SE398751B - Analogiforfarande for framstellning av pyrazolo/1,5-a/pyrimidiner - Google Patents

Analogiforfarande for framstellning av pyrazolo/1,5-a/pyrimidiner

Info

Publication number: SE398751B
Authority: SE; Sweden
Prior art keywords: pyrimidines; preparing pyrazolo; analogical procedure; analogical; procedure
Prior art date: 1971-12-09

Application number

SE7215829A

Other languages

English (en)

Swedish (sv)

Inventor

R K Robins

D E O'brien

T Novinson

R H Springer

Original Assignee

Icn Pharmaceuticals

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1971-12-09

Filing date

1972-12-05

Publication date

1978-01-16

1972-04-20 Priority claimed from US245870A external-priority patent/US3925385A/en

1972-12-05 Application filed by Icn Pharmaceuticals filed Critical Icn Pharmaceuticals

1978-01-16 Publication of SE398751B publication Critical patent/SE398751B/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

SE7215829A 1971-12-09 1972-12-05 Analogiforfarande for framstellning av pyrazolo/1,5-a/pyrimidiner SE398751B (sv)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US20653871A	1971-12-09	1971-12-09
US245870A US3925385A (en)	1972-04-20	1972-04-20	6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines
US27346572A	1972-07-20	1972-07-20
US29984072A	1972-10-24	1972-10-24

Publications (1)

Publication Number	Publication Date
SE398751B true SE398751B (sv)	1978-01-16

Family

ID=27498614

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE7215829A SE398751B (sv)	1971-12-09	1972-12-05	Analogiforfarande for framstellning av pyrazolo/1,5-a/pyrimidiner

Country Status (15)

Country	Link
JP (1)	JPS4864097A (de)
BE (1)	BE792533A (de)
BG (1)	BG22401A3 (de)
CH (1)	CH603652A5 (de)
DD (1)	DD104530A5 (de)
DE (1)	DE2257547A1 (de)
GB (1)	GB1412017A (de)
HU (1)	HU168530B (de)
IE (1)	IE37189B1 (de)
IL (1)	IL40895A (de)
LU (1)	LU66597A1 (de)
NL (1)	NL7216539A (de)
NO (1)	NO137012C (de)
RO (1)	RO62762A (de)
SE (1)	SE398751B (de)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4281000A (en) *	1979-07-09	1981-07-28	American Cyanamid Company	Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents
AU557300B2 (en) *	1982-03-16	1986-12-18	Farmitalia Carlo Erba S.P.A.	Substituted 1h-pyrazolo(1,5-alpha)pyrimidines and processes for their preparation
ZA831407B (en) *	1982-03-25	1983-11-30	Erba Farmitalia	Substituted ethenyl derivatives of 1h-pyrazolo(1,5-a)pyrimidine and process for their preparation
NZ208554A (en) *	1983-06-23	1987-06-30	American Cyanamid Co	(aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions
DE3533050A1 (de) *	1985-09-17	1987-03-26	Basf Ag	7-amino-azolo(1,5-a)pyrimidine, verfahren zu ihrer herstellung und diese enthaltende fungizide, bzw. deren verwendung als fungizide
CA1330079C (en) *	1988-10-13	1994-06-07	Michihiko Tsujitani	Pyrrolo (3,2-e)pyrazolo(1,5-a)pyrimidine derivative and medicine comprising the same
CA2107479C (en) *	1991-04-22	1997-12-16	Makoto Inoue	Pyrazolo[1,5-a]pyrimidine derivatives and anti-inflammatory agent containing the same
DE4333705C2 (de) *	1993-10-02	2003-10-30	Guenter Ege	Arylmethylsubstituierte Pyrazolo-azine, insbesondere 3-Arylmethylpyrazolo[1,5-a]pyrimidine und Verfahren zur Herstellung von 8-Arylmethyl-pyrazolo[5,1-c][1,2,4]triazinen
CA2169719C (en) *	1994-06-21	2002-04-16	Yasuo Shoji	Pyrazolo[1,5-a]pyrimidine derivative
KR100260292B1 (ko) *	1995-09-28	2000-07-01	오쓰카 요시미쓰	진통제
FR2771631B1 (fr) *	1997-12-03	2001-02-02	Oreal	Compositions de teinture des fibres keratiniques contenant des 3-amino pyrazolo-[1,5-a]-pyrimidines, procede de teinture, nouvelles 3-amino pyrazolo- [1,5-a]-pyrimidines et leur procede de preparation
US7119200B2 (en) *	2002-09-04	2006-10-10	Schering Corporation	Pyrazolopyrimidines as cyclin dependent kinase inhibitors
US7161003B1 (en) *	2002-09-04	2007-01-09	Schering Corporation	Pyrazolopyrimidines as cyclin dependent kinase inhibitors
KR101088922B1 (ko) *	2002-09-04	2011-12-01	파마코페이아, 엘엘씨.	사이클린 의존성 키나제 억제제로서의 피라졸로피리미딘
TWI252851B (en) *	2003-07-24	2006-04-11	Ferrer Int	7-substituted 3-nitro-pyrazolo[1,5-a]pyrimidines and compositions and methods related thereto
ES2222813B1 (es) *	2003-07-24	2005-12-16	Ferrer Internacional, S.A.	N-(3-(3-sustituidas-pirazolo(1,5-a)pirimidin-7-il)-fenil)-sulfonamidas y composiciones y metodos relacionados.
ES2619125T3 (es)	2013-04-25	2017-06-23	Beigene, Ltd.	Compuestos heterocíclicos fusionados como inhibidores de proteína cinasa
HRP20221262T1 (hr)	2013-09-13	2022-12-09	Beigene Switzerland Gmbh	Protutijela anti-pd1 i njihova uporaba kao terapeutskih i dijagnostičkih sredstava
WO2016000619A1 (en)	2014-07-03	2016-01-07	Beigene, Ltd.	Anti-pd-l1 antibodies and their use as therapeutics and diagnostics
AU2017293423B2 (en)	2016-07-05	2023-05-25	Beigene, Ltd.	Combination of a PD-1 antagonist and a RAF inhibitor for treating cancer
CN116478166A (zh)	2016-08-16	2023-07-25	百济神州(苏州)生物科技有限公司	一种化合物的晶型、其制备和用途
EP3500299B1 (de)	2016-08-19	2023-12-13	BeiGene Switzerland GmbH	Kombination von zanubrutinib mit einem anti-cd20 oder anti-pd-1 antikörper zur verwendung in der behandlung von krebs
US11555038B2 (en)	2017-01-25	2023-01-17	Beigene, Ltd.	Crystalline forms of (S)-7-(1-(but-2-ynoyl)piperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof
CN110799543A (zh)	2017-06-26	2020-02-14	百济神州有限公司	肝细胞癌的免疫治疗
US11377449B2 (en)	2017-08-12	2022-07-05	Beigene, Ltd.	BTK inhibitors with improved dual selectivity
CN111801334B (zh)	2017-11-29	2023-06-09	百济神州瑞士有限责任公司	使用包含btk抑制剂的组合治疗惰性或侵袭性b-细胞淋巴瘤
US11786531B1 (en)	2022-06-08	2023-10-17	Beigene Switzerland Gmbh	Methods of treating B-cell proliferative disorder

0
- BE BE792533D patent/BE792533A/xx unknown
1972
- 1972-11-21 IE IE1612/72A patent/IE37189B1/xx unknown
- 1972-11-22 IL IL40895A patent/IL40895A/en unknown
- 1972-11-23 DE DE2257547A patent/DE2257547A1/de active Pending
- 1972-12-01 GB GB5558772A patent/GB1412017A/en not_active Expired
- 1972-12-05 SE SE7215829A patent/SE398751B/xx unknown
- 1972-12-05 LU LU66597A patent/LU66597A1/xx unknown
- 1972-12-06 CH CH1775172A patent/CH603652A5/xx not_active IP Right Cessation
- 1972-12-06 NL NL7216539A patent/NL7216539A/xx not_active Application Discontinuation
- 1972-12-06 NO NO4476/72A patent/NO137012C/no unknown
- 1972-12-07 DD DD167370A patent/DD104530A5/xx unknown
- 1972-12-08 HU HUIE548A patent/HU168530B/hu unknown
- 1972-12-09 RO RO7200073093A patent/RO62762A/ro unknown
- 1972-12-09 BG BG22071A patent/BG22401A3/xx unknown
- 1972-12-09 JP JP47123877A patent/JPS4864097A/ja active Pending

Also Published As

Publication number	Publication date
DE2257547A1 (de)	1973-06-14
IE37189B1 (en)	1977-05-25
IL40895A0 (en)	1973-01-30
JPS4864097A (de)	1973-09-05
IE37189L (en)	1973-06-09
HU168530B (de)	1976-05-28
DD104530A5 (de)	1974-03-12
RO62762A (fr)	1978-05-15
NO137012C (no)	1977-12-14
LU66597A1 (de)	1973-03-15
NL7216539A (de)	1973-06-13
CH603652A5 (de)	1978-08-31
BG22401A3 (de)	1977-02-20
IL40895A (en)	1976-12-31
NO137012B (no)	1977-09-05
BE792533A (fr)	1973-06-08
GB1412017A (en)	1975-10-29

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