MX2016009219A - Compuestos heteroarilo bicíclicos sustituidos como agonistas rxr. - Google Patents

Compuestos heteroarilo bicíclicos sustituidos como agonistas rxr.

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Publication number
MX2016009219A
MX2016009219A MX2016009219A MX2016009219A MX2016009219A MX 2016009219 A MX2016009219 A MX 2016009219A MX 2016009219 A MX2016009219 A MX 2016009219A MX 2016009219 A MX2016009219 A MX 2016009219A MX 2016009219 A MX2016009219 A MX 2016009219A
Authority
MX
Mexico
Prior art keywords
substituted bicyclic
compounds
bicyclic heteroaryl
heteroaryl compounds
rxr agonists
Prior art date
Application number
MX2016009219A
Other languages
English (en)
Inventor
Gurram Ranga Madhavan
Madanahall Ranganath Rao Jagannath
Sekhar GUDLA Chandra
Original Assignee
Connexios Life Sciences Pvt Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Connexios Life Sciences Pvt Ltd filed Critical Connexios Life Sciences Pvt Ltd
Publication of MX2016009219A publication Critical patent/MX2016009219A/es

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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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Abstract

La presente invención se relaciona con ciertos compuestos bicíclicos sustituidos que son agonistas de RXR y que son, por lo tanto, útiles en el tratamiento de ciertos trastornos que pueden ser prevenidos o tratados por medio de la activación de este receptor. Adicionalmente, la invención se relaciona con los compuestos, métodos para su preparación, composiciones farmacéuticas conteniendo los compuestos y los usos de estos compuestos en el tratamiento de ciertos trastornos.
MX2016009219A 2014-01-14 2015-01-09 Compuestos heteroarilo bicíclicos sustituidos como agonistas rxr. MX2016009219A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN161CH2014 2014-01-14
PCT/IN2015/000010 WO2015107549A1 (en) 2014-01-14 2015-01-09 Substituted bicyclic heteroaryl compounds as rxr agonists

Publications (1)

Publication Number Publication Date
MX2016009219A true MX2016009219A (es) 2017-03-06

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MX2016009219A MX2016009219A (es) 2014-01-14 2015-01-09 Compuestos heteroarilo bicíclicos sustituidos como agonistas rxr.

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EP (1) EP3094626B1 (es)
JP (1) JP6625057B2 (es)
KR (1) KR102372599B1 (es)
CN (1) CN107074800B (es)
AU (1) AU2015207690B2 (es)
BR (1) BR112016016348B1 (es)
CA (1) CA2936162C (es)
CL (1) CL2016001803A1 (es)
DK (1) DK3094626T3 (es)
ES (1) ES2795660T3 (es)
MA (1) MA39253B1 (es)
MX (1) MX2016009219A (es)
MY (1) MY192609A (es)
PH (1) PH12016501393A1 (es)
PL (1) PL3094626T3 (es)
PT (1) PT3094626T (es)
RU (1) RU2721283C2 (es)
SG (1) SG11201605721XA (es)
WO (1) WO2015107549A1 (es)
ZA (1) ZA201605102B (es)

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CN106565761A (zh) * 2016-11-15 2017-04-19 贵州大学 一种4‑羧基苯硼酸的制备工艺
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