MEP59708A - 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments - Google Patents
8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicamentsInfo
- Publication number
- MEP59708A MEP59708A MEP-597/08A MEP59708A MEP59708A ME P59708 A MEP59708 A ME P59708A ME P59708 A MEP59708 A ME P59708A ME P59708 A MEP59708 A ME P59708A
- Authority
- ME
- Montenegro
- Prior art keywords
- xanthines
- piperidin
- medicaments
- amino
- production
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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- C07D473/12—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1, 3, and 7, e.g. caffeine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
- Reproductive Health (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pain & Pain Management (AREA)
- Communicable Diseases (AREA)
- Urology & Nephrology (AREA)
- Virology (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Emergency Medicine (AREA)
- Dermatology (AREA)
- Molecular Biology (AREA)
- Child & Adolescent Psychology (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10238243A DE10238243A1 (de) | 2002-08-21 | 2002-08-21 | 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
DE10312353A DE10312353A1 (de) | 2003-03-20 | 2003-03-20 | 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
PCT/EP2003/009127 WO2004018468A2 (de) | 2002-08-21 | 2003-08-18 | 8-[3-amino-piperidin-1-yl]-xanthine, deren herstellung und deren verwendung als arzneimittel |
Publications (2)
Publication Number | Publication Date |
---|---|
ME00396B ME00396B (me) | 2011-05-10 |
MEP59708A true MEP59708A (en) | 2011-05-10 |
Family
ID=31947613
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MEP-597/08A MEP59708A (en) | 2002-08-21 | 2003-08-18 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments |
Country Status (38)
Country | Link |
---|---|
EP (6) | EP2070539A1 (xx) |
JP (6) | JP4233524B2 (xx) |
KR (2) | KR101111101B1 (xx) |
CN (4) | CN105001222B (xx) |
AR (3) | AR041025A1 (xx) |
AT (1) | ATE453644T1 (xx) |
AU (2) | AU2003253418B2 (xx) |
BE (1) | BE2011C038I2 (xx) |
BR (2) | BRPI0313648B8 (xx) |
CA (1) | CA2496249C (xx) |
CY (3) | CY1109928T1 (xx) |
DE (2) | DE50312295D1 (xx) |
DK (1) | DK1532149T3 (xx) |
EA (3) | EA010303B1 (xx) |
EC (2) | ECSP055617A (xx) |
EG (1) | EG25011A (xx) |
ES (1) | ES2339112T3 (xx) |
FR (1) | FR11C0052I2 (xx) |
HK (6) | HK1081552A1 (xx) |
HR (2) | HRP20050157B1 (xx) |
HU (1) | HUS1100028I1 (xx) |
IL (1) | IL166964A (xx) |
IN (2) | IN2015DN01132A (xx) |
LU (2) | LU91889I2 (xx) |
ME (1) | MEP59708A (xx) |
MX (1) | MXPA05001684A (xx) |
MY (2) | MY165643A (xx) |
NO (4) | NO333970B1 (xx) |
PE (1) | PE20040897A1 (xx) |
PL (2) | PL403104A1 (xx) |
PT (1) | PT1532149E (xx) |
RS (2) | RS52142B (xx) |
SA (1) | SA03240448B1 (xx) |
SI (1) | SI1532149T1 (xx) |
TW (3) | TWI469783B (xx) |
UA (1) | UA84275C2 (xx) |
UY (1) | UY27946A1 (xx) |
WO (1) | WO2004018468A2 (xx) |
Families Citing this family (176)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1509525B9 (en) * | 2002-05-31 | 2007-10-31 | Schering Corporation | Process for preparing xanthine phosphodiesterase v inhibitors and precursors thereof |
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