JPS61151172A - インドール、その製造方法及びそれを含有する製薬組成物 - Google Patents

インドール、その製造方法及びそれを含有する製薬組成物

Info

Publication number
JPS61151172A
JPS61151172A JP60278124A JP27812485A JPS61151172A JP S61151172 A JPS61151172 A JP S61151172A JP 60278124 A JP60278124 A JP 60278124A JP 27812485 A JP27812485 A JP 27812485A JP S61151172 A JPS61151172 A JP S61151172A
Authority
JP
Japan
Prior art keywords
group
indole
general formula
formula
hydrogen atom
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP60278124A
Other languages
English (en)
Japanese (ja)
Inventor
デイビツド・エドマンド・ベイズ
コリン・フレデリツク・ウエブ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of JPS61151172A publication Critical patent/JPS61151172A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
JP60278124A 1984-12-13 1985-12-12 インドール、その製造方法及びそれを含有する製薬組成物 Pending JPS61151172A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8431426 1984-12-13
GB848431426A GB8431426D0 (en) 1984-12-13 1984-12-13 Chemical compounds

Publications (1)

Publication Number Publication Date
JPS61151172A true JPS61151172A (ja) 1986-07-09

Family

ID=10571103

Family Applications (1)

Application Number Title Priority Date Filing Date
JP60278124A Pending JPS61151172A (ja) 1984-12-13 1985-12-12 インドール、その製造方法及びそれを含有する製薬組成物

Country Status (11)

Country Link
JP (1) JPS61151172A (it)
AU (1) AU579687B2 (it)
BE (1) BE903846A (it)
CH (1) CH667454A5 (it)
DE (1) DE3543982A1 (it)
FR (1) FR2574793B1 (it)
GB (2) GB8431426D0 (it)
IT (1) IT1182089B (it)
NL (1) NL8503424A (it)
SE (1) SE8505887L (it)
ZA (1) ZA859520B (it)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011168608A (ja) * 2002-12-20 2011-09-01 Ciba Holding Inc アミン類の合成及びその合成のための中間体

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds
GB8607824D0 (en) * 1986-03-27 1986-04-30 Glaxo Group Ltd Chemical compounds
GB8614287D0 (en) * 1986-06-12 1986-07-16 Glaxo Group Ltd Chemical compounds
US4894386A (en) * 1987-04-15 1990-01-16 Ici Americas Inc. Aliphatic carboxamides
GB8719167D0 (en) * 1987-08-13 1987-09-23 Glaxo Group Ltd Chemical compounds
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
SI21560B (sl) * 1990-06-07 2005-04-30 Astrazeneca Ab 3,5-disubstituirani indolni derivati kot "5-HT1-podobni" receptorski agonisti
GB9209882D0 (en) * 1992-05-07 1992-06-24 Glaxo Lab Sa Compositions
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
GB9216009D0 (en) * 1992-07-28 1992-09-09 Almirall Lab New indol derivatives
ES2056025B1 (es) * 1992-10-08 1995-05-01 Almirall Lab Nuevos derivados de indol.
FR2707639B1 (fr) * 1993-06-30 1995-10-13 Pf Medicament Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B.
WO2005118551A2 (en) 2004-05-28 2005-12-15 Ligand Pharmaceuticals Inc. Thrombopoietin activity modulating compounds and methods
CA2583764C (en) 2004-10-25 2009-06-09 Ligand Pharmaceuticals, Inc. Thrombopoietin activity modulating compounds and methods
JP5164972B2 (ja) 2007-03-29 2013-03-21 第一三共株式会社 ｃＰＬＡ２阻害活性を有するインドール誘導体およびその用途並びに製造方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA795239B (en) * 1978-10-12 1980-11-26 Glaxo Group Ltd Heterocyclic compounds
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
FR2574077A1 (fr) * 1984-12-04 1986-06-06 Glaxo Group Ltd Derives d'indoles, leur preparation et les compositions pharmaceutiques les contenant
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011168608A (ja) * 2002-12-20 2011-09-01 Ciba Holding Inc アミン類の合成及びその合成のための中間体
JP2012072174A (ja) * 2002-12-20 2012-04-12 Ciba Holding Inc アミン類の合成及びその合成のための中間体
US8710093B2 (en) 2002-12-20 2014-04-29 BASF SE Ludwigshafen Synthesis of amines and intermediates for the synthesis thereof

Also Published As

Publication number Publication date
IT1182089B (it) 1987-09-30
IT8548921A0 (it) 1985-12-12
DE3543982A1 (de) 1986-06-19
FR2574793A1 (fr) 1986-06-20
GB8431426D0 (en) 1985-01-23
ZA859520B (en) 1986-08-27
NL8503424A (nl) 1986-07-01
GB8530591D0 (en) 1986-01-22
BE903846A (fr) 1986-06-12
AU5115185A (en) 1986-06-19
GB2168347B (en) 1988-02-03
SE8505887L (sv) 1986-06-14
SE8505887D0 (sv) 1985-12-12
GB2168347A (en) 1986-06-18
AU579687B2 (en) 1988-12-01
FR2574793B1 (fr) 1988-10-14
CH667454A5 (fr) 1988-10-14

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