GT200500157A - Difenilimidazopirimidina e imidazol aminas como inhibidores de beta-secretasa - Google Patents
Difenilimidazopirimidina e imidazol aminas como inhibidores de beta-secretasaInfo
- Publication number
- GT200500157A GT200500157A GT200500157A GT200500157A GT200500157A GT 200500157 A GT200500157 A GT 200500157A GT 200500157 A GT200500157 A GT 200500157A GT 200500157 A GT200500157 A GT 200500157A GT 200500157 A GT200500157 A GT 200500157A
- Authority
- GT
- Guatemala
- Prior art keywords
- secretasa
- difenylimidazopirimidine
- aminas
- imidazol
- inhibitors
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, ***e
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
Abstract
LA PRESENTE INVENCIÒN SE REFIERE A COMPUESTOS DE LA FÒRMULA GENERAL I EN LA QUE R1,R2,R3,R4,R5,R6,R7,R8,R9,R10,Z,Y,X,M,N, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS SON DE UTILIDAD EN LA ENFERMEDAD DE ALZHEIMER LA CUAL ES UNA ENFERMEDAD DEGENERATIVA PROGRESIVA DEL CEREBRO.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58018704P | 2004-06-16 | 2004-06-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
GT200500157A true GT200500157A (es) | 2006-11-07 |
Family
ID=34982285
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT200500157A GT200500157A (es) | 2004-06-16 | 2005-06-16 | Difenilimidazopirimidina e imidazol aminas como inhibidores de beta-secretasa |
Country Status (24)
Country | Link |
---|---|
US (2) | US7456186B2 (es) |
EP (1) | EP1758907B1 (es) |
JP (1) | JP2008503460A (es) |
KR (1) | KR20070026811A (es) |
CN (1) | CN1997646A (es) |
AR (1) | AR049399A1 (es) |
AT (1) | ATE423121T1 (es) |
AU (1) | AU2005264917A1 (es) |
BR (1) | BRPI0512220A (es) |
CA (1) | CA2578600A1 (es) |
DE (1) | DE602005012825D1 (es) |
EC (1) | ECSP067080A (es) |
ES (1) | ES2321853T3 (es) |
GT (1) | GT200500157A (es) |
IL (1) | IL180018A0 (es) |
MX (1) | MXPA06014792A (es) |
NO (1) | NO20065847L (es) |
PA (1) | PA8637201A1 (es) |
PE (1) | PE20060299A1 (es) |
RU (1) | RU2006144075A (es) |
SV (1) | SV2007002146A (es) |
TW (1) | TW200602048A (es) |
WO (1) | WO2006009655A1 (es) |
ZA (1) | ZA200610593B (es) |
Families Citing this family (77)
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US7592348B2 (en) | 2003-12-15 | 2009-09-22 | Schering Corporation | Heterocyclic aspartyl protease inhibitors |
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US7763609B2 (en) | 2003-12-15 | 2010-07-27 | Schering Corporation | Heterocyclic aspartyl protease inhibitors |
NZ552031A (en) * | 2004-06-16 | 2009-06-26 | Wyeth Corp | Amino-5,5-diphenylimidazolone derivatives for the inhibition of beta-secretase |
AR050184A1 (es) * | 2004-07-28 | 2006-10-04 | Schering Corp | Inhibidores macrociclicos de beta-secretasa |
JP2008526966A (ja) * | 2005-01-14 | 2008-07-24 | ワイス | β−セクレターゼの阻害のためのアミノ−イミダゾロン |
AU2006211159A1 (en) * | 2005-02-01 | 2006-08-10 | Wyeth | Amino-pyridines as inhibitors of beta-secretase |
BRPI0606902A2 (pt) * | 2005-02-14 | 2009-07-28 | Wyeth Corp | composto; método para o tratamento de uma doença ou distúrbio associado a atividade excessiva de bace em um paciente que dele necessite; método para modular a atividade de bace; composição farmacêutica |
TW200800959A (en) * | 2005-06-10 | 2008-01-01 | Wyeth Corp | Piperazine-piperidine antagonists and agonists of the 5-HT1a receptor |
ATE482214T1 (de) * | 2005-06-14 | 2010-10-15 | Schering Corp | Aspartylproteasehemmer |
US7759353B2 (en) * | 2005-06-14 | 2010-07-20 | Schering Corporation | Substituted spiro iminopyrimidinones as aspartyl protease inhibitors, compositions, and methods of treatment |
TWI332005B (en) | 2005-06-14 | 2010-10-21 | Schering Corp | Aspartyl protease inhibitors |
CA2610829A1 (en) | 2005-06-14 | 2006-12-28 | Schering Corporation | The preparation and use of compounds as aspartyl protease inhibitors |
US8722708B2 (en) | 2005-06-14 | 2014-05-13 | Merck Sharp & Dohme Inc. | Substituted isoindolines as aspartyl protease inhibitors |
MX2007016186A (es) * | 2005-06-14 | 2008-03-07 | Schering Corp | Preparacion y uso de inhibidores de proteasas. |
TW200738683A (en) * | 2005-06-30 | 2007-10-16 | Wyeth Corp | Amino-5-(5-membered)heteroarylimidazolone compounds and the use thereof for β-secretase modulation |
WO2007005404A1 (en) * | 2005-06-30 | 2007-01-11 | Wyeth | AMINO-5-(6-MEMBERED)HETEROARYLIMIDAZOLONE COMPOUNDS AND THE USE THEREOF FOR ß-SECRETASE MODULATION |
TW200730523A (en) * | 2005-07-29 | 2007-08-16 | Wyeth Corp | Cycloalkyl amino-hydantoin compounds and use thereof for β-secretase modulation |
TW200800213A (en) * | 2005-09-02 | 2008-01-01 | Abbott Lab | Novel imidazo based heterocycles |
BRPI0616757A2 (pt) * | 2005-09-26 | 2011-06-28 | Wyeth Corp | composto da fórmula i; processo para o tratamento de uma doença ou de um distúrbio associado com a atividade excessiva de bace; processo para a modulação da atividade de bace; processo para o tratamento da doença de alzheimer; e composição farmacêutica |
ES2537898T3 (es) | 2005-10-25 | 2015-06-15 | Shionogi & Co., Ltd. | Derivados de aminotiazolidina y aminotetrahidrotiazepina como inhibidores de BACE 1 |
CA2634037A1 (en) * | 2005-12-19 | 2007-07-12 | Wyeth | 2-amino-5-piperidinylimidazolone compounds and use thereof for .beta.-secretase modulation |
WO2007100536A1 (en) * | 2006-02-24 | 2007-09-07 | Wyeth | DIHYDROSPIRO[DIBENZO[A,D][7]ANNULENE-5,4'-IMIDAZOL] COMPOUNDS FOR THE INHIBITION OF β-SECRETASE |
TW200808741A (en) * | 2006-06-09 | 2008-02-16 | Wyeth Corp | 6-methoxy-8-[4-(1-(5-fluoro)-quinolin-8-yl-piperidin-4-yl)-piperazin-1-yl]-quinoline hydrochloric acid salts |
TW200808796A (en) * | 2006-06-14 | 2008-02-16 | Astrazeneca Ab | New compounds III |
TW200815449A (en) * | 2006-06-14 | 2008-04-01 | Astrazeneca Ab | Novel compounds II |
TW200815447A (en) * | 2006-06-14 | 2008-04-01 | Astrazeneca Ab | Novel compounds IV |
TW200815443A (en) * | 2006-06-14 | 2008-04-01 | Astrazeneca Ab | Novel compounds I |
TW200815349A (en) | 2006-06-22 | 2008-04-01 | Astrazeneca Ab | New compounds |
US7700606B2 (en) * | 2006-08-17 | 2010-04-20 | Wyeth Llc | Imidazole amines as inhibitors of β-secretase |
TW200817406A (en) * | 2006-08-17 | 2008-04-16 | Wyeth Corp | Imidazole amines as inhibitors of β-secretase |
MX2009003102A (es) * | 2006-09-21 | 2009-04-01 | Wyeth Corp | INDOLILALQUILPIRIDIN-2-AMINAS PARA LA INHIBICION DE ß-SECRETASA. |
WO2008063114A1 (en) * | 2006-11-20 | 2008-05-29 | Astrazeneca Ab | Amino- imidazolones and their use as medicament for treating cognitive impairment alzheimer disease, neurodegeneration and dementia |
TW200831096A (en) * | 2006-11-28 | 2008-08-01 | Wyeth Corp | Metabolites of 5-Fluoro-8-{4-[4-(6-methoxyquinolin-8-yl)piperazin-1-yl]piperidin-1-yl} quinoline and methods of preparation and uses thereof |
WO2008073365A1 (en) | 2006-12-12 | 2008-06-19 | Schering Corporation | Aspartyl protease inhibitors |
CA2672295A1 (en) * | 2006-12-12 | 2008-06-19 | Schering Corporation | Aspartyl protease inhibitors containing a tricyclic ring system |
CL2008000119A1 (es) * | 2007-01-16 | 2008-05-16 | Wyeth Corp | Compuestos derivados de pirazol, antagonistas del receptor nicotinico de acetilcolina; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como demencia senil, alzheimer y esquizofrenia. |
PE20090160A1 (es) * | 2007-03-20 | 2009-02-11 | Wyeth Corp | COMPUESTOS AMINO-5-[4-(DIFLUOROMETOXI)FENIL SUSTITUIDO]-5-FENILIMIDAZOLONA COMO INHIBIDORES DE ß-SECRETASA |
AR065814A1 (es) * | 2007-03-23 | 2009-07-01 | Wyeth Corp | Derivados de 5-fenilimidazolona,inhibidores de beta-secretasa,composiciones farmaceuticas que los contienen y usos para prevenir y/o tratar trastornos asociados a niveles beta-amiloides elevados. |
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US8637504B2 (en) | 2008-06-13 | 2014-01-28 | Shionogi & Co., Ltd. | Sulfur-containing heterocyclic derivative having beta secretase inhibitory activity |
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JP5417860B2 (ja) * | 2008-08-26 | 2014-02-19 | 住友化学株式会社 | α−ヒドロキシエステル類の製造方法 |
JPWO2010047372A1 (ja) | 2008-10-22 | 2012-03-22 | 塩野義製薬株式会社 | Bace1阻害活性を有する2−アミノピリミジン−4−オンおよび2−アミノピリジン誘導体 |
WO2010056195A1 (en) * | 2008-11-14 | 2010-05-20 | Astrazeneca Ab | New compounds 575 |
TW201020244A (en) | 2008-11-14 | 2010-06-01 | Astrazeneca Ab | New compounds |
US20100125081A1 (en) * | 2008-11-14 | 2010-05-20 | Astrazeneca Ab | New compounds 574 |
SG173466A1 (en) | 2009-03-13 | 2011-09-29 | Vitae Pharmaceuticals Inc | Inhibitors of beta-secretase |
EP2281824A1 (en) | 2009-08-07 | 2011-02-09 | Noscira, S.A. | Furan-imidazolone derivatives, for the treatment of cognitive, neurodegenerative or neuronal diseases or disorders |
US8563543B2 (en) | 2009-10-08 | 2013-10-22 | Merck Sharp & Dohme Corp. | Iminothiadiazine dioxide compounds as bace inhibitors, compositions, and their use |
US8569310B2 (en) | 2009-10-08 | 2013-10-29 | Merck Sharp & Dohme Corp. | Pentafluorosulfur imino heterocyclic compounds as BACE-1 inhibitors, compositions and their use |
UA108363C2 (uk) | 2009-10-08 | 2015-04-27 | Похідні імінотіадіазиндіоксиду як інгібітори bace, композиція на їх основі і їх застосування | |
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JP5816630B2 (ja) | 2010-10-29 | 2015-11-18 | 塩野義製薬株式会社 | ナフチリジン誘導体 |
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BR112014004181A2 (pt) | 2011-08-22 | 2017-06-13 | Merck Sharp & Dohme | composto, composição farmacêutica, e, método de tratamento, prevenção, e / ou retardo do início de uma doença ou patologia |
TWI557112B (zh) | 2012-03-05 | 2016-11-11 | 百靈佳殷格翰國際股份有限公司 | β-分泌酶抑制劑 |
AU2013235422B2 (en) | 2012-03-19 | 2016-12-15 | Buck Institute For Research On Aging | APP specific BACE inhibitors (ASBIs) and uses thereof |
TW201422592A (zh) | 2012-08-27 | 2014-06-16 | Boehringer Ingelheim Int | β-分泌酶抑制劑 |
JP2015532282A (ja) | 2012-09-28 | 2015-11-09 | ヴァイティー ファーマシューティカルズ,インコーポレイテッド | β−セクレターゼの阻害剤 |
WO2014062549A1 (en) | 2012-10-17 | 2014-04-24 | Merck Sharp & Dohme Corp. | Tricyclic substituted thiadiazine dioxide compounds as bace inhibitors, compositions, and their use |
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EP2956443B1 (en) | 2013-02-12 | 2019-09-25 | Buck Institute For Research On Aging | Hydantoins that modulate bace-mediated app processing |
KR101668857B1 (ko) | 2015-01-08 | 2016-10-24 | 한양대학교 에리카산학협력단 | 이미다졸-1-일 피리미딘 유도체, 또는 이의 약학적으로 허용가능한 염 및 이를 유효성분으로 포함하는 약학적 조성물 |
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US7700606B2 (en) | 2006-08-17 | 2010-04-20 | Wyeth Llc | Imidazole amines as inhibitors of β-secretase |
-
2005
- 2005-06-14 JP JP2007516603A patent/JP2008503460A/ja active Pending
- 2005-06-14 MX MXPA06014792A patent/MXPA06014792A/es active IP Right Grant
- 2005-06-14 AT AT05758187T patent/ATE423121T1/de not_active IP Right Cessation
- 2005-06-14 BR BRPI0512220-1A patent/BRPI0512220A/pt not_active IP Right Cessation
- 2005-06-14 CA CA002578600A patent/CA2578600A1/en not_active Abandoned
- 2005-06-14 CN CNA2005800194504A patent/CN1997646A/zh active Pending
- 2005-06-14 PE PE2005000678A patent/PE20060299A1/es not_active Application Discontinuation
- 2005-06-14 TW TW094119581A patent/TW200602048A/zh unknown
- 2005-06-14 RU RU2006144075/04A patent/RU2006144075A/ru not_active Application Discontinuation
- 2005-06-14 WO PCT/US2005/020736 patent/WO2006009655A1/en active Application Filing
- 2005-06-14 DE DE602005012825T patent/DE602005012825D1/de active Active
- 2005-06-14 EP EP05758187A patent/EP1758907B1/en active Active
- 2005-06-14 ES ES05758187T patent/ES2321853T3/es active Active
- 2005-06-14 AU AU2005264917A patent/AU2005264917A1/en not_active Abandoned
- 2005-06-14 KR KR1020077000970A patent/KR20070026811A/ko not_active Application Discontinuation
- 2005-06-15 PA PA20058637201A patent/PA8637201A1/es unknown
- 2005-06-15 US US11/152,925 patent/US7456186B2/en not_active Expired - Fee Related
- 2005-06-15 AR ARP050102450A patent/AR049399A1/es unknown
- 2005-06-16 GT GT200500157A patent/GT200500157A/es unknown
- 2005-06-16 SV SV2005002146A patent/SV2007002146A/es unknown
-
2006
- 2006-12-12 IL IL180018A patent/IL180018A0/en unknown
- 2006-12-13 EC EC2006007080A patent/ECSP067080A/es unknown
- 2006-12-15 ZA ZA200610593A patent/ZA200610593B/xx unknown
- 2006-12-18 NO NO20065847A patent/NO20065847L/no not_active Application Discontinuation
-
2008
- 2008-10-07 US US12/246,790 patent/US20090042912A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
TW200602048A (en) | 2006-01-16 |
AU2005264917A1 (en) | 2006-01-26 |
RU2006144075A (ru) | 2008-07-27 |
PE20060299A1 (es) | 2006-05-18 |
PA8637201A1 (es) | 2006-06-02 |
JP2008503460A (ja) | 2008-02-07 |
BRPI0512220A (pt) | 2008-02-19 |
NO20065847L (no) | 2006-12-18 |
WO2006009655A1 (en) | 2006-01-26 |
CA2578600A1 (en) | 2006-01-26 |
KR20070026811A (ko) | 2007-03-08 |
ES2321853T3 (es) | 2009-06-12 |
MXPA06014792A (es) | 2007-02-16 |
ECSP067080A (es) | 2007-05-30 |
DE602005012825D1 (de) | 2009-04-02 |
IL180018A0 (en) | 2007-05-15 |
EP1758907B1 (en) | 2009-02-18 |
US7456186B2 (en) | 2008-11-25 |
US20050282826A1 (en) | 2005-12-22 |
EP1758907A1 (en) | 2007-03-07 |
AR049399A1 (es) | 2006-07-26 |
CN1997646A (zh) | 2007-07-11 |
ATE423121T1 (de) | 2009-03-15 |
SV2007002146A (es) | 2007-03-20 |
US20090042912A1 (en) | 2009-02-12 |
ZA200610593B (en) | 2009-09-30 |
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