MXPA03007166A - Pirido-pirimidinas 6-sustituidas. - Google Patents

Pirido-pirimidinas 6-sustituidas.

Info

Publication number
MXPA03007166A
MXPA03007166A MXPA03007166A MXPA03007166A MXPA03007166A MX PA03007166 A MXPA03007166 A MX PA03007166A MX PA03007166 A MXPA03007166 A MX PA03007166A MX PA03007166 A MXPA03007166 A MX PA03007166A MX PA03007166 A MXPA03007166 A MX PA03007166A
Authority
MX
Mexico
Prior art keywords
pyrimidines
substituted pyrido
pyrido
substituted
Prior art date
Application number
MXPA03007166A
Other languages
English (en)
Inventor
James Patrick Dunn
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MXPA03007166A publication Critical patent/MXPA03007166A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
MXPA03007166A 2001-02-12 2002-02-04 Pirido-pirimidinas 6-sustituidas. MXPA03007166A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US26837501P 2001-02-12 2001-02-12
US33465401P 2001-11-30 2001-11-30
PCT/EP2002/001106 WO2002064594A2 (en) 2001-02-12 2002-02-04 6-substituted pyrido-pyrimidines

Publications (1)

Publication Number Publication Date
MXPA03007166A true MXPA03007166A (es) 2003-11-18

Family

ID=26953040

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03007166A MXPA03007166A (es) 2001-02-12 2002-02-04 Pirido-pirimidinas 6-sustituidas.

Country Status (32)

Country Link
US (3) US6696566B2 (es)
EP (1) EP1361880B1 (es)
JP (1) JP4064818B2 (es)
KR (1) KR100639772B1 (es)
CN (1) CN100376571C (es)
AR (1) AR035854A1 (es)
AT (1) ATE305303T1 (es)
AU (1) AU2002256615B2 (es)
BR (1) BRPI0207172B8 (es)
CA (1) CA2434834C (es)
CZ (1) CZ20032416A3 (es)
DE (1) DE60206363T2 (es)
DK (1) DK1361880T3 (es)
ES (1) ES2249574T3 (es)
HK (1) HK1066170A1 (es)
HR (1) HRP20030624B1 (es)
HU (1) HU229604B1 (es)
IL (2) IL156872A0 (es)
JO (1) JO2410B1 (es)
MA (1) MA26993A1 (es)
MX (1) MXPA03007166A (es)
MY (1) MY131518A (es)
NO (1) NO326133B1 (es)
NZ (1) NZ526961A (es)
PA (1) PA8539201A1 (es)
PE (1) PE20020976A1 (es)
PL (1) PL366918A1 (es)
RU (1) RU2269527C2 (es)
SK (1) SK11322003A3 (es)
WO (1) WO2002064594A2 (es)
YU (1) YU63703A (es)
ZA (1) ZA200305938B (es)

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HU229604B1 (en) 2001-02-12 2014-02-28 Hoffmann La Roche 6-substituted pyrido-pyrimidines, process for their preparation and pharmaceutical compositions containing them
ATE314370T1 (de) * 2002-01-22 2006-01-15 Warner Lambert Co 2-(pyridin-2-ylamino)-pyrido(2,3-d)pyrimidin-7- one
EP1492790A1 (en) 2002-04-03 2005-01-05 F. Hoffmann-La Roche Ag Imidazo fused compounds
DE60316581T2 (de) 2002-08-06 2008-07-03 F. Hoffmann-La Roche Ag 6-alkoxypyridopyrimidine als inhibitoren der p-38-map-kinase
US20040225077A1 (en) 2002-12-30 2004-11-11 Angiotech International Ag Drug delivery from rapid gelling polymer composition
ES2401330T3 (es) * 2003-02-26 2013-04-18 Sugen, Inc. Compuesto de heteroarilamino inhibidores de proteín quinasas
RU2005135329A (ru) * 2003-04-16 2006-08-10 Ф.Хоффманн-Ля Рош Аг (Ch) Замещенные 7-азахиназолины
DK1685131T3 (da) * 2003-11-13 2007-07-09 Hoffmann La Roche Hydroxyalkylsubstituerede pyrido-7-pyrimidin-7-oner
WO2006056863A1 (en) * 2004-11-23 2006-06-01 Ranbaxy Laboratories Limited Pyrido’2, 3-d!pyrimidines as anti-inflammatory agents
US20060142312A1 (en) * 2004-12-23 2006-06-29 Pfizer Inc C6-aryl and heteroaryl substituted pyrido[2,3-D] pyrimidin-7-ones
WO2006082492A1 (en) * 2005-02-02 2006-08-10 Ranbaxy Laboratories Limited Azabicyclo derivatives as anti-inflammatory agents
ES2552804T3 (es) * 2005-05-04 2015-12-02 Evotec Ag Compuestos heterocíclicos condensados, y sus composiciones y usos
CN101243081A (zh) * 2005-07-21 2008-08-13 霍夫曼-拉罗奇有限公司 作为PTP1B抑制剂的吡啶并[2,3-d]嘧啶-2,4-二胺化合物
RU2008108898A (ru) * 2005-08-09 2009-09-20 Айрм Ллк (Bm) Соединения и композиции в качестве ингибиторов протеинкиназы
US8686002B2 (en) 2005-08-21 2014-04-01 AbbVie Deutschland GmbH & Co. KG Heterocyclic compounds and their use as binding partners for 5-HT5 receptors
JO2783B1 (en) * 2005-09-30 2014-03-15 نوفارتيس ايه جي Compounds 2-Amino-7, 8-dihydro-6H-Bayredo (3,4-D) Pyrimidine-5-Ones
WO2008150260A1 (en) * 2007-06-06 2008-12-11 Gpc Biotech, Inc. 8-oxy-2-aminopyrido (2, 3-d) pyrimidin-7-one derivatives as kinase inhibitors and anticancer agents
WO2008078249A1 (en) * 2006-12-21 2008-07-03 Ranbaxy Laboratories Limited Anti-inflammatory agents
EP2152706A1 (en) 2007-05-07 2010-02-17 Amgen Inc. Pyrazolo-pyridinone and pyrazolo-pyrazinone compounds as p38 modulators, process for their preparation, and their pharmaceutical use
JP2010529973A (ja) 2007-06-15 2010-09-02 エフ.ホフマン−ラ ロシュ アーゲー 3−アミノ−ペンタン−1,5−ジオールの新規製造方法
US8367671B2 (en) 2008-03-21 2013-02-05 Amgen Inc. Pyrazolo[3.4-B]pyrazine compounds as p38 modulators and methods of use as anti-inflamatory agents
EP2112150B1 (en) 2008-04-22 2013-10-16 Forma Therapeutics, Inc. Improved raf inhibitors
CN102177161A (zh) * 2008-10-22 2011-09-07 霍夫曼-拉罗奇有限公司 Jnk的嘧啶基吡啶酮抑制剂
US8674095B2 (en) 2008-12-19 2014-03-18 Afraxis Holdings, Inc. Compounds for treating neuropsychiatric conditions
US8372970B2 (en) * 2009-10-09 2013-02-12 Afraxis, Inc. 8-ethyl-6-(aryl)pyrido[2,3-D]pyrimidin-7(8H)-ones for the treatment of CNS disorders
CA2784749C (en) 2009-12-18 2017-12-12 E. Premkumar Reddy Substituted pyrido[2,3-d]pyrimidin-7(8h)-ones and therapeutic uses thereof
JP6631616B2 (ja) 2014-07-26 2020-01-15 ノース・アンド・サウス・ブラザー・ファーマシー・インベストメント・カンパニー・リミテッド CDK阻害剤としての2−アミノ−ピリド[2,3−d]ピリミジン−7(8H)−オン誘導体及びその使用
CN115105601A (zh) * 2016-06-08 2022-09-27 投资支持有限公司 用于治疗癌症的药物组合
LT3497103T (lt) 2016-08-15 2021-07-26 Pfizer Inc. Piridopirimidinono cdk2/4/6 inhibitoriai
EP3500258A1 (en) * 2016-08-17 2019-06-26 Support-Venture GmbH Method of preventing or treating hearing loss
WO2018132550A1 (en) * 2017-01-11 2018-07-19 The General Hospital Corporation Voltage gated sodium channel imaging agents
MY202289A (en) * 2017-04-04 2024-04-22 Kinarus Ag Methods of preventing or treating ophthalmic diseases
AU2018325442B2 (en) * 2017-08-31 2023-04-13 Dana-Farber Cancer Institute, Inc. Inhibitors of EGFR and/or HER2 and methods of use
CA3128468A1 (en) 2017-10-05 2019-04-11 Fulcrum Therapeutics, Inc. P38 kinase inhibitors reduce dux4 and downstream gene expression for the treatment of fshd
US10342786B2 (en) 2017-10-05 2019-07-09 Fulcrum Therapeutics, Inc. P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD
WO2020006210A1 (en) * 2018-06-27 2020-01-02 Tufts Medical Center, Inc. Pyridopyrimidine compounds and methods of their use
AU2019300135A1 (en) 2018-07-13 2021-01-28 Kinarus Ag Combinations of PPAR agonists and p38 kinase inhibitors for preventing or treating fibrotic diseases
TW202112368A (zh) 2019-06-13 2021-04-01 荷蘭商法西歐知識產權股份有限公司 用於治療有關dux4表現之疾病的抑制劑組合
US20230263803A1 (en) 2020-08-11 2023-08-24 Kinarus Ag Methods of preventing or treating covid-19 and related viral diseases or disorders

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ATE314370T1 (de) * 2002-01-22 2006-01-15 Warner Lambert Co 2-(pyridin-2-ylamino)-pyrido(2,3-d)pyrimidin-7- one

Also Published As

Publication number Publication date
NO326133B1 (no) 2008-10-06
HRP20030624B1 (en) 2007-03-31
DE60206363D1 (de) 2006-02-09
CZ20032416A3 (cs) 2004-07-14
ZA200305938B (en) 2005-01-26
SK11322003A3 (en) 2004-10-05
HRP20030624A2 (en) 2005-06-30
EP1361880A2 (en) 2003-11-19
KR100639772B1 (ko) 2006-10-30
NZ526961A (en) 2005-03-24
CA2434834A1 (en) 2002-08-22
HUP0303458A2 (hu) 2004-01-28
RU2269527C2 (ru) 2006-02-10
HU229604B1 (en) 2014-02-28
CN100376571C (zh) 2008-03-26
US20070135458A1 (en) 2007-06-14
PA8539201A1 (es) 2004-08-31
PL366918A1 (en) 2005-02-07
EP1361880B1 (en) 2005-09-28
IL156872A0 (en) 2004-02-08
WO2002064594A3 (en) 2003-01-09
BR0207172A (pt) 2004-03-30
US7169794B2 (en) 2007-01-30
KR20040018254A (ko) 2004-03-02
BRPI0207172B8 (pt) 2021-05-25
JP4064818B2 (ja) 2008-03-19
RU2003125887A (ru) 2005-03-20
MA26993A1 (fr) 2004-12-20
PE20020976A1 (es) 2002-10-29
HK1066170A1 (en) 2005-03-18
ATE305303T1 (de) 2005-10-15
DK1361880T3 (da) 2006-01-23
BRPI0207172B1 (pt) 2019-04-09
US6696566B2 (en) 2004-02-24
US20040116698A1 (en) 2004-06-17
US7449581B2 (en) 2008-11-11
HUP0303458A3 (en) 2012-12-28
CA2434834C (en) 2010-09-14
WO2002064594A2 (en) 2002-08-22
US20030171584A1 (en) 2003-09-11
AU2002256615B2 (en) 2007-09-13
NO20033540L (no) 2003-08-11
YU63703A (sh) 2006-05-25
IL156872A (en) 2009-07-20
JP2004525896A (ja) 2004-08-26
CN1503672A (zh) 2004-06-09
MY131518A (en) 2007-08-30
DE60206363T2 (de) 2006-07-06
ES2249574T3 (es) 2006-04-01
NO20033540D0 (no) 2003-08-11
JO2410B1 (en) 2007-06-17
AR035854A1 (es) 2004-07-21

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