IT1314191B1 - Derivati isossazolcarbossamidici - Google Patents
Derivati isossazolcarbossamidiciInfo
- Publication number
- IT1314191B1 IT1314191B1 IT1999MI002173A ITMI992173A IT1314191B1 IT 1314191 B1 IT1314191 B1 IT 1314191B1 IT 1999MI002173 A IT1999MI002173 A IT 1999MI002173A IT MI992173 A ITMI992173 A IT MI992173A IT 1314191 B1 IT1314191 B1 IT 1314191B1
- Authority
- IT
- Italy
- Prior art keywords
- isossazolcarbossamidic
- derivatives
- isossazolcarbossamidic derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
Priority Applications (28)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT1999MI002173A IT1314191B1 (it) | 1999-10-18 | 1999-10-18 | Derivati isossazolcarbossamidici |
MYPI20004718A MY120400A (en) | 1999-10-18 | 2000-10-10 | Isoxazolecarboxamide derivatives |
JP2001531815A JP2003512362A (ja) | 1999-10-18 | 2000-10-16 | イソオキサゾールカルボキサミド誘導体 |
PCT/EP2000/010144 WO2001029015A2 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives as alpha1-adrenergic receptor antagonists |
HU0203184A HUP0203184A3 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives, process for their preparation and pharmaceutical compositions containing them |
PL00356990A PL356990A1 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives as alpha1-adrenergic receptor antagonists |
EP00992436A EP1226131B1 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives |
MXPA02003432A MXPA02003432A (es) | 1999-10-18 | 2000-10-16 | Derivados de isoxazolcarboxamida. |
ES00992436T ES2210033T3 (es) | 1999-10-18 | 2000-10-16 | Derivados de isoxazolcarboxamida. |
AT00992436T ATE256670T1 (de) | 1999-10-18 | 2000-10-16 | Isoxazolcarboxamid-derivate als antagonisten des alpha1-adrenergischen rezeptors |
CNB008143226A CN1139579C (zh) | 1999-10-18 | 2000-10-16 | 异噁唑甲酰胺衍生物 |
DE60007347T DE60007347T2 (de) | 1999-10-18 | 2000-10-16 | Isoxazolcarboxamid-derivate als antagonisten des alpha1-adrenergischen rezeptors |
NZ517884A NZ517884A (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives |
RU2002113096/04A RU2002113096A (ru) | 1999-10-18 | 2000-10-16 | Производные изоксазолкарбоксамида |
IL14883700A IL148837A0 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives |
BR0014851-2A BR0014851A (pt) | 1999-10-18 | 2000-10-16 | Derivados de isoxazolcarboxamida |
DK00992436T DK1226131T3 (da) | 1999-10-18 | 2000-10-16 | Isoxazolcarboxamidderivater |
PT00992436T PT1226131E (pt) | 1999-10-18 | 2000-10-16 | Derivados de isoxazolecarboxamida como antagonistas do receptor adrenergico alfa1 |
SI200030299T SI1226131T1 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives |
CA002385472A CA2385472A1 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives |
KR1020027004663A KR20020038944A (ko) | 1999-10-18 | 2000-10-16 | 아이속사졸카르복사미드 유도체 |
AU28347/01A AU757614B2 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives as alpha1-adrenergic receptor antagonists |
ARP000105475A AR029400A1 (es) | 1999-10-18 | 2000-10-18 | Derivados de isoxazolcarboxamida, un metodo para su preparacion y una composicion farmaceutica que los comprende |
US09/691,778 US6365591B1 (en) | 1999-10-18 | 2000-10-18 | Isoxazolecarboxamide derivatives |
US10/052,325 US6680319B2 (en) | 1999-10-18 | 2002-01-17 | Isoxazolecarboxamide derivatives |
NO20021803A NO20021803L (no) | 1999-10-18 | 2002-04-17 | Isoksazolkarboksamid-derivater |
ZA200203942A ZA200203942B (en) | 1999-10-18 | 2002-05-17 | Isoxazolecarboxamide derivatives. |
HK02105918.6A HK1044940A1 (zh) | 1999-10-18 | 2002-08-13 | 異噁唑咪唑羧酰胺衍生物 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT1999MI002173A IT1314191B1 (it) | 1999-10-18 | 1999-10-18 | Derivati isossazolcarbossamidici |
Publications (3)
Publication Number | Publication Date |
---|---|
ITMI992173A0 ITMI992173A0 (it) | 1999-10-18 |
ITMI992173A1 ITMI992173A1 (it) | 2001-04-18 |
IT1314191B1 true IT1314191B1 (it) | 2002-12-06 |
Family
ID=11383797
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT1999MI002173A IT1314191B1 (it) | 1999-10-18 | 1999-10-18 | Derivati isossazolcarbossamidici |
Country Status (25)
Country | Link |
---|---|
EP (1) | EP1226131B1 (it) |
JP (1) | JP2003512362A (it) |
KR (1) | KR20020038944A (it) |
CN (1) | CN1139579C (it) |
AR (1) | AR029400A1 (it) |
AT (1) | ATE256670T1 (it) |
AU (1) | AU757614B2 (it) |
BR (1) | BR0014851A (it) |
CA (1) | CA2385472A1 (it) |
DE (1) | DE60007347T2 (it) |
DK (1) | DK1226131T3 (it) |
ES (1) | ES2210033T3 (it) |
HK (1) | HK1044940A1 (it) |
HU (1) | HUP0203184A3 (it) |
IL (1) | IL148837A0 (it) |
IT (1) | IT1314191B1 (it) |
MX (1) | MXPA02003432A (it) |
MY (1) | MY120400A (it) |
NO (1) | NO20021803L (it) |
NZ (1) | NZ517884A (it) |
PL (1) | PL356990A1 (it) |
PT (1) | PT1226131E (it) |
RU (1) | RU2002113096A (it) |
WO (1) | WO2001029015A2 (it) |
ZA (1) | ZA200203942B (it) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0617306A2 (pt) | 2005-10-11 | 2011-07-19 | Hoffmann La Roche | derivados de isoxazol |
WO2007054444A2 (en) | 2005-11-09 | 2007-05-18 | F. Hoffmann-La Roche Ag | 3-aryl-isoxazole-4-carbonyl-benzofuran derivatives |
CA2633425A1 (en) | 2005-12-23 | 2007-06-28 | F. Hoffmann-La Roche Ag | Aryl-isoxazolo-4-yl-oxadiazole derivatives |
JP2009521516A (ja) | 2005-12-27 | 2009-06-04 | エフ.ホフマン−ラ ロシュ アーゲー | アリール−イソオキサゾール−4−イル−イミダゾール誘導体 |
RU2426732C2 (ru) | 2006-01-17 | 2011-08-20 | Ф. Хоффманн-Ля Рош Аг | АРИЛ-ИЗОКСАЗОЛ-4-ИЛ-ИМИДАЗО[1,2-a]ПИРИДИН, ПРИГОДНЫЙ ДЛЯ ЛЕЧЕНИЯ БОЛЕЗНИ АЛЬЦГЕЙМЕРА ЧЕРЕЗ ПОСРЕДСТВО GABA-РЕЦЕПТОРОВ |
ES2328185T3 (es) | 2006-05-31 | 2009-11-10 | F. Hoffmann-La Roche Ag | Derivados de aril-4-etinil-isoxazol. |
AU2008267894B2 (en) | 2007-06-22 | 2012-08-23 | F. Hoffmann-La Roche Ag | Isoxazole-imidazole derivatives |
CA2706990C (en) | 2007-12-04 | 2016-05-10 | F. Hoffmann-La Roche Ag | Isoxazolo-pyrazine derivatives |
US7902201B2 (en) | 2007-12-04 | 2011-03-08 | Hoffmann-La Roche Inc. | Isoxazolo-pyrazine derivatives |
US7943619B2 (en) | 2007-12-04 | 2011-05-17 | Hoffmann-La Roche Inc. | Isoxazolo-pyridazine derivatives |
WO2010081851A1 (en) | 2009-01-14 | 2010-07-22 | Genoscience Pharma | Piperidin-4-ylpiperazine compounds for the treatment of hcv infection |
TW201033201A (en) | 2009-02-19 | 2010-09-16 | Hoffmann La Roche | Isoxazole-isoxazole and isoxazole-isothiazole derivatives |
US8389550B2 (en) | 2009-02-25 | 2013-03-05 | Hoffmann-La Roche Inc. | Isoxazoles / O-pyridines with ethyl and ethenyl linker |
US8222246B2 (en) | 2009-04-02 | 2012-07-17 | Hoffmann-La Roche Inc. | Substituted isoxazoles |
US20100280019A1 (en) | 2009-04-30 | 2010-11-04 | Roland Jakob-Roetne | Isoxazoles |
CA2759598C (en) | 2009-05-05 | 2017-09-12 | F. Hoffmann-La Roche Ag | Isoxazole-thiazole derivatives as gaba a receptor inverse agonists for use in the treatment of cognitive disorders |
WO2010127976A1 (en) | 2009-05-05 | 2010-11-11 | F. Hoffmann-La Roche Ag | Isoxazole-pyridine derivatives |
EP2427458B1 (en) | 2009-05-05 | 2014-05-07 | F.Hoffmann-La Roche Ag | Isoxazole-pyridazine derivatives |
AU2010244552A1 (en) | 2009-05-05 | 2011-09-29 | F. Hoffmann-La Roche Ag | Isoxazole-pyrazole derivatives |
SG175318A1 (en) | 2009-05-07 | 2011-11-28 | Hoffmann La Roche | Isoxazole-pyridine derivatives as gaba modulators |
US8785435B2 (en) | 2011-10-20 | 2014-07-22 | Hoffmann-La Roche Inc. | Solid forms |
CN113121540B (zh) * | 2020-01-15 | 2024-01-26 | 鲁南制药集团股份有限公司 | 一种西格列汀游离碱的合成方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1254469B (it) * | 1992-02-25 | 1995-09-25 | Recordati Chem Pharm | Derivati benzopiranici e benzotiopiranici |
IT1266582B1 (it) * | 1993-07-30 | 1997-01-09 | Recordati Chem Pharm | Derivati (di)azacicloesanici e diazacicloeptanici |
DE4425146A1 (de) * | 1994-07-15 | 1996-01-18 | Basf Ag | Verwendung heterocyclischer Verbindungen |
-
1999
- 1999-10-18 IT IT1999MI002173A patent/IT1314191B1/it active
-
2000
- 2000-10-10 MY MYPI20004718A patent/MY120400A/en unknown
- 2000-10-16 DE DE60007347T patent/DE60007347T2/de not_active Expired - Fee Related
- 2000-10-16 BR BR0014851-2A patent/BR0014851A/pt not_active IP Right Cessation
- 2000-10-16 PT PT00992436T patent/PT1226131E/pt unknown
- 2000-10-16 EP EP00992436A patent/EP1226131B1/en not_active Expired - Lifetime
- 2000-10-16 NZ NZ517884A patent/NZ517884A/en unknown
- 2000-10-16 PL PL00356990A patent/PL356990A1/xx not_active Application Discontinuation
- 2000-10-16 HU HU0203184A patent/HUP0203184A3/hu unknown
- 2000-10-16 JP JP2001531815A patent/JP2003512362A/ja active Pending
- 2000-10-16 CN CNB008143226A patent/CN1139579C/zh not_active Expired - Fee Related
- 2000-10-16 AT AT00992436T patent/ATE256670T1/de not_active IP Right Cessation
- 2000-10-16 RU RU2002113096/04A patent/RU2002113096A/ru not_active Application Discontinuation
- 2000-10-16 WO PCT/EP2000/010144 patent/WO2001029015A2/en active IP Right Grant
- 2000-10-16 MX MXPA02003432A patent/MXPA02003432A/es not_active Application Discontinuation
- 2000-10-16 AU AU28347/01A patent/AU757614B2/en not_active Ceased
- 2000-10-16 KR KR1020027004663A patent/KR20020038944A/ko not_active Application Discontinuation
- 2000-10-16 CA CA002385472A patent/CA2385472A1/en not_active Abandoned
- 2000-10-16 IL IL14883700A patent/IL148837A0/xx unknown
- 2000-10-16 ES ES00992436T patent/ES2210033T3/es not_active Expired - Lifetime
- 2000-10-16 DK DK00992436T patent/DK1226131T3/da active
- 2000-10-18 AR ARP000105475A patent/AR029400A1/es not_active Application Discontinuation
-
2002
- 2002-04-17 NO NO20021803A patent/NO20021803L/no not_active Application Discontinuation
- 2002-05-17 ZA ZA200203942A patent/ZA200203942B/en unknown
- 2002-08-13 HK HK02105918.6A patent/HK1044940A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
MY120400A (en) | 2005-10-31 |
HUP0203184A3 (en) | 2004-12-28 |
HUP0203184A2 (hu) | 2003-01-28 |
ATE256670T1 (de) | 2004-01-15 |
PL356990A1 (en) | 2004-07-12 |
DE60007347T2 (de) | 2004-09-02 |
WO2001029015A3 (en) | 2001-11-01 |
NO20021803L (no) | 2002-06-17 |
ES2210033T3 (es) | 2004-07-01 |
WO2001029015A2 (en) | 2001-04-26 |
KR20020038944A (ko) | 2002-05-24 |
DE60007347D1 (de) | 2004-01-29 |
ITMI992173A0 (it) | 1999-10-18 |
NO20021803D0 (no) | 2002-04-17 |
AU757614B2 (en) | 2003-02-27 |
EP1226131A2 (en) | 2002-07-31 |
ZA200203942B (en) | 2003-01-02 |
MXPA02003432A (es) | 2002-08-20 |
HK1044940A1 (zh) | 2002-11-08 |
JP2003512362A (ja) | 2003-04-02 |
AR029400A1 (es) | 2003-06-25 |
IL148837A0 (en) | 2002-09-12 |
AU2834701A (en) | 2001-04-30 |
CN1139579C (zh) | 2004-02-25 |
DK1226131T3 (da) | 2004-04-19 |
RU2002113096A (ru) | 2003-11-10 |
ITMI992173A1 (it) | 2001-04-18 |
BR0014851A (pt) | 2002-06-11 |
CA2385472A1 (en) | 2001-04-26 |
CN1379767A (zh) | 2002-11-13 |
EP1226131B1 (en) | 2003-12-17 |
NZ517884A (en) | 2003-08-29 |
PT1226131E (pt) | 2004-05-31 |
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