NO159658C - Mellomprodukt for fremstilling av 1,1-diokso-penicillanoyloksymetyl-6-(2-amino-2-fenyl-acetamido)penicillanat-antibiotika. - Google Patents

Mellomprodukt for fremstilling av 1,1-diokso-penicillanoyloksymetyl-6-(2-amino-2-fenyl-acetamido)penicillanat-antibiotika.

Info

Publication number
NO159658C
NO159658C NO820898A NO820898A NO159658C NO 159658 C NO159658 C NO 159658C NO 820898 A NO820898 A NO 820898A NO 820898 A NO820898 A NO 820898A NO 159658 C NO159658 C NO 159658C
Authority
NO
Norway
Prior art keywords
penicillanoyloxymethyl
penicillanate
acetamido
dioxo
antibiotics
Prior art date
Application number
NO820898A
Other languages
English (en)
Other versions
NO159658B (no
NO820898L (no
Inventor
Vytautas John Jasys
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO820898L publication Critical patent/NO820898L/no
Priority to NO831024A priority Critical patent/NO159659C/no
Publication of NO159658B publication Critical patent/NO159658B/no
Publication of NO159658C publication Critical patent/NO159658C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Cephalosporin Compounds (AREA)
NO820898A 1981-03-23 1982-03-18 Mellomprodukt for fremstilling av 1,1-diokso-penicillanoyloksymetyl-6-(2-amino-2-fenyl-acetamido)penicillanat-antibiotika. NO159658C (no)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NO831024A NO159659C (no) 1981-03-23 1983-03-23 Fremgangsm te for fremstilling av 1,1-dioksopenicilksymetyl-6-(2-amino-2-fenylacetamido)penicillanat-antibiotika.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24645681A 1981-03-23 1981-03-23

Publications (3)

Publication Number Publication Date
NO820898L NO820898L (no) 1982-09-24
NO159658B NO159658B (no) 1988-10-17
NO159658C true NO159658C (no) 1989-01-25

Family

ID=22930766

Family Applications (1)

Application Number Title Priority Date Filing Date
NO820898A NO159658C (no) 1981-03-23 1982-03-18 Mellomprodukt for fremstilling av 1,1-diokso-penicillanoyloksymetyl-6-(2-amino-2-fenyl-acetamido)penicillanat-antibiotika.

Country Status (32)

Country Link
EP (1) EP0061274B1 (no)
JP (3) JPS57169493A (no)
KR (1) KR860001368B1 (no)
AU (1) AU531892B2 (no)
BG (2) BG37380A3 (no)
CA (1) CA1213581A (no)
CS (1) CS227345B2 (no)
DD (1) DD202163A5 (no)
DE (1) DE3267505D1 (no)
DK (3) DK162392C (no)
EG (1) EG15803A (no)
ES (2) ES8305768A1 (no)
FI (1) FI74284C (no)
GB (1) GB2095250A (no)
GR (1) GR75935B (no)
GT (1) GT198274393A (no)
HK (1) HK52487A (no)
HU (2) HU187667B (no)
IE (1) IE52835B1 (no)
IL (1) IL65308A (no)
IN (1) IN159362B (no)
MY (1) MY8700499A (no)
NO (1) NO159658C (no)
NZ (1) NZ200066A (no)
PH (1) PH17602A (no)
PL (3) PL139261B1 (no)
PT (1) PT74621B (no)
RO (2) RO84278B (no)
SG (1) SG23387G (no)
SU (2) SU1277898A3 (no)
YU (2) YU42761B (no)
ZA (1) ZA821899B (no)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0084730A1 (en) * 1982-01-22 1983-08-03 Beecham Group Plc Esters of penicillin derivatives with beta-lactamase inhibitors, their preparation and their use
PH20068A (en) * 1982-12-06 1986-09-18 Pfizer Process and intermediates for sultamicillin and analogs
GB8808701D0 (en) * 1988-04-13 1988-05-18 Erba Carlo Spa Beta-lactam derivatives
ES2039299B1 (es) * 1991-10-04 1994-05-16 Asturpharma S A Procedimiento de obtencion de esteres de acido 1,1-dioxopenicilanico y sus sales.
ES2100125B1 (es) * 1995-06-02 1998-04-01 Asturpharma S A Procedimiento de preparacion de esteres de metanodiol de acido dioxopenicilanico.
CN112724162B (zh) * 2020-12-28 2022-06-10 华南农业大学 一种阿莫西林-舒巴坦杂合分子的合成方法及应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
ZA80796B (en) * 1979-02-13 1981-02-25 Leo Pharm Prod Ltd Chemical compounds
SE449103B (sv) * 1979-03-05 1987-04-06 Pfizer Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
ZA80646B (en) * 1979-03-05 1981-02-25 Pfizer Process and intermediates for penicillanic acid,1,1-dioxide and esters thereof
IE50650B1 (en) * 1979-10-11 1986-06-11 Leo Pharm Prod Ltd Method for producing penicillanic acid derivatives

Also Published As

Publication number Publication date
NO159658B (no) 1988-10-17
RO87946A (ro) 1985-12-20
HK52487A (en) 1987-07-17
PT74621B (en) 1984-11-26
FI74284B (fi) 1987-09-30
SG23387G (en) 1987-07-10
IL65308A0 (en) 1982-05-31
PL240664A1 (en) 1983-09-12
DK162392B (da) 1991-10-21
PT74621A (en) 1982-04-01
BG37380A3 (en) 1985-05-15
ES518970A0 (es) 1984-03-01
MY8700499A (en) 1987-12-31
AU8176482A (en) 1982-11-04
DK162392C (da) 1992-03-09
GT198274393A (es) 1983-09-08
FI820991L (fi) 1982-09-24
DE3267505D1 (en) 1986-01-02
RO84278B (ro) 1984-07-30
ES510655A0 (es) 1983-04-16
ES8305768A1 (es) 1983-04-16
CS227345B2 (en) 1984-04-16
HUT34985A (en) 1985-05-28
ZA821899B (en) 1983-01-26
PL240663A1 (en) 1983-09-12
PH17602A (en) 1984-10-05
AU531892B2 (en) 1983-09-08
EP0061274B1 (en) 1985-11-21
YU181084A (en) 1987-06-30
DK21892A (da) 1992-02-20
RO84278A (ro) 1984-05-23
NO820898L (no) 1982-09-24
GB2095250A (en) 1982-09-29
GR75935B (no) 1984-08-02
DK165746C (da) 1993-06-07
CA1213581A (en) 1986-11-04
JPH0331717B2 (no) 1991-05-08
DK121491A (da) 1991-06-21
DK167119B1 (da) 1993-08-30
HU187667B (en) 1986-02-28
KR860001368B1 (ko) 1986-09-17
PL138851B1 (en) 1986-11-29
KR830009113A (ko) 1983-12-17
RO87946B (ro) 1985-12-02
JPS57169493A (en) 1982-10-19
IN159362B (no) 1987-05-09
PL134250B1 (en) 1985-08-31
DK21892D0 (da) 1992-02-20
ES8403132A1 (es) 1984-03-01
IE52835B1 (en) 1988-03-16
SU1277897A3 (ru) 1986-12-15
EP0061274A1 (en) 1982-09-29
EG15803A (en) 1990-08-30
YU43585B (en) 1989-08-31
BG38939A3 (en) 1986-03-14
HU189917B (en) 1986-08-28
DK127182A (da) 1982-09-24
DK121491D0 (da) 1991-06-21
IE820659L (en) 1982-09-23
NZ200066A (en) 1985-08-16
PL235578A1 (en) 1983-06-20
IL65308A (en) 1985-03-31
JPS63146886A (ja) 1988-06-18
YU42761B (en) 1988-12-31
DD202163A5 (de) 1983-08-31
FI74284C (fi) 1988-01-11
JPS6345287A (ja) 1988-02-26
DK165746B (da) 1993-01-11
YU61982A (en) 1985-03-20
PL139261B1 (en) 1987-01-31
SU1277898A3 (ru) 1986-12-15

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MK1K Patent expired

Free format text: EXPIRED IN MARCH 2002