NO20063380L - Triazolderivater som vasopressinantagonister - Google Patents
Triazolderivater som vasopressinantagonisterInfo
- Publication number
- NO20063380L NO20063380L NO20063380A NO20063380A NO20063380L NO 20063380 L NO20063380 L NO 20063380L NO 20063380 A NO20063380 A NO 20063380A NO 20063380 A NO20063380 A NO 20063380A NO 20063380 L NO20063380 L NO 20063380L
- Authority
- NO
- Norway
- Prior art keywords
- triazole derivatives
- vasopressin antagonists
- ring
- vasopressin
- antagonists
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A61P9/12—Antihypertensives
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Ophthalmology & Optometry (AREA)
- Hospice & Palliative Care (AREA)
- Pulmonology (AREA)
- Gynecology & Obstetrics (AREA)
- Urology & Nephrology (AREA)
- Pain & Pain Management (AREA)
- Pregnancy & Childbirth (AREA)
- Rheumatology (AREA)
- Vascular Medicine (AREA)
- Obesity (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Child & Adolescent Psychology (AREA)
- Communicable Diseases (AREA)
- Emergency Medicine (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0329693A GB0329693D0 (en) | 2003-12-22 | 2003-12-22 | Compounds useful in therapy |
GB0408789A GB0408789D0 (en) | 2004-04-20 | 2004-04-20 | Triazole derivatives |
PCT/IB2004/004059 WO2005063754A1 (fr) | 2003-12-22 | 2004-12-09 | Derives de triazole utiles comme antagonistes de la vasopressine |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20063380L true NO20063380L (no) | 2006-09-22 |
Family
ID=34740750
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20063380A NO20063380L (no) | 2003-12-22 | 2006-07-21 | Triazolderivater som vasopressinantagonister |
Country Status (25)
Country | Link |
---|---|
EP (1) | EP1701959A1 (fr) |
JP (1) | JP4698604B2 (fr) |
KR (1) | KR100854872B1 (fr) |
AP (1) | AP2331A (fr) |
AR (1) | AR047340A1 (fr) |
AU (1) | AU2004309164B2 (fr) |
BR (1) | BRPI0417267A (fr) |
CA (1) | CA2551038C (fr) |
CR (1) | CR8481A (fr) |
DO (1) | DOP2004001062A (fr) |
EA (1) | EA010132B1 (fr) |
EC (1) | ECSP066647A (fr) |
GE (1) | GEP20084571B (fr) |
HK (1) | HK1095822A1 (fr) |
IL (1) | IL176349A (fr) |
IS (1) | IS8472A (fr) |
MA (1) | MA28393B1 (fr) |
NL (1) | NL1027833C2 (fr) |
NO (1) | NO20063380L (fr) |
OA (1) | OA13347A (fr) |
PA (1) | PA8620501A1 (fr) |
PE (1) | PE20051051A1 (fr) |
TW (1) | TWI287541B (fr) |
UY (1) | UY28693A1 (fr) |
WO (1) | WO2005063754A1 (fr) |
Families Citing this family (52)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2261218B1 (fr) | 2004-05-26 | 2013-04-03 | Eisai R&D Management Co., Ltd. | Imidazolverbindung zur Verwendung als Intermediat in der Herstellung von Cinnamid-Verbindungen |
CN101083982A (zh) | 2004-09-20 | 2007-12-05 | 泽农医药公司 | 用于治疗硬脂酰CoA去饱和酶介导的疾病的杂环衍生物 |
TW200626138A (en) | 2004-09-20 | 2006-08-01 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as therapeutic agents |
JP4958786B2 (ja) * | 2004-09-20 | 2012-06-20 | ゼノン・ファーマシューティカルズ・インコーポレイテッド | 複素環誘導体および治療薬としてのそれらの使用 |
AR051091A1 (es) | 2004-09-20 | 2006-12-20 | Xenon Pharmaceuticals Inc | Derivados heterociclicos y su uso como inhibidores de la estearoil-coa desaturasa |
AU2005329423A1 (en) | 2004-09-20 | 2006-09-28 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors |
WO2006034441A1 (fr) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Derives heterocycliques et leur utilisation en tant qu'inhibiteurs de la stearoyl-coa desaturase |
CN101083992A (zh) | 2004-09-20 | 2007-12-05 | 泽农医药公司 | 抑制人硬脂酰CoA去饱和酶的哒嗪衍生物 |
ATE458729T1 (de) | 2004-10-26 | 2010-03-15 | Eisai R&D Man Co Ltd | Amorphe form einer zimtsäureamidverbindung |
AP2007004047A0 (en) | 2005-01-20 | 2007-06-30 | Pfizer Ltd | Substituted triazole derivatives as oxtocin antagonists |
MX2007015216A (es) | 2005-06-03 | 2008-02-22 | Xenon Pharmaceuticals Inc | Derivados de aminotiazol y sus usos como agentes terapeuticos. |
AU2006274884B2 (en) * | 2005-07-29 | 2012-04-05 | F. Hoffmann-La Roche Ag | Indol-3-yl-carbonyl-piperidin and piperazin derivatives |
TWI370130B (en) | 2005-11-24 | 2012-08-11 | Eisai R&D Man Co Ltd | Two cyclic cinnamide compound |
TWI378091B (en) | 2006-03-09 | 2012-12-01 | Eisai R&D Man Co Ltd | Multi-cyclic cinnamide derivatives |
US9090604B2 (en) | 2006-07-27 | 2015-07-28 | E I Du Pont De Nemours And Company | Fungicidal azocyclic amides |
WO2008013622A2 (fr) * | 2006-07-27 | 2008-01-31 | E. I. Du Pont De Nemours And Company | Amides azocycliques fongicides |
SA07280403B1 (ar) | 2006-07-28 | 2010-12-01 | إيساي أر أند دي منجمنت كو. ليمتد | ملح رباعي لمركب سيناميد |
JP2010511661A (ja) | 2006-12-07 | 2010-04-15 | エフ.ホフマン−ラ ロシュ アーゲー | V1a受容体アンタゴニストとしてのスピロ−ピペリジン誘導体 |
AU2007329066B2 (en) * | 2006-12-07 | 2012-04-12 | F. Hoffmann-La Roche Ag | Spiro-piperidine derivatives |
RU2009123134A (ru) * | 2006-12-22 | 2011-01-27 | Ф.Хоффманн-Ля Рош Аг (Ch) | Производные спиро-пиперидина |
EP2125827B1 (fr) * | 2006-12-29 | 2010-11-03 | F. Hoffmann-La Roche AG | Dérivés azaspiro |
CL2008000582A1 (es) | 2007-02-28 | 2008-06-27 | Eisai R&D Man Co Ltd | Compuestos ciclicos derivados de oximorfolina condensados; farmacos que comprenden a dichos compuestos; y su uso para tratar enfermedad de alzheimer, demencia senil, sindrome de down o amiloidosis. |
NZ583515A (en) | 2007-08-31 | 2011-05-27 | Eisai R&D Man Co Ltd | Imidazole-pyridine derivative featuring a 1,2,4-triazole ring fused to a 5-7 membered ring, for treating a disease caused by amyloid-beta such as Alzheimer's, dementia, Down's syndrome, and amyloidosis |
US7935815B2 (en) | 2007-08-31 | 2011-05-03 | Eisai R&D Management Co., Ltd. | Imidazoyl pyridine compounds and salts thereof |
US8470819B2 (en) | 2008-11-03 | 2013-06-25 | Merck Sharp & Dohme Corp. | Benzimidazole and aza-benzimidazole carboxamides |
CA2811192C (fr) * | 2010-10-01 | 2018-02-27 | Taisho Pharmaceutical Co., Ltd. | Derive de 1,2,4-triazolone |
CA2903431C (fr) | 2013-03-14 | 2022-12-06 | Kalyra Pharmaceuticals, Inc. | Composes analgesiques bicyclopentanes |
EP3080072A4 (fr) | 2013-12-12 | 2017-07-19 | Kalyra Pharmaceuticals, inc. | Composés d'alkyle bicyclique et synthèse |
CN106232567B (zh) | 2014-03-07 | 2021-11-02 | 里科瑞尔姆Ip控股有限责任公司 | 螺桨烷衍生物及合成 |
KR20170048588A (ko) | 2014-09-17 | 2017-05-08 | 카리라 파마슈티컬스, 아이앤씨. | 바이사이클릭 화합물 |
US10138236B2 (en) | 2014-09-24 | 2018-11-27 | Bayer Pharma Aktiengesellschaft | Factor xia-inhibiting pyridobenzazepine and pyridobenzazocine derivatives |
SG11201703199UA (en) | 2014-11-03 | 2017-05-30 | Bayer Pharma AG | Hydroxyalkyl-substituted phenyltriazole derivatives and uses thereof |
RU2637101C2 (ru) * | 2016-01-11 | 2017-11-29 | Федеральное государственное бюджетное научное учреждение "Федеральный исследовательский центр вирусологии и микробиологии" (ФГБНУ ФИЦВиМ) | Устройство для определения аспирированной дозы аэрозолей |
JP2019509338A (ja) * | 2016-02-23 | 2019-04-04 | セルビシオ アンダルーサ デ サルー | 治療活性が増加した抗ウイルス剤としてのピペラジン誘導体 |
CN109071464A (zh) | 2016-05-03 | 2018-12-21 | 拜耳制药股份公司 | 氧代烷基取代的苯基***衍生物及其用途 |
EP3452469A1 (fr) | 2016-05-03 | 2019-03-13 | Bayer Pharma Aktiengesellschaft | Dérivés d'aryltriazole à substitution fluoroalkyle et utilisations desdits dérivés |
AR108263A1 (es) | 2016-05-03 | 2018-08-01 | Bayer Pharma AG | Procedimiento para la preparación de derivados de 1-fenilo-1,2,4-triazol sustituidos por 5-hidroxialquilo |
EP3452472A1 (fr) | 2016-05-03 | 2019-03-13 | Bayer Aktiengesellschaft | Dérivés d'hétéroaryltriazole substitués par hydroxyalkyle et utilisations associées |
WO2017191105A1 (fr) | 2016-05-03 | 2017-11-09 | Bayer Pharma Aktiengesellschaft | Dérivés d'aryltriazole à substitution amide et leurs utilisations |
US9988367B2 (en) * | 2016-05-03 | 2018-06-05 | Bayer Pharma Aktiengesellschaft | Amide-substituted pyridinyltriazole derivatives and uses thereof |
JP6710273B2 (ja) * | 2016-05-09 | 2020-06-17 | 日本曹達株式会社 | 環状アミン化合物および有害生物防除剤 |
US10927098B2 (en) | 2016-10-20 | 2021-02-23 | Bayer Pharma Aktiengesellschaft | Hydroxyalkyl-substituted triazole derivatives and uses thereof |
CA3063729A1 (fr) | 2017-05-15 | 2018-11-22 | Recurium Ip Holdings, Llc | Composes analgesiques |
SI3700913T1 (sl) | 2017-10-24 | 2022-02-28 | Bayer Aktiengesellschaft | Predzdravila derivatov substituiranega triazola in njihove uporabe |
WO2019081303A1 (fr) | 2017-10-24 | 2019-05-02 | Bayer Pharma Aktiengesellschaft | Dérivés de triazole substitués et utilisations associées |
WO2019081307A1 (fr) | 2017-10-24 | 2019-05-02 | Bayer Aktiengesellschaft | Dérivés de triazole substitués et utilisations associées |
CA3079770A1 (fr) | 2017-10-24 | 2019-05-02 | Bayer Pharma Aktiengesellschaft | Derives de triazole substitues par une amine et utilisations associees |
WO2019081291A1 (fr) | 2017-10-24 | 2019-05-02 | Bayer Aktiengesellschaft | Promédicaments de dérivés de triazole substitués, et utilisations de ceux-ci |
US11230540B2 (en) | 2017-10-24 | 2022-01-25 | Bayer Pharma Aktiengesellschaft | Substituted triazole derivatives and uses thereof |
WO2019081302A1 (fr) | 2017-10-24 | 2019-05-02 | Bayer Pharma Aktiengesellschaft | Dérivés de triazole substitués et utilisations associées |
TW201938171A (zh) | 2017-12-15 | 2019-10-01 | 匈牙利商羅特格登公司 | 作為血管升壓素V1a受體拮抗劑之三環化合物 |
HU231206B1 (hu) | 2017-12-15 | 2021-10-28 | Richter Gedeon Nyrt. | Triazolobenzazepinek |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4481360A (en) * | 1983-08-26 | 1984-11-06 | The Upjohn Company | 4H-1,2,4-Triazol-3-yl compounds |
AU2000223275A1 (en) * | 2000-02-08 | 2001-08-20 | Yamanouchi Pharmaceutical Co..Ltd. | Novel triazole derivatives |
SK16242002A3 (sk) * | 2000-05-19 | 2003-04-01 | Merck Patent Gmbh | Derivát triazolu a farmaceutický prostriedok, ktorý ho obsahuje |
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2004
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- 2004-12-09 KR KR1020067012328A patent/KR100854872B1/ko not_active IP Right Cessation
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- 2004-12-09 CA CA2551038A patent/CA2551038C/fr not_active Expired - Fee Related
- 2004-12-09 WO PCT/IB2004/004059 patent/WO2005063754A1/fr active Application Filing
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- 2004-12-09 JP JP2006546356A patent/JP4698604B2/ja not_active Expired - Fee Related
- 2004-12-09 EP EP04801354A patent/EP1701959A1/fr not_active Withdrawn
- 2004-12-17 TW TW093139507A patent/TWI287541B/zh active
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Also Published As
Publication number | Publication date |
---|---|
TWI287541B (en) | 2007-10-01 |
JP4698604B2 (ja) | 2011-06-08 |
AU2004309164B2 (en) | 2007-11-15 |
KR100854872B1 (ko) | 2008-08-28 |
KR20060101546A (ko) | 2006-09-25 |
NL1027833C2 (nl) | 2006-03-06 |
MA28393B1 (fr) | 2007-01-02 |
CA2551038C (fr) | 2010-04-27 |
EA200600925A1 (ru) | 2006-12-29 |
JP2007515468A (ja) | 2007-06-14 |
EA010132B1 (ru) | 2008-06-30 |
CA2551038A1 (fr) | 2005-07-14 |
ECSP066647A (es) | 2006-10-25 |
TW200528099A (en) | 2005-09-01 |
IL176349A0 (en) | 2006-10-05 |
PA8620501A1 (es) | 2005-08-04 |
OA13347A (en) | 2007-04-13 |
IS8472A (is) | 2006-05-18 |
AP2006003631A0 (en) | 2006-06-30 |
EP1701959A1 (fr) | 2006-09-20 |
IL176349A (en) | 2011-11-30 |
WO2005063754A1 (fr) | 2005-07-14 |
CR8481A (es) | 2007-12-04 |
NL1027833A1 (nl) | 2005-06-23 |
DOP2004001062A (es) | 2005-06-30 |
AU2004309164A1 (en) | 2005-07-14 |
UY28693A1 (es) | 2005-07-29 |
PE20051051A1 (es) | 2005-12-17 |
GEP20084571B (en) | 2008-12-25 |
AR047340A1 (es) | 2006-01-18 |
HK1095822A1 (en) | 2007-07-06 |
BRPI0417267A (pt) | 2007-04-17 |
AP2331A (en) | 2011-12-05 |
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