LU82795A1 - Composes penam acetoxymethyles et composition pharmaceutique les contenant - Google Patents

Composes penam acetoxymethyles et composition pharmaceutique les contenant Download PDF

Info

Publication number: LU82795A1
Authority: LU; Luxembourg
Prior art keywords: group; compound; formula; penam; hydrogen
Prior art date: 1979-09-26

Application number

LU82795A

Other languages

English (en)

French (fr)

Inventor

W Barth

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-09-26

Filing date

1980-09-24

Publication date

1981-04-17

1980-09-24 Application filed by Pfizer filed Critical Pfizer

1981-04-17 Publication of LU82795A1 publication Critical patent/LU82795A1/fr

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
- C07D499/32—Esters

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Saccharide Compounds (AREA)

LU82795A 1979-09-26 1980-09-24 Composes penam acetoxymethyles et composition pharmaceutique les contenant LU82795A1 (fr)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US7912779		1979-09-26
US06/079,127 US4256733A (en)	1979-09-26	1979-09-26	Acetoxymethyl penam compounds as β-lactamase inhibitors

Publications (1)

Publication Number	Publication Date
LU82795A1 true LU82795A1 (fr)	1981-04-17

Family

ID=22148609

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
LU82795A LU82795A1 (fr)	1979-09-26	1980-09-24	Composes penam acetoxymethyles et composition pharmaceutique les contenant

Country Status (36)

Country	Link
US (1)	US4256733A (no)
JP (1)	JPS6016958B2 (no)
KR (1)	KR840000796B1 (no)
AR (1)	AR224547A1 (no)
AT (1)	AT366384B (no)
AU (1)	AU517074B2 (no)
BE (1)	BE885389A (no)
CA (1)	CA1150242A (no)
CH (1)	CH645646A5 (no)
CS (1)	CS212284B2 (no)
DD (1)	DD153123A5 (no)
DE (1)	DE3035995C2 (no)
DK (1)	DK404980A (no)
EG (1)	EG14888A (no)
ES (1)	ES8106528A1 (no)
FI (2)	FI67552C (no)
FR (1)	FR2465736A1 (no)
GB (2)	GB2059420B (no)
GR (1)	GR70065B (no)
HU (1)	HU183212B (no)
IE (2)	IE50506B1 (no)
IL (1)	IL61117A (no)
IN (1)	IN154557B (no)
IT (1)	IT1132754B (no)
LU (1)	LU82795A1 (no)
MX (1)	MX6580E (no)
NL (1)	NL185923C (no)
NO (2)	NO160370C (no)
NZ (1)	NZ195058A (no)
PH (1)	PH15697A (no)
PL (1)	PL126949B1 (no)
PT (1)	PT71837B (no)
SE (2)	SE449865B (no)
SU (1)	SU959628A3 (no)
YU (1)	YU41733B (no)
ZA (1)	ZA805132B (no)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4364957A (en) *	1979-09-26	1982-12-21	Pfizer Inc.	Bis-esters of alkanediols as antibacterial agents
US4511512A (en) *	1980-05-01	1985-04-16	Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Produktionsaktiensel skab)	Substantially pure dicyclohexyl ammonium 6-β-bromo-penicillanate
US4474698A (en) *	1980-12-11	1984-10-02	Pfizer Inc.	Process for preparing esters of penicillanic acid sulfone
US4361513A (en) *	1980-12-11	1982-11-30	Pfizer Inc.	Esters of penicillanic acid sulfone
US4558042A (en) *	1981-05-06	1985-12-10	Farmitalia Carlo Erba S.P.A.	β-Lactam-containing antibacterial agents and β-lactamase inhibitors
ZA826687B (en) *	1981-09-14	1983-07-27	Pfizer	Beta-lactamase inhibiting 2-beta-substituted-2-alpha-methyl 5(r)penam-3-alpha-carboxylic acid 1,1-dioxides and intermediates therefor
JPS58185589A (ja) *	1982-04-23	1983-10-29	Taiho Yakuhin Kogyo Kk	ペニシリン誘導体
JPS62198687A (ja) *	1986-02-27	1987-09-02	Taiho Yakuhin Kogyo Kk	２β−置換チオメチルペニシリン誘導体
US4861768A (en) *	1986-02-27	1989-08-29	Taiho Pharmaceutical Company, Limited	2 β-substituted thiomethylpenicillin derivatives and their preparation and use
DE618979T1 (de) *	1991-12-19	1995-05-18	Novonordisk As	Verbesserte methode zur herstellung von bestimmten -g(b)-lactam-antibiotika.
CN115385934A (zh) *	2022-10-26	2022-11-25	北京纳百生物科技有限公司	一种舒巴坦半抗原及其合成方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IN149747B (no) *	1977-06-07	1982-04-03	Pfizer

1979
- 1979-09-26 US US06/079,127 patent/US4256733A/en not_active Expired - Lifetime
1980
- 1980-08-13 SE SE8005714A patent/SE449865B/sv not_active IP Right Cessation
- 1980-08-20 ZA ZA00805132A patent/ZA805132B/xx unknown
- 1980-08-20 IN IN607/DEL/80A patent/IN154557B/en unknown
- 1980-09-19 HU HU802310A patent/HU183212B/hu unknown
- 1980-09-19 SU SU802983144A patent/SU959628A3/ru active
- 1980-09-22 CS CS806403A patent/CS212284B2/cs unknown
- 1980-09-22 PL PL1980226868A patent/PL126949B1/pl unknown
- 1980-09-23 CA CA000360886A patent/CA1150242A/en not_active Expired
- 1980-09-23 GR GR62939A patent/GR70065B/el unknown
- 1980-09-23 IL IL61117A patent/IL61117A/xx unknown
- 1980-09-23 GB GB8030639A patent/GB2059420B/en not_active Expired
- 1980-09-23 EG EG584/80A patent/EG14888A/xx active
- 1980-09-23 AT AT0474680A patent/AT366384B/de not_active IP Right Cessation
- 1980-09-24 AR AR282629A patent/AR224547A1/es active
- 1980-09-24 KR KR1019800003721A patent/KR840000796B1/ko active
- 1980-09-24 DE DE3035995A patent/DE3035995C2/de not_active Expired
- 1980-09-24 LU LU82795A patent/LU82795A1/fr unknown
- 1980-09-24 PH PH24617A patent/PH15697A/en unknown
- 1980-09-24 MX MX809044U patent/MX6580E/es unknown
- 1980-09-25 YU YU2449/80A patent/YU41733B/xx unknown
- 1980-09-25 AU AU62713/80A patent/AU517074B2/en not_active Ceased
- 1980-09-25 NO NO802836A patent/NO160370C/no unknown
- 1980-09-25 NZ NZ195058A patent/NZ195058A/xx unknown
- 1980-09-25 ES ES495354A patent/ES8106528A1/es not_active Expired
- 1980-09-25 FI FI803028A patent/FI67552C/fi not_active IP Right Cessation
- 1980-09-25 IE IE1998/80A patent/IE50506B1/en not_active IP Right Cessation
- 1980-09-25 CH CH719980A patent/CH645646A5/fr not_active IP Right Cessation
- 1980-09-25 IT IT24920/80A patent/IT1132754B/it active
- 1980-09-25 IE IE1095/85A patent/IE50507B1/en unknown
- 1980-09-25 DD DD80224128A patent/DD153123A5/de unknown
- 1980-09-25 DK DK404980A patent/DK404980A/da not_active Application Discontinuation
- 1980-09-25 FR FR8020618A patent/FR2465736A1/fr active Granted
- 1980-09-25 PT PT71837A patent/PT71837B/pt unknown
- 1980-09-25 BE BE0/202222A patent/BE885389A/fr not_active IP Right Cessation
- 1980-09-25 NL NLAANVRAGE8005344,A patent/NL185923C/xx not_active IP Right Cessation
- 1980-09-25 JP JP55133639A patent/JPS6016958B2/ja not_active Expired
1983
- 1983-03-25 NO NO83831082A patent/NO160299C/no unknown
- 1983-07-22 GB GB08319784A patent/GB2125037B/en not_active Expired
1984
- 1984-01-30 FI FI840367A patent/FI67854C/fi not_active IP Right Cessation
1985
- 1985-02-27 SE SE8500965A patent/SE461528B/sv not_active IP Right Cessation

Also Published As

Publication number	Publication date
IE50507B1 (en)	1986-04-30
GR70065B (no)	1982-07-26
CA1150242A (en)	1983-07-19
ATA474680A (de)	1981-08-15
SE8500965D0 (sv)	1985-02-27
NZ195058A (en)	1982-12-07
GB2125037A (en)	1984-02-29
AU517074B2 (en)	1981-07-09
YU41733B (en)	1987-12-31
DK404980A (da)	1981-03-27
NO160370C (no)	1989-04-12
NL185923B (nl)	1990-03-16
AT366384B (de)	1982-04-13
FI803028A (fi)	1981-03-27
AU6271380A (en)	1981-04-09
NO160299B (no)	1988-12-27
BE885389A (fr)	1981-03-25
SE461528B (sv)	1990-02-26
JPS5657788A (en)	1981-05-20
PH15697A (en)	1983-03-14
ZA805132B (en)	1981-12-30
CS212284B2 (en)	1982-03-26
FI67854C (fi)	1985-06-10
DE3035995C2 (de)	1985-01-10
FI67552B (fi)	1984-12-31
FR2465736A1 (fr)	1981-03-27
IT1132754B (it)	1986-07-02
US4256733A (en)	1981-03-17
FI67552C (fi)	1985-04-10
GB2059420B (en)	1984-03-14
IE801998L (en)	1981-03-26
IL61117A (en)	1983-10-31
IL61117A0 (en)	1980-11-30
FI840367A0 (fi)	1984-01-30
SE8005714L (sv)	1981-03-27
IN154557B (no)	1984-11-10
IE50506B1 (en)	1986-04-30
NO160299C (no)	1989-04-05
ES495354A0 (es)	1981-08-16
PL126949B1 (en)	1983-09-30
NL8005344A (nl)	1981-03-30
CH645646A5 (fr)	1984-10-15
AR224547A1 (es)	1981-12-15
GB2125037B (en)	1984-08-01
IT8024920A0 (it)	1980-09-25
GB2059420A (en)	1981-04-23
PT71837A (en)	1980-10-01
DE3035995A1 (de)	1981-04-02
NO831082L (no)	1981-03-27
NO160370B (no)	1989-01-02
EG14888A (en)	1985-06-30
MX6580E (es)	1985-07-24
PT71837B (en)	1981-07-09
FR2465736B1 (no)	1982-04-30
PL226868A1 (no)	1981-10-16
SU959628A3 (ru)	1982-09-15
DD153123A5 (de)	1981-12-23
HU183212B (en)	1984-04-28
FI67854B (fi)	1985-02-28
JPS6016958B2 (ja)	1985-04-30
KR830003494A (ko)	1983-06-20
ES8106528A1 (es)	1981-08-16
FI840367A (fi)	1984-01-30
NO802836L (no)	1981-03-27
NL185923C (nl)	1990-08-16
KR840000796B1 (ko)	1984-06-12
IE801095L (en)	1981-01-09
GB8319784D0 (en)	1983-08-24
SE449865B (sv)	1987-05-25
YU244980A (en)	1983-02-28

Similar Documents

Publication	Publication Date	Title
LU82880A1 (fr)	1981-06-04	Derives d'acides 6 beta-hydroxyalkylpenicillaniques,leur procede de production et compositions pharmaceutiques les contenant
CH634073A5 (en)	1983-01-14	1,1-Dioxides of penicillanic acid and its esters which are useful as beta-lactamase inhibitors
LU82452A1 (fr)	1980-12-16	Bis-esters de methanediol avec des penicillines et le 1,1-dioxyde d'acide penicillanique,leur procede de production et composition pharmaceutique les contenant
CH655114A5 (fr)	1986-03-27	Derives de l'imidazotetrazinone, leur preparation et compositions pharmaceutiques les contenant.
LU82192A1 (fr)	1980-06-06	Composes antibacteriens et inhibituers de beta-lactamase, procede pour les preparer et leur usage comme medicaments
LU82795A1 (fr)	1981-04-17	Composes penam acetoxymethyles et composition pharmaceutique les contenant
BE881862A (fr)	1980-08-22	Composes antibacteriens et inhibiteurs de beta-lactamase, procede pour les preparer et leur usage comme medicaments
LU82215A1 (fr)	1980-09-24	Procede et composes intermediaires pour la prouduction du 1,1-dioxyde d'acide penicillanique et de ses esters
CH642080A5 (fr)	1984-03-30	Antibiotiques du type beta-lactame, leur procede de production et medicament les contenant.
LU82219A1 (fr)	1980-09-24	Acides penicillamiques 6- -substitues inhibiteurs de -lac-tamase, leur procede de production et composition pharmaceutique les contenant
BE875054A (fr)	1979-07-16	Composes analogues aux cephalosporines
BE700422A (no)	1967-12-27
FR2482103A1 (fr)	1981-11-13	Sulfone d'acide 2b-chloromethyl-2a-methylpename-3a-carboxylique, son procede de preparation et son utilisation en association avec des antibiotiques de la classe des b-lactamines
FR2467210A1 (fr)	1981-04-17	Procede de preparation de derives de l'acide 1,1-dioxopenicillanique
BE821243A (fr)	1975-04-18	Derives de la penicilline
FR2520362A1 (fr)	1983-07-29	Nouveaux composes de type b-lactame, y compris leurs sels formes avec des acides ou des bases acceptables en pharmacie, procedes pour produire ces composes, medicaments les contenant et leur utilisation pour combattre les maladies infectieuses
BE887886A (fr)	1981-09-10	Derivés de l'acide 2-peneme-3-carboxylique leur preparation et leur application thérapeutique.
FR2483925A1 (fr)	1981-12-11	Procede de preparation de derives de l'acide peneme-3-carboxylique
BE832435R (fr)	1976-02-16	Perfectionnements relatifs aux antibiotiques
BE882027A (fr)	1980-09-03	Acides penicillaniques 6-beta-substitues, procede de preparation et utilisation comme inhibiteurs des beta-lactamases
LU81475A1 (fr)	1980-02-14	Composition pharmaceutique a base d'acide 7-(d-2-(4-ethylpiperazine-2,3-dione-1-carboxamido)-2-(4-hydroxyphenyl)acetamido)-3-((1-methyl-5-tetrazolyl)thiomethyl)-3-desacetoxy-methylcephalosporanique et de 1,1-dioxyde d'acide penicillanique
FR2509311A1 (fr)	1983-01-14	Derives de beta-lactame, les compositions pharmaceutiques les contenant et leur procede de preparation
LU82458A1 (fr)	1980-10-08	Nouveaux derives d'acide penicillanique substitues en 6- et 6- et leur procede de production
BE609039A (no)
CH644127A5 (fr)	1984-07-13	Oxazolino-azetidinones et leur procede de preparation.