MX2023000198A - Inhibidores de atr y usos de estos. - Google Patents

Inhibidores de atr y usos de estos.

Info

Publication number
MX2023000198A
MX2023000198A MX2023000198A MX2023000198A MX2023000198A MX 2023000198 A MX2023000198 A MX 2023000198A MX 2023000198 A MX2023000198 A MX 2023000198A MX 2023000198 A MX2023000198 A MX 2023000198A MX 2023000198 A MX2023000198 A MX 2023000198A
Authority
MX
Mexico
Prior art keywords
atr inhibitors
compounds
pharmaceutical compositions
inhibitors
atr
Prior art date
Application number
MX2023000198A
Other languages
English (en)
Inventor
Bo Shan
Bing Hou
Zhongyang Shi
Peng Chen
Hui Yuwen
Jay Mei
Original Assignee
Antengene Discovery Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Antengene Discovery Ltd filed Critical Antengene Discovery Ltd
Publication of MX2023000198A publication Critical patent/MX2023000198A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Abstract

La presente divulgación se refiere a nuevos compuestos útiles como inhibidores de la cinasa ATR, así como a composiciones farmacéuticas que comprenden estos compuestos y métodos de tratamiento mediante la administración de estos compuestos o las composiciones farmacéuticas.
MX2023000198A 2020-07-03 2021-07-02 Inhibidores de atr y usos de estos. MX2023000198A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CN2020100088 2020-07-03
CN2020110396 2020-08-21
CN2020134732 2020-12-09
CN2020135604 2020-12-11
PCT/CN2021/104232 WO2022002245A1 (en) 2020-07-03 2021-07-02 Atr inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
MX2023000198A true MX2023000198A (es) 2023-02-22

Family

ID=79317475

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2023000198A MX2023000198A (es) 2020-07-03 2021-07-02 Inhibidores de atr y usos de estos.

Country Status (13)

Country Link
US (1) US20230339927A1 (es)
EP (1) EP4175948A1 (es)
JP (1) JP2023532303A (es)
KR (1) KR20230035070A (es)
CN (1) CN116134022A (es)
AU (1) AU2021302146A1 (es)
BR (1) BR112022024700A2 (es)
CA (1) CA3185491A1 (es)
CO (1) CO2023000858A2 (es)
IL (1) IL299510A (es)
MX (1) MX2023000198A (es)
TW (1) TW202216701A (es)
WO (1) WO2022002245A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023131234A1 (en) * 2022-01-06 2023-07-13 Shanghai Antengene Corporation Limited Crystalline forms of an atr inhibitor

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI656121B (zh) * 2014-08-04 2019-04-11 德商拜耳製藥公司 2-(嗎啉-4-基)-1,7-萘啶
US11690911B2 (en) * 2017-08-04 2023-07-04 Bayer Aktiengesellschaft Combination of ATR kinase inhibitors and PD-1/PD-L1 inhibitors
RS65147B1 (sr) * 2018-02-07 2024-02-29 Wuxi Biocity Biopharmaceutics Co Ltd Inhibitor atr i njegova primena
ES2954572T3 (es) * 2018-09-07 2023-11-23 Merck Patent Gmbh Derivados de 5-morfolin-4-il-pirazolo[4,3-b]piridina

Also Published As

Publication number Publication date
AU2021302146A1 (en) 2023-01-19
EP4175948A1 (en) 2023-05-10
CN116134022A (zh) 2023-05-16
TW202216701A (zh) 2022-05-01
IL299510A (en) 2023-02-01
BR112022024700A2 (pt) 2023-12-05
JP2023532303A (ja) 2023-07-27
KR20230035070A (ko) 2023-03-10
CO2023000858A2 (es) 2023-02-16
WO2022002245A1 (en) 2022-01-06
CA3185491A1 (en) 2022-01-06
US20230339927A1 (en) 2023-10-26

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