NL1005338C2 - Werkwijze voor de bereiding van een optisch actief fenylglycidylzuurderivaat. - Google Patents
Werkwijze voor de bereiding van een optisch actief fenylglycidylzuurderivaat. Download PDFInfo
- Publication number
- NL1005338C2 NL1005338C2 NL1005338A NL1005338A NL1005338C2 NL 1005338 C2 NL1005338 C2 NL 1005338C2 NL 1005338 A NL1005338 A NL 1005338A NL 1005338 A NL1005338 A NL 1005338A NL 1005338 C2 NL1005338 C2 NL 1005338C2
- Authority
- NL
- Netherlands
- Prior art keywords
- formula
- compound
- optically active
- derived
- hetero
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/48—Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C219/00—Compounds containing amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C219/24—Compounds containing amino and esterified hydroxy groups bound to the same carbon skeleton having esterified hydroxy groups or amino groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Epoxy Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Priority Applications (10)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
NL1005338A NL1005338C2 (nl) | 1997-02-21 | 1997-02-21 | Werkwijze voor de bereiding van een optisch actief fenylglycidylzuurderivaat. |
CA002228196A CA2228196A1 (en) | 1997-02-21 | 1998-01-29 | Process for preparing an optically active phenylglycidyl acid derivative |
AT98200484T ATE202094T1 (de) | 1997-02-21 | 1998-02-16 | Verfahren zur herstellung eines optisch aktiven phenylglycidylsäurederivates |
EP98200484A EP0860439B1 (en) | 1997-02-21 | 1998-02-16 | Process for preparing an optically active phenylglycidyl acid derivative |
DE69800900T DE69800900D1 (de) | 1997-02-21 | 1998-02-16 | Verfahren zur Herstellung eines optisch aktiven Phenylglycidylsäurederivates |
IL12339198A IL123391A0 (en) | 1997-02-21 | 1998-02-19 | Process for preparing an optically active phenylglycidyl acid derivative |
JP10076391A JPH10279572A (ja) | 1997-02-21 | 1998-02-19 | 光学活性なフェニルグリシジル酸誘導体の製造法 |
CN98107076A CN1197070A (zh) | 1997-02-21 | 1998-02-20 | 旋光苯基缩水甘油酸衍生物的制备方法 |
HU9800372A HUP9800372A3 (en) | 1997-02-21 | 1998-02-20 | Process for producing trans-phenyl-glycidyl-acid derivatives |
US09/027,619 US6025506A (en) | 1997-02-21 | 1998-02-23 | Process for preparing an optically active phenylglycidyl acid derivative |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
NL1005338A NL1005338C2 (nl) | 1997-02-21 | 1997-02-21 | Werkwijze voor de bereiding van een optisch actief fenylglycidylzuurderivaat. |
NL1005338 | 1997-02-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
NL1005338C2 true NL1005338C2 (nl) | 1998-08-24 |
Family
ID=19764467
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NL1005338A NL1005338C2 (nl) | 1997-02-21 | 1997-02-21 | Werkwijze voor de bereiding van een optisch actief fenylglycidylzuurderivaat. |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP0860439B1 (ja) |
JP (1) | JPH10279572A (ja) |
CN (1) | CN1197070A (ja) |
AT (1) | ATE202094T1 (ja) |
CA (1) | CA2228196A1 (ja) |
DE (1) | DE69800900D1 (ja) |
HU (1) | HUP9800372A3 (ja) |
IL (1) | IL123391A0 (ja) |
NL (1) | NL1005338C2 (ja) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1302261B1 (it) * | 1998-09-24 | 2000-09-05 | Zambon Spa | Processo per la risoluzione cinetica enzimatica di 3-fenilglicidatiper transesterificazione con amminoalcoli |
US7060471B2 (en) * | 2003-03-12 | 2006-06-13 | Council Of Scientific & Industrial Research | Stereoselective chemoenzymatic process for the preparation of optically enriched phenylglycidates as precursors of taxol side chain |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0342904A2 (en) * | 1988-05-18 | 1989-11-23 | MARION LABORATORIES, INC. (a Delaware corporation) | 2-Hydroxy-3-(4-methoxyphenyl)-3-(2-aminophenylthio)propionic acid, 8'-phenylmenthyl ester, especially for diltiazem |
-
1997
- 1997-02-21 NL NL1005338A patent/NL1005338C2/nl not_active IP Right Cessation
-
1998
- 1998-01-29 CA CA002228196A patent/CA2228196A1/en not_active Abandoned
- 1998-02-16 AT AT98200484T patent/ATE202094T1/de active
- 1998-02-16 EP EP98200484A patent/EP0860439B1/en not_active Expired - Lifetime
- 1998-02-16 DE DE69800900T patent/DE69800900D1/de not_active Expired - Lifetime
- 1998-02-19 IL IL12339198A patent/IL123391A0/xx unknown
- 1998-02-19 JP JP10076391A patent/JPH10279572A/ja active Pending
- 1998-02-20 HU HU9800372A patent/HUP9800372A3/hu unknown
- 1998-02-20 CN CN98107076A patent/CN1197070A/zh active Pending
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0342904A2 (en) * | 1988-05-18 | 1989-11-23 | MARION LABORATORIES, INC. (a Delaware corporation) | 2-Hydroxy-3-(4-methoxyphenyl)-3-(2-aminophenylthio)propionic acid, 8'-phenylmenthyl ester, especially for diltiazem |
Non-Patent Citations (1)
Title |
---|
A. SCHWARTZ ET AL.: "Enantioselective synthesis of calcium channel blockers of the diltiazem group", JOURNAL OF ORGANIC CHEMISTRY, vol. 57, no. 3, 1992, WASHINGTON DC, US, pages 851 - 6, XP002042991 * |
Also Published As
Publication number | Publication date |
---|---|
IL123391A0 (en) | 1998-09-24 |
EP0860439B1 (en) | 2001-06-13 |
HUP9800372A3 (en) | 2001-02-28 |
CA2228196A1 (en) | 1998-08-21 |
HU9800372D0 (en) | 1998-04-28 |
DE69800900D1 (de) | 2001-07-19 |
CN1197070A (zh) | 1998-10-28 |
ATE202094T1 (de) | 2001-06-15 |
HUP9800372A2 (hu) | 1999-09-28 |
EP0860439A1 (en) | 1998-08-26 |
JPH10279572A (ja) | 1998-10-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PD2B | A search report has been drawn up | ||
VD1 | Lapsed due to non-payment of the annual fee |
Effective date: 20010901 |