PT97505A - Processo para a preparacao de composicoes farmaceuticas para administracao transdermica, contendo 1-(4-etilfenil)-2-metil-3-(1-piperidinil)-1-propanona (eperisona) ou 2-metil-1-(4-metilfenil)-3-(1-piperidinil)-1-propanona (tolperisona) ou um dos seus sais, como ingrediente activo - Google Patents

Processo para a preparacao de composicoes farmaceuticas para administracao transdermica, contendo 1-(4-etilfenil)-2-metil-3-(1-piperidinil)-1-propanona (eperisona) ou 2-metil-1-(4-metilfenil)-3-(1-piperidinil)-1-propanona (tolperisona) ou um dos seus sais, como ingrediente activo

Info

Publication number
PT97505A
PT97505A PT97505A PT9750591A PT97505A PT 97505 A PT97505 A PT 97505A PT 97505 A PT97505 A PT 97505A PT 9750591 A PT9750591 A PT 9750591A PT 97505 A PT97505 A PT 97505A
Authority
PT
Portugal
Prior art keywords
piperidinyl
methyl
eperisone
tolperisone
propanean
Prior art date
Application number
PT97505A
Other languages
English (en)
Other versions
PT97505B (pt
Inventor
Masato Azuma
Tsutomu Negama
Mitsuhiro Yoshida
Hiroyuki Fujimori
Original Assignee
Eisai Co Ltd
Seikisui Chemical Co Ltd
Sansho Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai Co Ltd, Seikisui Chemical Co Ltd, Sansho Co filed Critical Eisai Co Ltd
Publication of PT97505A publication Critical patent/PT97505A/pt
Publication of PT97505B publication Critical patent/PT97505B/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Inorganic Chemistry (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
PT97505A 1990-04-27 1991-04-26 Processo para a preparacao de composicoes farmaceuticas para administracao transdermica, contendo 1-(4-etilfenil)-2-metil-3-(1-piperidinil)-1-propanona (eperisona) ou 2-metil-1-(4-metilfenil)-3-(1-piperidinil)-1-propanona (tolperisona) ou um dos seus sais, como ingrediente activo PT97505B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP11279290 1990-04-27

Publications (2)

Publication Number Publication Date
PT97505A true PT97505A (pt) 1992-01-31
PT97505B PT97505B (pt) 1998-08-31

Family

ID=14595632

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97505A PT97505B (pt) 1990-04-27 1991-04-26 Processo para a preparacao de composicoes farmaceuticas para administracao transdermica, contendo 1-(4-etilfenil)-2-metil-3-(1-piperidinil)-1-propanona (eperisona) ou 2-metil-1-(4-metilfenil)-3-(1-piperidinil)-1-propanona (tolperisona) ou um dos seus sais, como ingrediente activo

Country Status (11)

Country Link
EP (1) EP0454089B1 (pt)
JP (1) JP3170304B2 (pt)
KR (1) KR930007407B1 (pt)
CN (1) CN1049817C (pt)
AT (1) ATE109980T1 (pt)
CA (1) CA2041330C (pt)
DE (1) DE69103459T2 (pt)
DK (1) DK0454089T3 (pt)
ES (1) ES2058977T3 (pt)
MY (1) MY115126A (pt)
PT (1) PT97505B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5252334A (en) * 1989-09-08 1993-10-12 Cygnus Therapeutic Systems Solid matrix system for transdermal drug delivery
JPH06247846A (ja) * 1993-02-22 1994-09-06 Toko Yakuhin Kogyo Kk 塩酸リトドリンの経皮吸収製剤用組成物
AU7396294A (en) 1993-06-25 1995-01-24 Alza Corporation Incorporating poly-n-vinyl amide in a transdermal system
CN1188189C (zh) * 1995-06-07 2005-02-09 奥瑟-麦内尔制药公司 基质层含有17-脱乙酰基诺孕酯的经皮贴片及基质的用途
AT409083B (de) * 1999-04-01 2002-05-27 Sanochemia Pharmazeutika Ag Pharmazeutische, tolperison enthaltende zubereitung zur oralen verabreichung
JP5209433B2 (ja) * 2007-10-19 2013-06-12 日東電工株式会社 貼付製剤
US20100266670A1 (en) * 2007-12-10 2010-10-21 Akira Yamamoto Transdermally absorptive preparation
JP5631854B2 (ja) * 2010-12-13 2014-11-26 久光製薬株式会社 医薬組成物および貼付剤
KR20140118410A (ko) * 2013-03-29 2014-10-08 초당약품공업 주식회사 저장 및 pH 안정성이 개선된 에페리손 의약 조성물
US10300025B2 (en) * 2016-07-27 2019-05-28 Corium, Inc. Donepezil transdermal delivery system
WO2020086046A2 (en) * 2018-10-26 2020-04-30 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Topical compositions comprising tolperisone and flurbiprofen combination

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL61721A (en) * 1980-12-16 1984-03-30 Blank Izhak Nitroglycerin preparations
AU563054B2 (en) * 1984-10-24 1987-06-25 Sekisui Kagaku Kogyo Kabushiki Kaisha Percutaneous tape of isdn
JPH0720866B2 (ja) * 1987-05-15 1995-03-08 三生製薬株式会社 エペリゾン又はトルペリゾン或いはそれらの塩類含有経皮適用製剤

Also Published As

Publication number Publication date
CA2041330C (en) 1996-05-28
JPH04217919A (ja) 1992-08-07
EP0454089A1 (en) 1991-10-30
PT97505B (pt) 1998-08-31
CN1056055A (zh) 1991-11-13
KR930007407B1 (ko) 1993-08-10
CN1049817C (zh) 2000-03-01
MY115126A (en) 2003-04-30
JP3170304B2 (ja) 2001-05-28
ES2058977T3 (es) 1994-11-01
DE69103459D1 (de) 1994-09-22
EP0454089B1 (en) 1994-08-17
KR910018024A (ko) 1991-11-30
DK0454089T3 (da) 1994-09-19
DE69103459T2 (de) 1995-01-19
CA2041330A1 (en) 1991-10-28
ATE109980T1 (de) 1994-09-15

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Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19910916

FG3A Patent granted, date of granting

Effective date: 19980514