PL2781519T3 - Nowa przeciwwirusowa pochodna pirolopirydyny i sposób jej wytwarzania - Google Patents

Nowa przeciwwirusowa pochodna pirolopirydyny i sposób jej wytwarzania

Info

Publication number
PL2781519T3
PL2781519T3 PL12849140T PL12849140T PL2781519T3 PL 2781519 T3 PL2781519 T3 PL 2781519T3 PL 12849140 T PL12849140 T PL 12849140T PL 12849140 T PL12849140 T PL 12849140T PL 2781519 T3 PL2781519 T3 PL 2781519T3
Authority
PL
Poland
Prior art keywords
same
production method
novel antiviral
pyrrolopyridine derivative
pyrrolopyridine
Prior art date
Application number
PL12849140T
Other languages
English (en)
Inventor
Jong Chan Son
Bong Jin Kim
Jae Hak Kim
Ill Young Lee
Chang Soo Yun
Sang Ho Lee
Chong Kgo Lee
Original Assignee
St Pharm Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by St Pharm Co., Ltd. filed Critical St Pharm Co., Ltd.
Publication of PL2781519T3 publication Critical patent/PL2781519T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
PL12849140T 2011-11-15 2012-11-15 Nowa przeciwwirusowa pochodna pirolopirydyny i sposób jej wytwarzania PL2781519T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR20110119102 2011-11-15
EP12849140.4A EP2781519B1 (en) 2011-11-15 2012-11-15 Novel antiviral pyrrolopyridine derivative and a production method for same
PCT/KR2012/009689 WO2013073875A1 (ko) 2011-11-15 2012-11-15 신규한 항바이러스성 피롤로피리딘 유도체 및 이의 제조방법

Publications (1)

Publication Number Publication Date
PL2781519T3 true PL2781519T3 (pl) 2020-06-29

Family

ID=48429876

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12849140T PL2781519T3 (pl) 2011-11-15 2012-11-15 Nowa przeciwwirusowa pochodna pirolopirydyny i sposób jej wytwarzania

Country Status (11)

Country Link
US (1) US9499537B2 (pl)
EP (1) EP2781519B1 (pl)
JP (1) JP5893156B2 (pl)
KR (1) KR101467477B1 (pl)
CN (1) CN104066732B (pl)
DK (1) DK2781519T3 (pl)
ES (1) ES2760981T3 (pl)
HU (1) HUE046795T2 (pl)
PL (1) PL2781519T3 (pl)
PT (1) PT2781519T (pl)
WO (1) WO2013073875A1 (pl)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2877468B1 (en) 2012-07-12 2017-08-23 ViiV Healthcare UK Limited Compounds and methods for treating hiv
TW201441197A (zh) 2013-01-31 2014-11-01 Shionogi & Co Hiv複製抑制劑
EP2821082A1 (en) 2013-07-05 2015-01-07 Laboratoire Biodim Method of producing an inactivated lentivirus, especially HIV, vaccine, kit and method of use
WO2015123230A1 (en) 2014-02-12 2015-08-20 Bristol-Myers Squibb Company Benzothiazole macrocycles as inhibitors of human immunodeficiency virus replication
WO2015126743A1 (en) 2014-02-18 2015-08-27 Bristol-Myers Squibb Company Pyrazolopyrimidine macrocycles as inhibitors of human immunodeficiency virus replication
US9409922B2 (en) 2014-02-18 2016-08-09 Bristol-Myers Squibb Company Imidazopyridine macrocycles as inhibitors of human immunodeficiency virus replication
EP3116879A1 (en) 2014-02-18 2017-01-18 VIIV Healthcare UK (No.5) Limited Imidazopyrimidine macrocycles as inhibitors of human immunodeficiency virus replication
US9273067B2 (en) 2014-02-19 2016-03-01 Bristol-Myers Squibb Company Pyrazolopyrimidine macrocycles as inhibitors of human immunodeficiency virus replication
JP6579549B2 (ja) 2014-05-16 2019-09-25 塩野義製薬株式会社 Hiv複製阻害作用を有する3環性複素環誘導体
KR101592370B1 (ko) * 2014-06-09 2016-02-11 한국화학연구원 신규한 피롤로피리딘 유도체 및 이의 hiv 저해제로서의 용도
CN104478911A (zh) * 2014-12-19 2015-04-01 成都安斯利生物医药有限公司 一种制备3-三氟甲基吡咯硼酸的方法
CA2987384A1 (en) 2015-05-29 2016-12-08 Shionogi & Co., Ltd. Nitrogen-containing tricyclic derivative having hiv replication inhibitory activity
PT3604303T (pt) * 2017-03-24 2023-02-14 St Pharm Co Ltd Novo derivado de pirrolopiridina, método para a produção do mesmo e utilizações do mesmo
AU2018243463C1 (en) 2017-03-29 2022-12-01 Siteone Therapeutics, Inc. 11,13-modified saxitoxins for the treatment of pain
JP7096686B2 (ja) * 2017-03-30 2022-07-06 住友化学株式会社 アミノ基を有する有機リチウム化合物およびその中間体の製造方法、並びに有機リチウム化合物を用いた共役ジエン系重合体の製造方法
TW202140495A (zh) 2020-01-10 2021-11-01 大陸商江蘇恆瑞醫藥股份有限公司 三環四氫異喹啉類衍生物、其製備方法及其在醫藥上的應用
KR20220023187A (ko) * 2020-08-20 2022-03-02 에스티팜 주식회사 피롤로피리딘 유도체 및 이들의 용도
EP4276101A1 (en) 2021-01-11 2023-11-15 ST Pharm Co., Ltd. Pyrrolopyridine derivative preparation method

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005103003A2 (en) * 2004-04-26 2005-11-03 Pfizer Inc. Pyrrolopyridine derivatives and their use as hiv-integrase inhibitors
DE102004060659A1 (de) * 2004-12-15 2006-07-06 Lanxess Deutschland Gmbh Neue substituierte 1H-Pyrrolo[2,3-b]pyridine und deren Herstellung
US7939545B2 (en) * 2006-05-16 2011-05-10 Boehringer Ingelheim International Gmbh Inhibitors of human immunodeficiency virus replication
GB0710528D0 (en) * 2007-06-01 2007-07-11 Glaxo Group Ltd Novel compounds
EP2220095B1 (en) * 2007-11-15 2013-01-02 Gilead Sciences, Inc. Inhibitors of human immunodeficiency virus replication
UA100250C2 (uk) * 2007-11-16 2012-12-10 Гілеад Сайнсіз, Інк. Інгібітори реплікації вірусу імунодефіциту людини
EP2220084B1 (en) * 2007-11-16 2014-02-19 Gilead Sciences, Inc. Inhibitors of human immunodeficiency virus replication
US8338441B2 (en) 2009-05-15 2012-12-25 Gilead Sciences, Inc. Inhibitors of human immunodeficiency virus replication
GB0908394D0 (en) * 2009-05-15 2009-06-24 Univ Leuven Kath Novel viral replication inhibitors
WO2012102985A1 (en) * 2011-01-24 2012-08-02 Glaxosmithkline Llc Isoquinoline compounds and methods for treating hiv
WO2013012649A1 (en) * 2011-07-15 2013-01-24 Glaxosmithkline Llc Azaindole compounds and methods for treating hiv

Also Published As

Publication number Publication date
EP2781519B1 (en) 2019-10-30
US9499537B2 (en) 2016-11-22
PT2781519T (pt) 2019-12-17
ES2760981T3 (es) 2020-05-18
EP2781519A4 (en) 2015-06-24
US20140249162A1 (en) 2014-09-04
CN104066732A (zh) 2014-09-24
CN104066732B (zh) 2016-04-13
EP2781519A1 (en) 2014-09-24
KR101467477B1 (ko) 2014-12-02
DK2781519T3 (da) 2019-12-16
JP2014533298A (ja) 2014-12-11
KR20130054211A (ko) 2013-05-24
HUE046795T2 (hu) 2020-03-30
WO2013073875A1 (ko) 2013-05-23
JP5893156B2 (ja) 2016-03-23

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