MA29873B1 - Composes - Google Patents

Composes

Info

Publication number
MA29873B1
MA29873B1 MA30851A MA30851A MA29873B1 MA 29873 B1 MA29873 B1 MA 29873B1 MA 30851 A MA30851 A MA 30851A MA 30851 A MA30851 A MA 30851A MA 29873 B1 MA29873 B1 MA 29873B1
Authority
MA
Morocco
Prior art keywords
compounds
antibacterial agents
tricyclic nitrogen
nitrogen compounds
tricyclic
Prior art date
Application number
MA30851A
Other languages
English (en)
Inventor
Nathalie Cailleau
David Thomas Davies
Joel Michael Esken
Alan Joseph Hennessy
Sukumar Senthil Kumar Kusalakumari
Roger Edward Markwell
Timothy James Miles
Neil David Pearson
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of MA29873B1 publication Critical patent/MA29873B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Composés Composés azotés tricycliques et leur utilisation comme agents antibactériens.
MA30851A 2005-10-21 2008-04-15 Composes MA29873B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72897505P 2005-10-21 2005-10-21
US82659006P 2006-09-22 2006-09-22

Publications (1)

Publication Number Publication Date
MA29873B1 true MA29873B1 (fr) 2008-10-03

Family

ID=38256822

Family Applications (1)

Application Number Title Priority Date Filing Date
MA30851A MA29873B1 (fr) 2005-10-21 2008-04-15 Composes

Country Status (27)

Country Link
US (2) US20080280892A1 (fr)
EP (1) EP1954697B1 (fr)
JP (1) JP2009512695A (fr)
KR (1) KR20080064173A (fr)
AR (1) AR057981A1 (fr)
AT (1) ATE458737T1 (fr)
AU (1) AU2006335042A1 (fr)
BR (1) BRPI0617467A2 (fr)
CA (1) CA2626641A1 (fr)
CR (1) CR9930A (fr)
CY (1) CY1110137T1 (fr)
DE (1) DE602006012535D1 (fr)
DK (1) DK1954697T3 (fr)
EA (1) EA200801128A1 (fr)
ES (1) ES2340531T3 (fr)
HK (1) HK1118546A1 (fr)
HR (1) HRP20100194T8 (fr)
IL (1) IL190803A0 (fr)
MA (1) MA29873B1 (fr)
NO (1) NO20082191L (fr)
NZ (1) NZ567315A (fr)
PE (1) PE20070793A1 (fr)
PL (1) PL1954697T3 (fr)
PT (1) PT1954697E (fr)
SI (1) SI1954697T1 (fr)
TW (1) TW200736263A (fr)
WO (1) WO2007081597A2 (fr)

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CA2626641A1 (fr) * 2005-10-21 2007-07-19 Glaxo Group Limited Composes
US20070185153A1 (en) 2005-12-22 2007-08-09 Nathalie Cailleau Compounds
ATE481406T1 (de) 2006-04-06 2010-10-15 Glaxo Group Ltd Pyrrolochinoxalinonderivate als antibakterielle mittel
GB0608263D0 (en) 2006-04-26 2006-06-07 Glaxo Group Ltd Compounds
GB0613208D0 (en) * 2006-07-03 2006-08-09 Glaxo Group Ltd Compounds
GB0705672D0 (en) * 2007-03-23 2007-05-02 Glaxo Group Ltd Compounds
CL2008001002A1 (es) 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.
DE602008002912D1 (de) * 2007-04-20 2010-11-18 Glaxo Group Ltd Tricyclische stickstoffhaltige verbindungen als antibakterielle wirkstoffe
GB0707706D0 (en) * 2007-04-20 2007-05-30 Glaxo Group Ltd Compounds
EP2005995A1 (fr) * 2007-06-22 2008-12-24 Glaxo Group Limited Composés hétérocycliques pour le traitement de la tuberculose
EP2080761A1 (fr) 2008-01-18 2009-07-22 Glaxo Group Limited Composés
US8349828B2 (en) 2008-02-20 2013-01-08 Actelion Pharmaceuticals Ltd. Azatricyclic antibiotic compounds
CA2720672A1 (fr) 2008-04-15 2009-10-22 Actelion Pharmaceuticals Ltd Antibiotiques tricycliques
CN102105467A (zh) 2008-08-04 2011-06-22 埃科特莱茵药品有限公司 三环烷氨基甲基噁唑烷酮衍生物
RU2530884C2 (ru) * 2008-10-07 2014-10-20 Актелион Фармасьютиклз Лтд Трициклические оксазолидиноновые антибиотические соединения
JP2012505866A (ja) * 2008-10-17 2012-03-08 グラクソ グループ リミテッド 抗菌剤として使用される三環式窒素化合物
NZ593891A (en) 2008-12-12 2013-05-31 Actelion Pharmaceuticals Ltd 5-amino-2-(1-hydroxy-ethyl)-tetrahydropyran derivatives
WO2010081874A1 (fr) 2009-01-15 2010-07-22 Glaxo Group Limited Composés naphthyridine-2(1h)-one utiles comme antibactériens
TW201313726A (zh) 2011-09-16 2013-04-01 Actelion Pharmaceuticals Ltd 製造合成之中間體之方法
US9029368B2 (en) 2011-11-30 2015-05-12 Actelion Pharmaceuticals Ltd. 3,7-disubstituted octahydro-2H-pyrido[4,3-E][1,3]oxazin-2-one antibiotics
SG11201700566SA (en) 2014-08-22 2017-03-30 Glaxosmithkline Ip Dev Ltd Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection
WO2018159609A1 (fr) 2017-02-28 2018-09-07 三井化学アグロ株式会社 Composition de prévention de maladies des plantes et procédé de prévention de maladies des plantes l'utilisant
WO2018207023A2 (fr) * 2017-05-10 2018-11-15 Albajuna Therapeutics, S.L. Dérivés de protéine de fusion fc présentant une double activité élevée immunomodulatrice et antivirale contre le vih
JP2023506147A (ja) 2019-12-02 2023-02-15 ストーム・セラピューティクス・リミテッド Ｍｅｔｔｌ３阻害剤としてのポリヘテロ環式化合物
AU2020397059A1 (en) 2019-12-06 2022-07-21 Vertex Pharmaceuticals Incorporated Substituted tetrahydrofurans as modulators of sodium channels

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ATE481406T1 (de) * 2006-04-06 2010-10-15 Glaxo Group Ltd Pyrrolochinoxalinonderivate als antibakterielle mittel
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GB0707706D0 (en) * 2007-04-20 2007-05-30 Glaxo Group Ltd Compounds

Also Published As

Publication number Publication date
AR057981A1 (es) 2008-01-09
DE602006012535D1 (de) 2010-04-08
NZ567315A (en) 2011-01-28
HRP20100194T8 (en) 2010-06-30
AU2006335042A1 (en) 2007-07-19
CY1110137T1 (el) 2015-01-14
US20080280892A1 (en) 2008-11-13
EP1954697B1 (fr) 2010-02-24
WO2007081597A3 (fr) 2008-06-12
KR20080064173A (ko) 2008-07-08
WO2007081597A2 (fr) 2007-07-19
DK1954697T3 (da) 2010-06-14
SI1954697T1 (sl) 2010-05-31
CA2626641A1 (fr) 2007-07-19
EA200801128A1 (ru) 2008-10-30
PT1954697E (pt) 2010-05-17
IL190803A0 (en) 2008-12-29
TW200736263A (en) 2007-10-01
NO20082191L (no) 2008-07-16
ATE458737T1 (de) 2010-03-15
PL1954697T3 (pl) 2010-07-30
EP1954697A2 (fr) 2008-08-13
HRP20100194T1 (hr) 2010-05-31
JP2009512695A (ja) 2009-03-26
PE20070793A1 (es) 2007-08-23
HK1118546A1 (en) 2009-02-13
CR9930A (es) 2008-07-29
US20080221110A1 (en) 2008-09-11
ES2340531T3 (es) 2010-06-04
BRPI0617467A2 (pt) 2011-07-26

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