SV2007002146A - Difenilimidazopirimidina e imidazol aminas como inhibidores de beta-secretasa ref. am101727 - Google Patents
Difenilimidazopirimidina e imidazol aminas como inhibidores de beta-secretasa ref. am101727Info
- Publication number
- SV2007002146A SV2007002146A SV2005002146A SV2005002146A SV2007002146A SV 2007002146 A SV2007002146 A SV 2007002146A SV 2005002146 A SV2005002146 A SV 2005002146A SV 2005002146 A SV2005002146 A SV 2005002146A SV 2007002146 A SV2007002146 A SV 2007002146A
- Authority
- SV
- El Salvador
- Prior art keywords
- beta
- secretasa
- difenylimidazopirimidine
- aminas
- imidazol
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, ***e
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
Abstract
LA PRESENTE INVENCION PROVEE UN COMPUESTO DE FORMULA I Y EL USO DEL MISMO PARA EL TRATAMIENTO TERAPEUTICO, PREVENCION O ALIVIO DE UNA ENFERMEDAD O TRASTORNO CARACTERIZADO POR DEPOSITOS BETA-AMILOIDES O NIVELES DE BETA-AMILOIDES ELEVADOS EN UN PACIENTE (VER FORMULA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58018704P | 2004-06-16 | 2004-06-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
SV2007002146A true SV2007002146A (es) | 2007-03-20 |
Family
ID=34982285
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SV2005002146A SV2007002146A (es) | 2004-06-16 | 2005-06-16 | Difenilimidazopirimidina e imidazol aminas como inhibidores de beta-secretasa ref. am101727 |
Country Status (24)
Country | Link |
---|---|
US (2) | US7456186B2 (es) |
EP (1) | EP1758907B1 (es) |
JP (1) | JP2008503460A (es) |
KR (1) | KR20070026811A (es) |
CN (1) | CN1997646A (es) |
AR (1) | AR049399A1 (es) |
AT (1) | ATE423121T1 (es) |
AU (1) | AU2005264917A1 (es) |
BR (1) | BRPI0512220A (es) |
CA (1) | CA2578600A1 (es) |
DE (1) | DE602005012825D1 (es) |
EC (1) | ECSP067080A (es) |
ES (1) | ES2321853T3 (es) |
GT (1) | GT200500157A (es) |
IL (1) | IL180018A0 (es) |
MX (1) | MXPA06014792A (es) |
NO (1) | NO20065847L (es) |
PA (1) | PA8637201A1 (es) |
PE (1) | PE20060299A1 (es) |
RU (1) | RU2006144075A (es) |
SV (1) | SV2007002146A (es) |
TW (1) | TW200602048A (es) |
WO (1) | WO2006009655A1 (es) |
ZA (1) | ZA200610593B (es) |
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TW200730523A (en) * | 2005-07-29 | 2007-08-16 | Wyeth Corp | Cycloalkyl amino-hydantoin compounds and use thereof for β-secretase modulation |
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JP5281794B2 (ja) | 2005-10-25 | 2013-09-04 | 塩野義製薬株式会社 | アミノジヒドロチアジン誘導体 |
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WO2007100536A1 (en) * | 2006-02-24 | 2007-09-07 | Wyeth | DIHYDROSPIRO[DIBENZO[A,D][7]ANNULENE-5,4'-IMIDAZOL] COMPOUNDS FOR THE INHIBITION OF β-SECRETASE |
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TW200808796A (en) * | 2006-06-14 | 2008-02-16 | Astrazeneca Ab | New compounds III |
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2005
- 2005-06-14 MX MXPA06014792A patent/MXPA06014792A/es active IP Right Grant
- 2005-06-14 AT AT05758187T patent/ATE423121T1/de not_active IP Right Cessation
- 2005-06-14 PE PE2005000678A patent/PE20060299A1/es not_active Application Discontinuation
- 2005-06-14 RU RU2006144075/04A patent/RU2006144075A/ru not_active Application Discontinuation
- 2005-06-14 WO PCT/US2005/020736 patent/WO2006009655A1/en active Application Filing
- 2005-06-14 CA CA002578600A patent/CA2578600A1/en not_active Abandoned
- 2005-06-14 KR KR1020077000970A patent/KR20070026811A/ko not_active Application Discontinuation
- 2005-06-14 EP EP05758187A patent/EP1758907B1/en active Active
- 2005-06-14 ES ES05758187T patent/ES2321853T3/es active Active
- 2005-06-14 DE DE602005012825T patent/DE602005012825D1/de active Active
- 2005-06-14 TW TW094119581A patent/TW200602048A/zh unknown
- 2005-06-14 JP JP2007516603A patent/JP2008503460A/ja active Pending
- 2005-06-14 AU AU2005264917A patent/AU2005264917A1/en not_active Abandoned
- 2005-06-14 CN CNA2005800194504A patent/CN1997646A/zh active Pending
- 2005-06-14 BR BRPI0512220-1A patent/BRPI0512220A/pt not_active IP Right Cessation
- 2005-06-15 US US11/152,925 patent/US7456186B2/en not_active Expired - Fee Related
- 2005-06-15 AR ARP050102450A patent/AR049399A1/es unknown
- 2005-06-15 PA PA20058637201A patent/PA8637201A1/es unknown
- 2005-06-16 GT GT200500157A patent/GT200500157A/es unknown
- 2005-06-16 SV SV2005002146A patent/SV2007002146A/es unknown
-
2006
- 2006-12-12 IL IL180018A patent/IL180018A0/en unknown
- 2006-12-13 EC EC2006007080A patent/ECSP067080A/es unknown
- 2006-12-15 ZA ZA200610593A patent/ZA200610593B/xx unknown
- 2006-12-18 NO NO20065847A patent/NO20065847L/no not_active Application Discontinuation
-
2008
- 2008-10-07 US US12/246,790 patent/US20090042912A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
IL180018A0 (en) | 2007-05-15 |
US20090042912A1 (en) | 2009-02-12 |
TW200602048A (en) | 2006-01-16 |
NO20065847L (no) | 2006-12-18 |
CN1997646A (zh) | 2007-07-11 |
PA8637201A1 (es) | 2006-06-02 |
RU2006144075A (ru) | 2008-07-27 |
ECSP067080A (es) | 2007-05-30 |
US7456186B2 (en) | 2008-11-25 |
AU2005264917A1 (en) | 2006-01-26 |
CA2578600A1 (en) | 2006-01-26 |
KR20070026811A (ko) | 2007-03-08 |
US20050282826A1 (en) | 2005-12-22 |
ZA200610593B (en) | 2009-09-30 |
WO2006009655A1 (en) | 2006-01-26 |
GT200500157A (es) | 2006-11-07 |
ATE423121T1 (de) | 2009-03-15 |
EP1758907B1 (en) | 2009-02-18 |
EP1758907A1 (en) | 2007-03-07 |
PE20060299A1 (es) | 2006-05-18 |
AR049399A1 (es) | 2006-07-26 |
JP2008503460A (ja) | 2008-02-07 |
BRPI0512220A (pt) | 2008-02-19 |
DE602005012825D1 (de) | 2009-04-02 |
MXPA06014792A (es) | 2007-02-16 |
ES2321853T3 (es) | 2009-06-12 |
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