MX2011007397A - Inhibidores de dpp-iv para el tratamiento de la diabetes en pacientes pediatricos. - Google Patents
Inhibidores de dpp-iv para el tratamiento de la diabetes en pacientes pediatricos.Info
- Publication number
- MX2011007397A MX2011007397A MX2011007397A MX2011007397A MX2011007397A MX 2011007397 A MX2011007397 A MX 2011007397A MX 2011007397 A MX2011007397 A MX 2011007397A MX 2011007397 A MX2011007397 A MX 2011007397A MX 2011007397 A MX2011007397 A MX 2011007397A
- Authority
- MX
- Mexico
- Prior art keywords
- inhibitors
- diabetes
- dpp
- treatment
- paediatric patients
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
- A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Abstract
La presente invención se refiere al hallazgo de que ciertos agentes inhibidores de DPP-4 son particularmente adecuados para tratar y/o prevenir enfermedades metabólicas, particularmente la diabetes, en pacientes pediátricos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP09151662 | 2009-01-29 | ||
PCT/EP2010/051093 WO2010086411A1 (en) | 2009-01-29 | 2010-01-29 | Dpp-iv inhibitors for treatment of diabetes in paediatric patients |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2011007397A true MX2011007397A (es) | 2011-08-03 |
Family
ID=42101817
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2011007397A MX2011007397A (es) | 2009-01-29 | 2010-01-29 | Inhibidores de dpp-iv para el tratamiento de la diabetes en pacientes pediatricos. |
Country Status (16)
Country | Link |
---|---|
US (1) | US20120122776A1 (es) |
EP (1) | EP2391359A1 (es) |
JP (2) | JP2012516309A (es) |
KR (1) | KR20110107823A (es) |
CN (1) | CN102300567A (es) |
AR (1) | AR075204A1 (es) |
AU (1) | AU2010209705A1 (es) |
BR (1) | BRPI1007877A2 (es) |
CA (1) | CA2750798A1 (es) |
CL (1) | CL2011001685A1 (es) |
EA (1) | EA201101117A1 (es) |
IL (1) | IL213404A0 (es) |
MX (1) | MX2011007397A (es) |
NZ (1) | NZ593754A (es) |
TW (1) | TWI466672B (es) |
WO (1) | WO2010086411A1 (es) |
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DE102004054054A1 (de) | 2004-11-05 | 2006-05-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine |
DE102005035891A1 (de) | 2005-07-30 | 2007-02-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
PE20080251A1 (es) | 2006-05-04 | 2008-04-25 | Boehringer Ingelheim Int | Usos de inhibidores de dpp iv |
MX2008014024A (es) | 2006-05-04 | 2008-11-14 | Boehringer Ingelheim Int | Formas poliformas. |
EP1852108A1 (en) | 2006-05-04 | 2007-11-07 | Boehringer Ingelheim Pharma GmbH & Co.KG | DPP IV inhibitor formulations |
CL2008002427A1 (es) | 2007-08-16 | 2009-09-11 | Boehringer Ingelheim Int | Composicion farmaceutica que comprende 1-cloro-4-(b-d-glucopiranos-1-il)-2-[4-((s)-tetrahidrofurano-3-iloxi)bencil]-benceno combinado con 1-[(4-metilquinazolin-2-il)metil]-3-metil-7-(2-butin-1-il)-8-(3-(r)-aminopiperidin-1-il)xantina; y su uso para tratar diabetes mellitus tipo 2. |
PE20091730A1 (es) | 2008-04-03 | 2009-12-10 | Boehringer Ingelheim Int | Formulaciones que comprenden un inhibidor de dpp4 |
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US20200155558A1 (en) * | 2018-11-20 | 2020-05-21 | Boehringer Ingelheim International Gmbh | Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug |
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AR074990A1 (es) | 2009-01-07 | 2011-03-02 | Boehringer Ingelheim Int | Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina |
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-
2010
- 2010-01-28 TW TW99102442A patent/TWI466672B/zh not_active IP Right Cessation
- 2010-01-28 AR ARP100100223A patent/AR075204A1/es unknown
- 2010-01-29 NZ NZ593754A patent/NZ593754A/en not_active IP Right Cessation
- 2010-01-29 CN CN2010800057616A patent/CN102300567A/zh active Pending
- 2010-01-29 CA CA2750798A patent/CA2750798A1/en not_active Abandoned
- 2010-01-29 WO PCT/EP2010/051093 patent/WO2010086411A1/en active Application Filing
- 2010-01-29 EP EP10701386A patent/EP2391359A1/en not_active Withdrawn
- 2010-01-29 US US13/145,857 patent/US20120122776A1/en not_active Abandoned
- 2010-01-29 BR BRPI1007877A patent/BRPI1007877A2/pt not_active IP Right Cessation
- 2010-01-29 JP JP2011546859A patent/JP2012516309A/ja active Pending
- 2010-01-29 MX MX2011007397A patent/MX2011007397A/es not_active Application Discontinuation
- 2010-01-29 KR KR1020117017748A patent/KR20110107823A/ko not_active Application Discontinuation
- 2010-01-29 EA EA201101117A patent/EA201101117A1/ru unknown
- 2010-01-29 AU AU2010209705A patent/AU2010209705A1/en not_active Abandoned
-
2011
- 2011-06-06 IL IL213404A patent/IL213404A0/en unknown
- 2011-07-11 CL CL2011001685A patent/CL2011001685A1/es unknown
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2014
- 2014-05-20 JP JP2014104463A patent/JP2014144987A/ja active Pending
Also Published As
Publication number | Publication date |
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CL2011001685A1 (es) | 2011-10-28 |
JP2014144987A (ja) | 2014-08-14 |
CN102300567A (zh) | 2011-12-28 |
WO2010086411A1 (en) | 2010-08-05 |
BRPI1007877A2 (pt) | 2018-03-13 |
TW201038272A (en) | 2010-11-01 |
JP2012516309A (ja) | 2012-07-19 |
TWI466672B (zh) | 2015-01-01 |
NZ593754A (en) | 2014-08-29 |
EA201101117A1 (ru) | 2012-03-30 |
IL213404A0 (en) | 2011-07-31 |
CA2750798A1 (en) | 2010-08-05 |
KR20110107823A (ko) | 2011-10-04 |
AR075204A1 (es) | 2011-03-16 |
AU2010209705A1 (en) | 2011-07-07 |
EP2391359A1 (en) | 2011-12-07 |
US20120122776A1 (en) | 2012-05-17 |
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