacetamido)penicillanate

Country Status (32)

Country	Link
EP (1)	EP0061274B1 (xx)
JP (3)	JPS57169493A (xx)
KR (1)	KR860001368B1 (xx)
AU (1)	AU531892B2 (xx)
BG (2)	BG37380A3 (xx)
CA (1)	CA1213581A (xx)
CS (1)	CS227345B2 (xx)
DD (1)	DD202163A5 (xx)
DE (1)	DE3267505D1 (xx)
DK (3)	DK162392C (xx)
EG (1)	EG15803A (xx)
ES (2)	ES8305768A1 (xx)
FI (1)	FI74284C (xx)
GB (1)	GB2095250A (xx)
GR (1)	GR75935B (xx)
GT (1)	GT198274393A (xx)
HK (1)	HK52487A (xx)
HU (2)	HU187667B (xx)
IE (1)	IE52835B1 (xx)
IL (1)	IL65308A (xx)
IN (1)	IN159362B (xx)
MY (1)	MY8700499A (xx)
NO (1)	NO159658C (xx)
NZ (1)	NZ200066A (xx)
PH (1)	PH17602A (xx)
PL (3)	PL139261B1 (xx)
PT (1)	PT74621B (xx)
RO (2)	RO84278B (xx)
SG (1)	SG23387G (xx)
SU (2)	SU1277898A3 (xx)
YU (2)	YU42761B (xx)
ZA (1)	ZA821899B (xx)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0084730A1 (en) *	1982-01-22	1983-08-03	Beecham Group Plc	Esters of penicillin derivatives with beta-lactamase inhibitors, their preparation and their use
PH20068A (en) *	1982-12-06	1986-09-18	Pfizer	Process and intermediates for sultamicillin and analogs
GB8808701D0 (en) *	1988-04-13	1988-05-18	Erba Carlo Spa	Beta-lactam derivatives
ES2039299B1 (es) *	1991-10-04	1994-05-16	Asturpharma S A	Procedimiento de obtencion de esteres de acido 1,1-dioxopenicilanico y sus sales.
ES2100125B1 (es) *	1995-06-02	1998-04-01	Asturpharma S A	Procedimiento de preparacion de esteres de metanodiol de acido dioxopenicilanico.
CN112724162B (zh) *	2020-12-28	2022-06-10	华南农业大学	一种阿莫西林-舒巴坦杂合分子的合成方法及应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IE49880B1 (en) *	1979-02-13	1986-01-08	Leo Pharm Prod Ltd	Penicillin derivatives
ZA80796B (en) *	1979-02-13	1981-02-25	Leo Pharm Prod Ltd	Chemical compounds
SE449103B (sv) *	1979-03-05	1987-04-06	Pfizer	Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
ZA80646B (en) *	1979-03-05	1981-02-25	Pfizer	Process and intermediates for penicillanic acid,1,1-dioxide and esters thereof
IE50650B1 (en) *	1979-10-11	1986-06-11	Leo Pharm Prod Ltd	Method for producing penicillanic acid derivatives

1982
- 1982-02-09 IN IN102/DEL/82A patent/IN159362B/en unknown
- 1982-03-15 BG BG8255782A patent/BG37380A3/xx unknown
- 1982-03-15 BG BG8467396A patent/BG38939A3/xx unknown
- 1982-03-15 DE DE8282301296T patent/DE3267505D1/de not_active Expired
- 1982-03-15 EP EP82301296A patent/EP0061274B1/en not_active Expired
- 1982-03-16 GB GB8207695A patent/GB2095250A/en not_active Withdrawn
- 1982-03-17 GT GT198274393A patent/GT198274393A/es unknown
- 1982-03-18 NO NO820898A patent/NO159658C/no not_active IP Right Cessation
- 1982-03-19 NZ NZ200066A patent/NZ200066A/en unknown
- 1982-03-19 DD DD82238305A patent/DD202163A5/de not_active IP Right Cessation
- 1982-03-21 EG EG148/82A patent/EG15803A/xx active
- 1982-03-22 HU HU82852A patent/HU187667B/hu unknown
- 1982-03-22 ES ES510655A patent/ES8305768A1/es not_active Expired
- 1982-03-22 HU HU842661A patent/HU189917B/hu unknown
- 1982-03-22 KR KR8201223A patent/KR860001368B1/ko active
- 1982-03-22 IE IE659/82A patent/IE52835B1/en unknown
- 1982-03-22 RO RO106986A patent/RO84278B/ro unknown
- 1982-03-22 YU YU619/82A patent/YU42761B/xx unknown
- 1982-03-22 AU AU81764/82A patent/AU531892B2/en not_active Expired
- 1982-03-22 CA CA000398989A patent/CA1213581A/en not_active Expired
- 1982-03-22 ZA ZA821899A patent/ZA821899B/xx unknown
- 1982-03-22 SU SU823408198K patent/SU1277898A3/ru active
- 1982-03-22 RO RO82113915A patent/RO87946A/ro unknown
- 1982-03-22 PT PT74621A patent/PT74621B/pt unknown
- 1982-03-22 DK DK127182A patent/DK162392C/da not_active IP Right Cessation
- 1982-03-22 GR GR67669A patent/GR75935B/el unknown
- 1982-03-22 SU SU823408198A patent/SU1277897A3/ru active
- 1982-03-22 IL IL65308A patent/IL65308A/xx not_active IP Right Cessation
- 1982-03-22 FI FI820991A patent/FI74284C/fi not_active IP Right Cessation
- 1982-03-23 PL PL1982240664A patent/PL139261B1/pl unknown
- 1982-03-23 PH PH27043A patent/PH17602A/en unknown
- 1982-03-23 CS CS822014A patent/CS227345B2/cs unknown
- 1982-03-23 PL PL1982235578A patent/PL134250B1/pl unknown
- 1982-03-23 JP JP57046185A patent/JPS57169493A/ja active Granted
- 1982-03-23 PL PL1982240663A patent/PL138851B1/pl unknown
1983
- 1983-01-13 ES ES518970A patent/ES8403132A1/es not_active Expired
1984
- 1984-10-23 YU YU1810/84A patent/YU43585B/xx unknown
1987
- 1987-03-09 SG SG233/87A patent/SG23387G/en unknown
- 1987-07-09 HK HK524/87A patent/HK52487A/xx not_active IP Right Cessation
- 1987-07-28 JP JP62188687A patent/JPS6345287A/ja active Pending
- 1987-07-28 JP JP62188686A patent/JPS63146886A/ja active Pending
- 1987-12-30 MY MY499/87A patent/MY8700499A/xx unknown
1991
- 1991-06-21 DK DK121491A patent/DK165746C/da not_active IP Right Cessation
1992
- 1992-02-20 DK DK021892A patent/DK167119B1/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
NO159658C (no)	1989-01-25
NO159658B (no)	1988-10-17
RO87946A (ro)	1985-12-20
HK52487A (en)	1987-07-17
PT74621B (en)	1984-11-26
FI74284B (fi)	1987-09-30
SG23387G (en)	1987-07-10
IL65308A0 (en)	1982-05-31
PL240664A1 (en)	1983-09-12
DK162392B (da)	1991-10-21
PT74621A (en)	1982-04-01
BG37380A3 (en)	1985-05-15
ES518970A0 (es)	1984-03-01
MY8700499A (en)	1987-12-31
AU8176482A (en)	1982-11-04
DK162392C (da)	1992-03-09
GT198274393A (es)	1983-09-08
FI820991L (fi)	1982-09-24
DE3267505D1 (en)	1986-01-02
RO84278B (ro)	1984-07-30
ES510655A0 (es)	1983-04-16
ES8305768A1 (es)	1983-04-16
CS227345B2 (en)	1984-04-16
HUT34985A (en)	1985-05-28
ZA821899B (en)	1983-01-26
PL240663A1 (en)	1983-09-12
PH17602A (en)	1984-10-05
AU531892B2 (en)	1983-09-08
EP0061274B1 (en)	1985-11-21
YU181084A (en)	1987-06-30
DK21892A (da)	1992-02-20
RO84278A (ro)	1984-05-23
NO820898L (no)	1982-09-24
GB2095250A (en)	1982-09-29
GR75935B (xx)	1984-08-02
DK165746C (da)	1993-06-07
CA1213581A (en)	1986-11-04
JPH0331717B2 (xx)	1991-05-08
DK121491A (da)	1991-06-21
DK167119B1 (da)	1993-08-30
HU187667B (en)	1986-02-28
KR860001368B1 (ko)	1986-09-17
PL138851B1 (en)	1986-11-29
KR830009113A (ko)	1983-12-17
RO87946B (ro)	1985-12-02
JPS57169493A (en)	1982-10-19
IN159362B (xx)	1987-05-09
PL134250B1 (en)	1985-08-31
DK21892D0 (da)	1992-02-20
ES8403132A1 (es)	1984-03-01
IE52835B1 (en)	1988-03-16
SU1277897A3 (ru)	1986-12-15
EP0061274A1 (en)	1982-09-29
EG15803A (en)	1990-08-30
BG38939A3 (en)	1986-03-14
HU189917B (en)	1986-08-28
DK127182A (da)	1982-09-24
DK121491D0 (da)	1991-06-21
IE820659L (en)	1982-09-23
NZ200066A (en)	1985-08-16
PL235578A1 (en)	1983-06-20
IL65308A (en)	1985-03-31
JPS63146886A (ja)	1988-06-18
YU42761B (en)	1988-12-31
DD202163A5 (de)	1983-08-31
FI74284C (fi)	1988-01-11
JPS6345287A (ja)	1988-02-26
DK165746B (da)	1993-01-11
YU61982A (en)	1985-03-20
PL139261B1 (en)	1987-01-31
SU1277898A3 (ru)	1986-12-15

Publication	Publication Date	Title
ZA826877B (en)	1983-08-31	Process for making 1,2-dichloroethane
DE3263757D1 (en)	1985-06-27	Process for preparing 1,2-dihydro-6-methyl-2-oxo-5-(pyridinyl)nicotinonitriles
DE3161380D1 (en)	1983-12-15	Process for preparing 2,3-dichloro-sulfonyl acrylonitriles
YU52082A (en)	1985-03-20	Process for preparing 2,3-dichloro-5-trichloro methylpyridine
YU42698B (en)	1988-10-31	Process for obtaining penicillanoyl-oxymethyl-penicillanate-1,1,1',1'-tetraoxide
DE3261973D1 (en)	1985-02-28	Process for preparing 1,1-dihalo-1,2,2,2,-tetrafluoroethanes
ZA828536B (en)	1983-10-26	Process for making 1,2-dichloroethane
RO87709B (ro)	1985-10-01	Procedeu pentru prepararea unor 1,1-alcandiol-carboxilati
YU105982A (en)	1985-03-20	Process for foam-flotation
YU43585B (en)	1989-08-31	Process for making 1,1-dioxopenicilano-iloximethyl-6-(2-amino-2-phenylacetamido) penicilanate
DE3166154D1 (en)	1984-10-25	Process for preparing 1,2-dimethyl-5-nitroimidazole
YU143082A (en)	1985-03-20	Process for obtaining 5,6,7,7a-tetrahydro-4h-thieno(3,2-c)-2-pyridinone
DE3169609D1 (en)	1985-05-02	Process for preparing m,m'-dinitrobenzophenone
YU42722B (en)	1988-12-31	Process for obtaining 6-hydrazono-pyrido (2,1-b)h quinazoline-11-one
PL235332A1 (en)	1983-07-18	Process for preparing 1-/1,3-benzoolioxol-5-yl/-2-pyrrolidinone
YU55383A (en)	1985-12-31	Process for obtaining 1,2,4-triazole-1-yl-propionitrile
YU284181A (en)	1983-10-31	Process for obtaining 2,3-dihydro-pyrane
YU192682A (en)	1984-12-31	Process for obtaining new 1,2,3-thiadiazole-5-yl-carbamides
DE3264300D1 (en)	1985-07-25	Process for making substituted 1,11-diaminoundecanes
DE3263234D1 (en)	1985-05-30	Process for preparing 0,s-dialkylphosphoroamido thioates
YU217682A (en)	1984-12-31	Process for obtaining thiazolo - and (1,3)-thiazino(2,3-c)(1,2,4)triaziones
GB2176777B (en)	1989-07-12	Method for preparing 2,2,6,6-tetramethyl-4-oxopiperidine
DE3260739D1 (en)	1984-10-18	Process for making 2-carbalkoxy-5-carboxynitrobenzenes
YU196982A (en)	1984-12-31	Process for obtaining 6,6-diiodopenicillanic acid
YU192582A (en)	1984-08-31	Process for obtaining new 1,2,3-thiadiazole-5-yl-carbamide derivatives