MA32382B1 - DÉRIVÉS INDAZOLES à SUBSTITUTION PHÉNYL OU PYRIDINYLE - Google Patents

DÉRIVÉS INDAZOLES à SUBSTITUTION PHÉNYL OU PYRIDINYLE

Info

Publication number
MA32382B1
MA32382B1 MA33398A MA33398A MA32382B1 MA 32382 B1 MA32382 B1 MA 32382B1 MA 33398 A MA33398 A MA 33398A MA 33398 A MA33398 A MA 33398A MA 32382 B1 MA32382 B1 MA 32382B1
Authority
MA
Morocco
Prior art keywords
pyridinyl
substitution
phenyl
derivatives
indazole derivatives
Prior art date
Application number
MA33398A
Other languages
Arabic (ar)
English (en)
Inventor
Markus Berger
Jan Dahmen
Karl Edman
Thomas Hansson
Martin Hemmerling
Nafizal Hossain
Henrik Johansson
Matti Lepistö
Stinabritt Nilsson
Hartmut Rehwinkel
Original Assignee
Bayer Schering Pharma Ag
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41340347&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA32382(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag, Astrazeneca Ab filed Critical Bayer Schering Pharma Ag
Publication of MA32382B1 publication Critical patent/MA32382B1/fr

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    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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Abstract

La présente invention concerne un composé de formule (Ia). La présente invention concerne donc des dérivés d'indazolyle, des compositions pharmaceutiques comportant de tels dérivés, des procédés de préparation de ces nouveaux dérivés et l'utilisation de ces dérivés en tant que médicaments.
MA33398A 2008-05-20 2010-12-06 DÉRIVÉS INDAZOLES à SUBSTITUTION PHÉNYL OU PYRIDINYLE MA32382B1 (fr)

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US5461608P 2008-05-20 2008-05-20
US8031208P 2008-07-14 2008-07-14
US14477609P 2009-01-15 2009-01-15
PCT/SE2009/000265 WO2009142569A1 (fr) 2008-05-20 2009-05-20 Dérivés indazoles à substitution phényl ou pyridinyle

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MA32382B1 true MA32382B1 (fr) 2011-06-01

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MA33398A MA32382B1 (fr) 2008-05-20 2010-12-06 DÉRIVÉS INDAZOLES à SUBSTITUTION PHÉNYL OU PYRIDINYLE
MA33399A MA32383B1 (fr) 2008-05-20 2010-12-06 DÉRIVÉS D'INDAZOLES à SUBSTITUTIONS PHÉNYLE ET BENZODIOXYNYLE

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EP2291369A4 (fr) 2011-05-11
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DOP2010000357A (es) 2010-12-15
EA201001683A1 (ru) 2011-06-30
IL209122A0 (en) 2011-01-31
CR11802A (es) 2011-01-12
US9512110B2 (en) 2016-12-06
CO6331310A2 (es) 2011-10-20
JP2011520954A (ja) 2011-07-21
CR11801A (es) 2011-02-15
TW200951128A (en) 2009-12-16
HK1154580A1 (zh) 2012-06-29
TW200951114A (en) 2009-12-16
UY31832A (es) 2010-01-05
US20100080786A1 (en) 2010-04-01
KR20110036699A (ko) 2011-04-08
AR071856A1 (es) 2010-07-21
CN102112449A (zh) 2011-06-29
PT2291369E (pt) 2016-03-11
ES2561598T3 (es) 2016-02-29
JP2011520955A (ja) 2011-07-21
ECSP10010620A (es) 2010-12-30
AU2009249874B2 (en) 2012-08-16
DK2291369T3 (en) 2016-02-01
PE20091925A1 (es) 2010-01-24
CO6351783A2 (es) 2011-12-20
EP2291369B1 (fr) 2015-11-04
UA102543C2 (uk) 2013-07-25
US20120302617A1 (en) 2012-11-29
EP2291359A4 (fr) 2011-05-11
EP2291369A1 (fr) 2011-03-09
CA2724584A1 (fr) 2009-11-26
NZ588994A (en) 2012-08-31
MX2010012390A (es) 2011-03-03
AU2009249874A1 (en) 2009-11-26
PA8827101A1 (es) 2009-12-16
JP2014185188A (ja) 2014-10-02
US8916600B2 (en) 2014-12-23
IL209121A (en) 2015-05-31
HUE027217T2 (en) 2016-08-29
HN2010002478A (es) 2013-01-15
PL2291369T3 (pl) 2016-04-29
US20150080434A1 (en) 2015-03-19
US9738632B2 (en) 2017-08-22
CY1117330T1 (el) 2017-04-26
CL2009001247A1 (es) 2010-07-23
ZA201007918B (en) 2011-07-27
WO2009142571A8 (fr) 2011-02-03
BRPI0912855A2 (pt) 2015-10-13
MY173448A (en) 2020-01-25
EP2291359A1 (fr) 2011-03-09
SV2010003738A (es) 2011-03-15
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UY31831A (es) 2010-01-05
WO2009142571A1 (fr) 2009-11-26
US20170081315A1 (en) 2017-03-23
MX2010012529A (es) 2011-03-29
KR101593253B1 (ko) 2016-02-11
CL2009001248A1 (es) 2010-06-11
AR071857A1 (es) 2010-07-21
AU2009249872A1 (en) 2009-11-26
ECSP10010619A (es) 2010-12-30
US8211930B2 (en) 2012-07-03
RS54700B1 (en) 2016-08-31
SV2010003737A (es) 2011-03-15
WO2009142569A1 (fr) 2009-11-26
US20100087489A1 (en) 2010-04-08
JP5579704B2 (ja) 2014-08-27
PA8827001A1 (es) 2009-12-16
BRPI0912878B1 (pt) 2021-11-03
NI201000199A (es) 2012-11-07
EA018629B8 (ru) 2013-12-30
CN102099355A (zh) 2011-06-15
SI2291369T1 (sl) 2016-02-29
BRPI0912878A2 (pt) 2020-08-18
SA109300309B1 (ar) 2013-01-22
EA018629B1 (ru) 2013-09-30
CA2724508A1 (fr) 2009-11-26
MA32383B1 (fr) 2011-06-01
DOP2010000359A (es) 2010-12-15
TWI445705B (zh) 2014-07-21
CA2724508C (fr) 2016-10-25
IL209121A0 (en) 2011-01-31
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EA201001682A1 (ru) 2011-06-30
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ZA201007919B (en) 2011-07-27

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