CL2011000729A1 - Compuestos derivados de metanopirazolo[3,4-e][1,3]diazepin; procedimiento de preparacion; composicion farmaceutica que los comprende; y su uso en el tratamiento de infecciones bacterianas. - Google Patents
Compuestos derivados de metanopirazolo[3,4-e][1,3]diazepin; procedimiento de preparacion; composicion farmaceutica que los comprende; y su uso en el tratamiento de infecciones bacterianas.Info
- Publication number
- CL2011000729A1 CL2011000729A1 CL2011000729A CL2011000729A CL2011000729A1 CL 2011000729 A1 CL2011000729 A1 CL 2011000729A1 CL 2011000729 A CL2011000729 A CL 2011000729A CL 2011000729 A CL2011000729 A CL 2011000729A CL 2011000729 A1 CL2011000729 A1 CL 2011000729A1
- Authority
- CL
- Chile
- Prior art keywords
- treatment
- pharmaceutical composition
- methanopyrazolo
- diazepine
- bacterial infections
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/18—Bridged systems
Abstract
Compuestos heterocíclicos nitrogenados; procedimiento de preparación; composición farmacéutica; y uso en el tratamiento de infecciones bacterianas.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0805472A FR2936798B1 (fr) | 2008-10-03 | 2008-10-03 | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens. |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2011000729A1 true CL2011000729A1 (es) | 2012-07-06 |
Family
ID=40548019
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2011000729A CL2011000729A1 (es) | 2008-10-03 | 2011-04-01 | Compuestos derivados de metanopirazolo[3,4-e][1,3]diazepin; procedimiento de preparacion; composicion farmaceutica que los comprende; y su uso en el tratamiento de infecciones bacterianas. |
Country Status (18)
Country | Link |
---|---|
US (1) | US8067435B2 (es) |
EP (2) | EP2845855A1 (es) |
JP (1) | JP5555240B2 (es) |
KR (1) | KR20110067137A (es) |
CN (1) | CN102203094B (es) |
AU (1) | AU2009299511A1 (es) |
BR (1) | BRPI0919810A8 (es) |
CA (1) | CA2739503A1 (es) |
CL (1) | CL2011000729A1 (es) |
CO (1) | CO6361957A2 (es) |
EA (1) | EA021799B1 (es) |
EC (1) | ECSP11010946A (es) |
FR (1) | FR2936798B1 (es) |
IL (1) | IL212059A0 (es) |
MX (1) | MX2011003573A (es) |
PE (1) | PE20110845A1 (es) |
WO (1) | WO2010038115A1 (es) |
ZA (1) | ZA201102429B (es) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8772490B2 (en) | 2010-12-22 | 2014-07-08 | Meiji Seika Pharma Co., Ltd. | Optically active diazabicyclooctane derivatives and process for preparing the same |
EP2872510B1 (en) | 2011-08-30 | 2016-11-23 | Wockhardt Limited | 1,6-diazabicyclo[3,2,1]octan-7-one derivatives and their use in the treatment of bacterial infections |
MX349827B (es) * | 2011-09-13 | 2017-08-14 | Wockhardt Ltd | Compuestos que contienen nitrogeno y su uso. |
SG11201406120SA (en) * | 2012-03-30 | 2014-10-30 | Cubist Pharm Inc | ISOXAZOLE β-LACTAMASE INHIBITORS |
AR090539A1 (es) * | 2012-04-02 | 2014-11-19 | Astrazeneca Ab | COMPUESTOS INHIBIDORES DE b LACTAMASA |
RU2693898C2 (ru) | 2012-05-30 | 2019-07-05 | Мейдзи Сейка Фарма Ко., Лтд. | НОВЫЙ ИНГИБИТОР бета-ЛАКТАМАЗЫ И СПОСОБ ЕГО ПОЛУЧЕНИЯ |
EP2961751B1 (en) * | 2012-08-25 | 2018-03-21 | Wockhardt Limited | 1,6- diazabicyclo [3,2,1]octan- 7- one derivatives and their use in the treatment of bacterial infections |
NZ718009A (en) | 2013-09-24 | 2018-03-23 | Meiji Seika Pharma Co Ltd | Process for producing diazabicyclooctane derivative and intermediate thereof |
HUE051925T2 (hu) | 2013-10-08 | 2021-04-28 | Meiji Seika Pharma Co Ltd | Dizabiciklooktán származék kristályai és diazabiciklooktán származék kristályainak elõállítási eljárása |
JP6411482B2 (ja) * | 2013-10-11 | 2018-10-24 | ウォックハート リミテッド | 窒素含有化合物およびその使用 |
JP6764862B2 (ja) | 2014-11-17 | 2020-10-07 | エンタシス・セラピューティックス・リミテッド | 耐性細菌感染症の治療のための併用療法 |
KR102555657B1 (ko) | 2014-12-05 | 2023-07-18 | 메이지 세이카 파루마 가부시키가이샤 | 디아자비시클로옥탄 유도체의 결정 및 안정된 동결 건조 제제의 제조법 |
EP3075733A1 (en) * | 2015-03-31 | 2016-10-05 | Mutabilis | Novel heterocyclic compounds and their use in preventing or treating bacterial infections |
US10072006B2 (en) * | 2015-03-31 | 2018-09-11 | Mutabilis | Heterocyclic compounds and their use in preventing or treating bacterial infections |
CA2980395A1 (en) | 2015-04-03 | 2016-10-06 | Mutabilis | Heterocyclic compounds and their use in preventing or treating bacterial infections |
US9951072B2 (en) | 2015-10-02 | 2018-04-24 | Legochem Biosciences, Inc. | Compositions and methods for inhibiting beta-lactamase |
IL289686B2 (en) | 2016-09-16 | 2023-03-01 | Entasis Therapeutics Ltd | Beta-lactamase inhibitor compounds |
PL3630111T3 (pl) | 2017-05-08 | 2022-05-23 | Entasis Therapeutics, Inc. | Związki i sposoby leczenia zakażeń bakteryjnych |
EP3604315A1 (en) | 2018-07-30 | 2020-02-05 | Mutabilis | Heterocyclic compounds and their use in preventing or treating bacterial infections |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6387928B1 (en) | 1997-09-15 | 2002-05-14 | The Procter & Gamble Co. | Antimicrobial quinolones, their compositions and uses |
ID24703A (id) | 1997-09-15 | 2000-08-03 | Procter & Gamble | Kuinolon antimikroba, komposisi dan penggunaannya |
FR2812635B1 (fr) | 2000-08-01 | 2002-10-11 | Aventis Pharma Sa | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
AU2002230891B2 (en) | 2000-12-14 | 2005-04-07 | The Procter & Gamble Company | Antimicrobial quinolones |
NZ525570A (en) | 2000-12-14 | 2005-04-29 | Procter & Gamble | Antimicrobial 2-pyridones, their compositions and uses |
FR2825705B1 (fr) * | 2001-06-08 | 2005-05-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens |
FR2833596B1 (fr) | 2001-12-14 | 2005-02-18 | Aventis Pharma Sa | Procede de preparation de derives d'echinocandine |
FR2835186B1 (fr) | 2002-01-28 | 2006-10-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases |
US6900224B2 (en) | 2002-07-31 | 2005-05-31 | The Procter & Gamble Company | Antimicrobial quinolones, their compositions and uses |
FR2844273B1 (fr) | 2002-09-05 | 2008-04-04 | Aventis Pharma Sa | Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens. |
FR2844270B1 (fr) | 2002-09-11 | 2006-05-19 | Aventis Pharma Sa | Derives de la quinolyl propyl piperidine, leur procede et intermediaires de preparation et les compositions qui les contiennent |
FR2844268B1 (fr) | 2002-09-11 | 2004-10-22 | Aventis Pharma Sa | Derives de la quinolyl propyl piperidine, leurs procedes et intermediaires de preparation et les compositions qui les contiennent |
FR2848210B1 (fr) * | 2002-12-06 | 2007-10-19 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens et inhibiteurs de beta-lactamases |
US7439253B2 (en) | 2002-12-06 | 2008-10-21 | Novexel | Heterocyclic compounds, their preparation and their use as medicaments, in particular as antibacterials and beta-lactamase inhibitors |
US7232833B2 (en) | 2003-03-28 | 2007-06-19 | Novexel | 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them |
US7449481B2 (en) | 2004-04-13 | 2008-11-11 | Cephalon, Inc. | Thio-substituted biaryl-methanesulfinyl derivatives |
FR2914923B1 (fr) * | 2007-04-12 | 2013-06-14 | Novexel | Nouveaux composes heterocycliques azotes,leur preparation et leur utilisation comme medicaments antibacteriens. |
FR2937034B1 (fr) * | 2008-10-10 | 2012-11-23 | Novexel | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens |
-
2008
- 2008-10-03 FR FR0805472A patent/FR2936798B1/fr not_active Expired - Fee Related
-
2009
- 2009-08-03 EP EP14188601.0A patent/EP2845855A1/fr not_active Withdrawn
- 2009-08-03 JP JP2011529643A patent/JP5555240B2/ja not_active Expired - Fee Related
- 2009-08-03 EP EP09786093A patent/EP2344499A1/fr not_active Withdrawn
- 2009-08-03 CA CA2739503A patent/CA2739503A1/fr not_active Abandoned
- 2009-08-03 WO PCT/IB2009/006433 patent/WO2010038115A1/fr active Application Filing
- 2009-08-03 KR KR1020117009615A patent/KR20110067137A/ko not_active Application Discontinuation
- 2009-08-03 AU AU2009299511A patent/AU2009299511A1/en not_active Abandoned
- 2009-08-03 EA EA201170522A patent/EA021799B1/ru not_active IP Right Cessation
- 2009-08-03 CN CN200980141781.3A patent/CN102203094B/zh not_active Expired - Fee Related
- 2009-08-03 BR BRPI0919810A patent/BRPI0919810A8/pt not_active IP Right Cessation
- 2009-08-03 PE PE2011000827A patent/PE20110845A1/es not_active Application Discontinuation
- 2009-08-03 MX MX2011003573A patent/MX2011003573A/es active IP Right Grant
- 2009-08-05 US US12/536,096 patent/US8067435B2/en not_active Expired - Fee Related
-
2011
- 2011-03-30 ZA ZA2011/02429A patent/ZA201102429B/en unknown
- 2011-03-31 IL IL212059A patent/IL212059A0/en unknown
- 2011-04-01 EC EC2011010946A patent/ECSP11010946A/es unknown
- 2011-04-01 CO CO11040684A patent/CO6361957A2/es active IP Right Grant
- 2011-04-01 CL CL2011000729A patent/CL2011000729A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
JP5555240B2 (ja) | 2014-07-23 |
PE20110845A1 (es) | 2011-11-17 |
CO6361957A2 (es) | 2012-01-20 |
JP2012504593A (ja) | 2012-02-23 |
BRPI0919810A2 (pt) | 2017-10-31 |
ZA201102429B (en) | 2012-05-30 |
WO2010038115A1 (fr) | 2010-04-08 |
KR20110067137A (ko) | 2011-06-21 |
US20100087648A1 (en) | 2010-04-08 |
US8067435B2 (en) | 2011-11-29 |
FR2936798B1 (fr) | 2012-09-28 |
BRPI0919810A8 (pt) | 2017-12-12 |
MX2011003573A (es) | 2011-08-12 |
EP2845855A1 (fr) | 2015-03-11 |
CA2739503A1 (fr) | 2010-04-08 |
FR2936798A1 (fr) | 2010-04-09 |
IL212059A0 (en) | 2011-06-30 |
AU2009299511A1 (en) | 2010-04-08 |
EA021799B1 (ru) | 2015-09-30 |
CN102203094A (zh) | 2011-09-28 |
EP2344499A1 (fr) | 2011-07-20 |
CN102203094B (zh) | 2014-04-02 |
EA201170522A1 (ru) | 2011-12-30 |
ECSP11010946A (es) | 2011-05-31 |
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