DOP2010000259A - Derivados heterociclicos de urea y metodos de uso de los mismos-211 - Google Patents
Derivados heterociclicos de urea y metodos de uso de los mismos-211Info
- Publication number
- DOP2010000259A DOP2010000259A DO2010000259A DO2010000259A DOP2010000259A DO P2010000259 A DOP2010000259 A DO P2010000259A DO 2010000259 A DO2010000259 A DO 2010000259A DO 2010000259 A DO2010000259 A DO 2010000259A DO P2010000259 A DOP2010000259 A DO P2010000259A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- heterociclical
- urea
- derivatives
- methods
- same
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Abstract
Se describen compuestos de fórmula (I) y sus sales farmacéuticamente aceptables. También se describen procesos para su preparación, composiciones farmacéuticas que los contienen, su uso como medicamentos y su uso en el tratamiento de infecciones bacterianas.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US3162108P | 2008-02-26 | 2008-02-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
DOP2010000259A true DOP2010000259A (es) | 2010-09-15 |
Family
ID=40474753
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DO2010000259A DOP2010000259A (es) | 2008-02-26 | 2010-08-24 | Derivados heterociclicos de urea y metodos de uso de los mismos-211 |
Country Status (23)
Country | Link |
---|---|
US (1) | US20120101100A1 (es) |
EP (1) | EP2262801A1 (es) |
JP (1) | JP2011513216A (es) |
KR (1) | KR20100117681A (es) |
CN (1) | CN102015699A (es) |
AR (1) | AR070493A1 (es) |
AU (1) | AU2009219883A1 (es) |
BR (1) | BRPI0907562A2 (es) |
CA (1) | CA2716365A1 (es) |
CL (1) | CL2009000426A1 (es) |
CO (1) | CO6290656A2 (es) |
CR (1) | CR11641A (es) |
DO (1) | DOP2010000259A (es) |
EA (1) | EA201001368A1 (es) |
EC (1) | ECSP10010419A (es) |
IL (1) | IL207731A0 (es) |
MX (1) | MX2010009163A (es) |
PE (1) | PE20091573A1 (es) |
SA (1) | SA109300138B1 (es) |
TW (1) | TW200940537A (es) |
UY (1) | UY31673A1 (es) |
WO (1) | WO2009106885A1 (es) |
ZA (1) | ZA201005997B (es) |
Families Citing this family (64)
Publication number | Priority date | Publication date | Assignee | Title |
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US9029411B2 (en) | 2008-01-25 | 2015-05-12 | Millennium Pharmaceuticals, Inc. | Thiophenes and uses thereof |
AU2012203026B2 (en) * | 2008-03-21 | 2014-06-12 | Novartis Ag | Novel heterocyclic compounds and uses thereof |
US8865732B2 (en) | 2008-03-21 | 2014-10-21 | Novartis Ag | Heterocyclic compounds and uses thereof |
EA201001858A1 (ru) * | 2008-06-04 | 2011-08-30 | Астразенека Аб | Гетероциклические производные мочевины для лечения бактериальных инфекций |
WO2010052448A2 (en) * | 2008-11-05 | 2010-05-14 | Ucb Pharma S.A. | Fused pyrazine derivatives as kinase inhibitors |
CN102264721B (zh) | 2008-11-10 | 2015-12-09 | 沃泰克斯药物股份有限公司 | 用作atr激酶抑制剂的化合物 |
KR101745331B1 (ko) | 2008-12-19 | 2017-06-09 | 버텍스 파마슈티칼스 인코포레이티드 | Atr 키나제의 억제제로서 유용한 피라진 유도체 |
US9090601B2 (en) * | 2009-01-30 | 2015-07-28 | Millennium Pharmaceuticals, Inc. | Thiazole derivatives |
CN102395585A (zh) | 2009-01-30 | 2012-03-28 | 米伦纽姆医药公司 | 杂芳基化合物和其作为pi3k抑制剂的用途 |
US8796314B2 (en) | 2009-01-30 | 2014-08-05 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
TW201102065A (en) | 2009-05-29 | 2011-01-16 | Astrazeneca Ab | Heterocyclic urea derivatives and methods of use thereof |
FR2953519B1 (fr) * | 2009-12-08 | 2012-02-10 | Commissariat Energie Atomique | Nouveaux composes chimiques aptes a complexer au moins un element metallique et complexe de coordination a base de ces composes |
BR112012024705A2 (pt) | 2010-03-31 | 2016-06-07 | Actelion Pharmaceuticals Ltd | derivados antibacterianos de isoquinolin-3-ilureia |
AR081331A1 (es) | 2010-04-23 | 2012-08-08 | Cytokinetics Inc | Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos |
EP2560488B1 (en) | 2010-04-23 | 2015-10-28 | Cytokinetics, Inc. | Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use |
AR081626A1 (es) | 2010-04-23 | 2012-10-10 | Cytokinetics Inc | Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos |
NZ603477A (en) | 2010-05-12 | 2014-09-26 | Vertex Pharma | Compounds useful as inhibitors of atr kinase |
JP2013529200A (ja) | 2010-05-12 | 2013-07-18 | バーテックス ファーマシューティカルズ インコーポレイテッド | Atrキナーゼ阻害剤として有用な化合物 |
US9334244B2 (en) | 2010-05-12 | 2016-05-10 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
EP2569284B1 (en) * | 2010-05-12 | 2015-07-08 | Vertex Pharmaceuticals Incorporated | 2-aminopyridine derivatives useful as inhibitors of atr kinase |
WO2011143419A1 (en) | 2010-05-12 | 2011-11-17 | Vertex Pharmaceuticals Incorporated | Pyrazines useful as inhibitors of atr kinase |
JP2013526538A (ja) | 2010-05-12 | 2013-06-24 | バーテックス ファーマシューティカルズ インコーポレイテッド | Atrキナーゼ阻害剤として有用な化合物 |
AU2011270807A1 (en) | 2010-06-23 | 2013-01-31 | Vertex Pharmaceuticals Incorporated | Pyrrolo- pyrazine derivatives useful as inhibitors of ATR kinase |
WO2012021611A1 (en) | 2010-08-11 | 2012-02-16 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
WO2012021615A1 (en) | 2010-08-11 | 2012-02-16 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
MX2013001660A (es) | 2010-08-11 | 2013-06-03 | Millenium Pharmaceuticals Inc | Heteroarilos y usos de los mismos. |
CN103153955A (zh) | 2010-09-17 | 2013-06-12 | 普渡制药公司 | 吡啶化合物及其用途 |
AU2011316016A1 (en) | 2010-10-13 | 2013-05-30 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
AR088729A1 (es) | 2011-03-29 | 2014-07-02 | Actelion Pharmaceuticals Ltd | Derivados de 3-ureidoisoquinolin-8-ilo y una composicion farmaceutica |
KR20140027974A (ko) | 2011-04-05 | 2014-03-07 | 버텍스 파마슈티칼스 인코포레이티드 | Tra 키나제의 억제제로서 유용한 아미노피라진 화합물 |
JP2014522818A (ja) | 2011-06-22 | 2014-09-08 | バーテックス ファーマシューティカルズ インコーポレイテッド | Atrキナーゼ阻害剤として有用な化合物 |
US9309250B2 (en) | 2011-06-22 | 2016-04-12 | Vertex Pharmaceuticals Incorporated | Substituted pyrrolo[2,3-b]pyrazines as ATR kinase inhibitors |
EP2723745A1 (en) | 2011-06-22 | 2014-04-30 | Vertex Pharmaceuticals Inc. | Compounds useful as inhibitors of atr kinase |
MX2014001860A (es) * | 2011-09-12 | 2014-05-30 | Hoffmann La Roche | Hidrazidas del acido 3-piridin carboxilico como agentes elevadores del colesterol de lipoproteina de alta densidad (hdl). |
WO2013049720A1 (en) | 2011-09-30 | 2013-04-04 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
WO2013049719A1 (en) | 2011-09-30 | 2013-04-04 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
HUE046429T2 (hu) | 2011-09-30 | 2020-03-30 | Vertex Pharma | ATR kináz inhibítoraként használható vegyületek elõállítására szolgáló eljárás |
ES2899880T3 (es) | 2011-09-30 | 2022-03-15 | Vertex Pharma | Tratamiento de cáncer de páncreas y cáncer de pulmón de células no pequeñas con inhibidores de ATR |
AU2012315611A1 (en) | 2011-09-30 | 2014-04-17 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
KR20140088194A (ko) * | 2011-11-04 | 2014-07-09 | 에프. 호프만-라 로슈 아게 | 아릴-퀴놀린 유도체 |
WO2013071093A1 (en) | 2011-11-09 | 2013-05-16 | Vertex Pharmaceuticals Incorporated | Pyrazine compounds useful as inhibitors of atr kinase |
WO2013071088A1 (en) | 2011-11-09 | 2013-05-16 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
EP2776419B1 (en) | 2011-11-09 | 2016-05-11 | Vertex Pharmaceuticals Incorporated | Pyrazine compounds useful as inhibitors of atr kinase |
WO2013071094A1 (en) | 2011-11-09 | 2013-05-16 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
EP2776422A1 (en) | 2011-11-09 | 2014-09-17 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
JP5957537B2 (ja) * | 2011-12-21 | 2016-07-27 | ビオタ ヨーロッパ リミテッドBiota Europe Ltd | 複素環式ウレア化合物 |
IN2014KN02410A (es) | 2012-04-05 | 2015-05-01 | Vertex Pharma | |
EP2862856B1 (en) | 2012-06-15 | 2018-08-01 | Mitsubishi Tanabe Pharma Corporation | Imidazole and triazole compounds as dgat-1 inhibitors |
EP2904406B1 (en) | 2012-10-04 | 2018-03-21 | Vertex Pharmaceuticals Incorporated | Method for measuring atr inhibition mediated increases in dna damage |
EP2909202A1 (en) | 2012-10-16 | 2015-08-26 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
EP3418281B1 (en) | 2012-12-07 | 2020-09-30 | Vertex Pharmaceuticals Inc. | Pyrazolo[1,5-a]pyrimidines useful as inhibitors of atr kinase for the treatment of cancer diseases |
US9242969B2 (en) | 2013-03-14 | 2016-01-26 | Novartis Ag | Biaryl amide compounds as kinase inhibitors |
EP2970286A1 (en) | 2013-03-15 | 2016-01-20 | Vertex Pharmaceuticals Inc. | Fused pyrazolopyrimidine derivatives useful as inhibitors of atr kinase |
AU2014316684A1 (en) | 2013-09-06 | 2016-04-28 | Aurigene Discovery Technologies Limited | 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives as immunomodulators |
MX370390B (es) | 2013-12-06 | 2019-12-11 | Vertex Pharma | Compuesto de 2-amino-6-fluoro-n-[5-fluoro-piridin-3-il]pirazolo[1, 5-a]pirimidin-3-carboxamida util como inhibidor de cinasa de ataxia telangiectasia mutada (atm) y rad3 relacionados (atr), su preparacion, diferentes formas solidas y sus derivados radiomarcados. |
CN110590787A (zh) | 2014-06-05 | 2019-12-20 | 沃泰克斯药物股份有限公司 | Atr激酶抑制剂的制备方法及其不同的固体形式 |
JP6936007B2 (ja) | 2014-06-17 | 2021-09-15 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | Chk1阻害剤とatr阻害剤との組み合わせを使用してがんを処置する方法 |
UY36294A (es) | 2014-09-12 | 2016-04-29 | Novartis Ag | Compuestos y composiciones como inhibidores de quinasa |
CN107427497A (zh) * | 2015-03-10 | 2017-12-01 | 奥瑞基尼探索技术有限公司 | 作为免疫调节剂的3‑取代的1,3,4‑噁二唑和噻二唑化合物 |
MX2018003657A (es) | 2015-09-30 | 2018-04-30 | Vertex Pharma | Metodo para tratar cancer usando una combinacion de agentes que dañan el adn e inhibidores de proteina relacionada con ataxia telangiectasia y rad3 (atr). |
CN106866571B (zh) * | 2017-01-20 | 2018-06-29 | 中国药科大学 | 杂环脲类化合物及其药物组合物和应用 |
AU2018239711A1 (en) | 2017-03-24 | 2019-11-07 | Taisho Pharmaceutical Co., Ltd. | 2(1h)-quinolinone derivative |
CN111116559A (zh) * | 2018-11-01 | 2020-05-08 | 复旦大学 | 吡啶脲类化合物及其制备方法和制药用途 |
WO2022147210A1 (en) * | 2020-12-31 | 2022-07-07 | Evrys Bio, Llc | Anti-tumor compositions and methods |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0014022D0 (en) * | 2000-06-08 | 2000-08-02 | Novartis Ag | Organic compounds |
US7569591B2 (en) * | 2003-01-31 | 2009-08-04 | Vertex Pharmaceuticals Incorporated | Gyrase inhibitors and uses thereof |
AR042956A1 (es) * | 2003-01-31 | 2005-07-13 | Vertex Pharma | Inhibidores de girasa y usos de los mismos |
MX2009005603A (es) * | 2006-12-04 | 2009-06-08 | Astrazeneca Ab | Compuestos de urea policiclicos antibacterianos. |
-
2009
- 2009-02-24 TW TW098105845A patent/TW200940537A/zh unknown
- 2009-02-25 EA EA201001368A patent/EA201001368A1/ru unknown
- 2009-02-25 UY UY031673A patent/UY31673A1/es not_active Application Discontinuation
- 2009-02-25 JP JP2010547261A patent/JP2011513216A/ja active Pending
- 2009-02-25 BR BRPI0907562A patent/BRPI0907562A2/pt not_active IP Right Cessation
- 2009-02-25 EP EP09715006A patent/EP2262801A1/en not_active Withdrawn
- 2009-02-25 CL CL2009000426A patent/CL2009000426A1/es unknown
- 2009-02-25 CA CA2716365A patent/CA2716365A1/en not_active Abandoned
- 2009-02-25 SA SA109300138A patent/SA109300138B1/ar unknown
- 2009-02-25 AU AU2009219883A patent/AU2009219883A1/en not_active Abandoned
- 2009-02-25 MX MX2010009163A patent/MX2010009163A/es unknown
- 2009-02-25 US US12/392,730 patent/US20120101100A1/en not_active Abandoned
- 2009-02-25 CN CN2009801157676A patent/CN102015699A/zh active Pending
- 2009-02-25 KR KR1020107021270A patent/KR20100117681A/ko not_active Application Discontinuation
- 2009-02-25 WO PCT/GB2009/050187 patent/WO2009106885A1/en active Application Filing
- 2009-02-26 AR ARP090100667A patent/AR070493A1/es not_active Application Discontinuation
- 2009-02-26 PE PE2009000289A patent/PE20091573A1/es not_active Application Discontinuation
-
2010
- 2010-08-19 IL IL207731A patent/IL207731A0/en unknown
- 2010-08-23 ZA ZA2010/05997A patent/ZA201005997B/en unknown
- 2010-08-24 CO CO10104182A patent/CO6290656A2/es not_active Application Discontinuation
- 2010-08-24 CR CR11641A patent/CR11641A/es not_active Application Discontinuation
- 2010-08-24 EC EC2010010419A patent/ECSP10010419A/es unknown
- 2010-08-24 DO DO2010000259A patent/DOP2010000259A/es unknown
Also Published As
Publication number | Publication date |
---|---|
IL207731A0 (en) | 2010-12-30 |
EA201001368A1 (ru) | 2011-04-29 |
BRPI0907562A2 (pt) | 2017-05-23 |
CL2009000426A1 (es) | 2011-02-11 |
JP2011513216A (ja) | 2011-04-28 |
TW200940537A (en) | 2009-10-01 |
CO6290656A2 (es) | 2011-06-20 |
CN102015699A (zh) | 2011-04-13 |
CR11641A (es) | 2010-10-05 |
KR20100117681A (ko) | 2010-11-03 |
ZA201005997B (en) | 2013-01-30 |
MX2010009163A (es) | 2010-09-14 |
UY31673A1 (es) | 2009-09-30 |
WO2009106885A1 (en) | 2009-09-03 |
CA2716365A1 (en) | 2009-09-03 |
AR070493A1 (es) | 2010-04-07 |
EP2262801A1 (en) | 2010-12-22 |
PE20091573A1 (es) | 2009-11-12 |
US20120101100A1 (en) | 2012-04-26 |
AU2009219883A1 (en) | 2009-09-03 |
SA109300138B1 (ar) | 2012-11-03 |
ECSP10010419A (es) | 2010-09-30 |
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