PA8852901A1 - Inhibidores de proteina cinasa - Google Patents

Inhibidores de proteina cinasa

Info

Publication number
PA8852901A1
PA8852901A1 PA20098852901A PA8852901A PA8852901A1 PA 8852901 A1 PA8852901 A1 PA 8852901A1 PA 20098852901 A PA20098852901 A PA 20098852901A PA 8852901 A PA8852901 A PA 8852901A PA 8852901 A1 PA8852901 A1 PA 8852901A1
Authority
PA
Panama
Prior art keywords
protein
cinase
inhibitors
cinase inhibitors
salt
Prior art date
Application number
PA20098852901A
Other languages
English (en)
Inventor
Andrew Coates David
De Dios Magana Alfonso
De Prado Ana
Filadelfa Del Prado Catalina Miriam
Garcia Paredes Cristina
Mark Gelbert Lawrence
Monte Knobeloch John
Maria Martin De La Nava Eva
Dolores Martin Ortega Finger Maria
Antonio Martinez Perez Jose
Isabel Mateo Herranz Ana
Perez Martinez Carlos
Sanchez Martinez Concepcion
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42267022&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PA8852901(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PA8852901A1 publication Critical patent/PA8852901A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

LA PRESENTE INVENCIÓN SE REFIERE A UN COMPUESTO DE FÓRMULA(I):O UNA SAL DEL MISMO FARMACÉUTICAMENTE ACEPTABLE,EL CUAL ES ÚTIL EN EL TRATAMIENTO DE ENFERMEDADES PROLIFERATIVAS CELULARES.
PA20098852901A 2008-12-22 2009-12-09 Inhibidores de proteina cinasa PA8852901A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08380343 2008-12-22
US15495409P 2009-02-24 2009-02-24

Publications (1)

Publication Number Publication Date
PA8852901A1 true PA8852901A1 (es) 2010-07-27

Family

ID=42267022

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20098852901A PA8852901A1 (es) 2008-12-22 2009-12-09 Inhibidores de proteina cinasa

Country Status (41)

Country Link
US (1) US7855211B2 (es)
EP (1) EP2379528B1 (es)
JP (1) JP5417453B2 (es)
KR (1) KR101297497B1 (es)
CN (1) CN102264725B (es)
AR (1) AR074575A1 (es)
AU (1) AU2009330365B2 (es)
BR (1) BRPI0924183B8 (es)
CA (1) CA2747055C (es)
CO (1) CO6382125A2 (es)
CR (1) CR20110343A (es)
CY (1) CY2019009I1 (es)
DK (1) DK2379528T3 (es)
DO (1) DOP2011000204A (es)
EA (1) EA018808B1 (es)
EC (1) ECSP11011157A (es)
ES (1) ES2435798T3 (es)
FI (1) FIC20190008I1 (es)
GT (1) GT201100181A (es)
HK (1) HK1159630A1 (es)
HN (1) HN2011001701A (es)
HR (1) HRP20131051T1 (es)
HU (1) HUS000509I2 (es)
IL (1) IL213350A (es)
JO (1) JO2885B1 (es)
MA (1) MA32903B1 (es)
MX (1) MX2011006757A (es)
MY (1) MY150547A (es)
NZ (1) NZ593114A (es)
PA (1) PA8852901A1 (es)
PE (1) PE20120107A1 (es)
PL (1) PL2379528T3 (es)
PT (1) PT2379528E (es)
RS (1) RS53061B (es)
SG (1) SG172331A1 (es)
SI (1) SI2379528T1 (es)
TN (1) TN2011000293A1 (es)
TW (1) TWI429635B (es)
UA (1) UA104603C2 (es)
WO (1) WO2010075074A1 (es)
ZA (1) ZA201104505B (es)

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