LU83781A1 - Nouveaux derives steroides 3-amino substitue et leurs selsprocede de preparation application a tire de medicaments et compositions les renfermant - Google Patents

Nouveaux derives steroides 3-amino substitue et leurs selsprocede de preparation application a tire de medicaments et compositions les renfermant Download PDF

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Publication number
LU83781A1
LU83781A1 LU83781A LU83781A LU83781A1 LU 83781 A1 LU83781 A1 LU 83781A1 LU 83781 A LU83781 A LU 83781A LU 83781 A LU83781 A LU 83781A LU 83781 A1 LU83781 A1 LU 83781A1
Authority
LU
Luxembourg
Prior art keywords
radical
amino
formula
carbon atoms
methyl
Prior art date
Application number
LU83781A
Other languages
English (en)
French (fr)
Inventor
R Deraedt
V Torelli
J Benzoni
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of LU83781A1 publication Critical patent/LU83781A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/007—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 17 (20)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0027—Azides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
LU83781A 1980-11-21 1981-11-20 Nouveaux derives steroides 3-amino substitue et leurs selsprocede de preparation application a tire de medicaments et compositions les renfermant LU83781A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8024750A FR2494698A1 (fr) 1980-11-21 1980-11-21 Nouveaux derives steroides 3-amino substitues, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant
FR8024750 1980-11-21

Publications (1)

Publication Number Publication Date
LU83781A1 true LU83781A1 (fr) 1982-06-30

Family

ID=9248226

Family Applications (1)

Application Number Title Priority Date Filing Date
LU83781A LU83781A1 (fr) 1980-11-21 1981-11-20 Nouveaux derives steroides 3-amino substitue et leurs selsprocede de preparation application a tire de medicaments et compositions les renfermant

Country Status (23)

Country Link
JP (1) JPS57116099A (de)
KR (1) KR880001239B1 (de)
AT (1) AT389703B (de)
AU (1) AU546100B2 (de)
BE (1) BE891201A (de)
CA (1) CA1175415A (de)
CH (1) CH651056A5 (de)
DE (1) DE3146117A1 (de)
DK (1) DK161093C (de)
ES (1) ES8207195A1 (de)
FI (1) FI77871C (de)
FR (1) FR2494698A1 (de)
GB (1) GB2087894B (de)
HU (1) HU184896B (de)
IE (1) IE52188B1 (de)
IL (1) IL64224A0 (de)
IT (1) IT1172086B (de)
LU (1) LU83781A1 (de)
NL (1) NL8105260A (de)
PT (1) PT74015B (de)
SE (1) SE451456B (de)
SU (1) SU1327789A3 (de)
ZA (1) ZA817806B (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9084800B2 (en) * 2011-11-07 2015-07-21 Natreon, Inc. Indolealkylamino-withasteroid conjugates and method of use

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2430467A (en) * 1944-02-11 1947-11-11 Glidden Co 3-amino-derivatives of steroids and method of making same
US2781342A (en) * 1952-05-17 1957-02-12 Upjohn Co Steroid enamines
DE1189074B (de) * 1959-09-12 1965-03-18 Clin Byla Ets Verfahren zur Herstellung von 3-Aminoverbindungen der Androstan- bzw. Pregnan-Reihe
FR1311761A (fr) * 1959-09-12 1962-12-14 Clin Byla Ets Composés aminés de la série des stéroïdes et procédé de préparation de tels composés
NL103735C (de) * 1961-02-17
US3503959A (en) * 1962-03-30 1970-03-31 Sterling Drug Inc 3-amino steroids
US3196168A (en) * 1964-02-18 1965-07-20 American Home Prod Aminoaroyl aminosteroids
BE647858A (de) * 1964-05-13
US3196169A (en) * 1964-11-03 1965-07-20 American Home Prod Aminoacyl aminosteroids
BE672238A (de) * 1965-11-12 1966-03-01
BE811304R (fr) * 1973-10-24 1974-06-17 Pr0cede de preparation du (20 s) 3 beta -n-dimethylamino
FR2463777A1 (fr) * 1979-08-17 1981-02-27 Roussel Uclaf Nouveaux derives du 5a-pregnan-20-ol, leur procede de preparation et leur application comme medicaments

Also Published As

Publication number Publication date
SU1327789A3 (ru) 1987-07-30
DK161093B (da) 1991-05-27
FI813677L (fi) 1982-05-22
IT1172086B (it) 1987-06-18
AT389703B (de) 1990-01-25
FI77871B (fi) 1989-01-31
FR2494698B1 (de) 1983-06-24
SE451456B (sv) 1987-10-12
DE3146117A1 (de) 1982-06-16
KR830007716A (ko) 1983-11-04
IE52188B1 (en) 1987-08-05
IT8149746A0 (it) 1981-11-20
CH651056A5 (fr) 1985-08-30
GB2087894B (en) 1984-09-26
DK161093C (da) 1991-11-18
FI77871C (fi) 1989-05-10
SE8105995L (sv) 1982-05-22
PT74015B (fr) 1983-11-30
JPH0247479B2 (de) 1990-10-19
NL8105260A (nl) 1982-06-16
IL64224A0 (en) 1982-02-28
ATA497081A (de) 1989-06-15
ZA817806B (en) 1982-10-27
GB2087894A (en) 1982-06-03
PT74015A (fr) 1981-12-01
AU546100B2 (en) 1985-08-15
HU184896B (en) 1984-10-29
ES507309A0 (es) 1982-09-01
ES8207195A1 (es) 1982-09-01
CA1175415A (fr) 1984-10-02
FR2494698A1 (fr) 1982-05-28
KR880001239B1 (ko) 1988-07-12
IE812732L (en) 1982-05-21
JPS57116099A (en) 1982-07-19
BE891201A (fr) 1982-05-21
AU7772381A (en) 1982-05-27
DK514981A (da) 1982-05-22

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