IL160810A0 - 1-glyoxlylamide indolizines for treating cancer - Google Patents

1-glyoxlylamide indolizines for treating cancer

Info

Publication number
IL160810A0
IL160810A0 IL16081002A IL16081002A IL160810A0 IL 160810 A0 IL160810 A0 IL 160810A0 IL 16081002 A IL16081002 A IL 16081002A IL 16081002 A IL16081002 A IL 16081002A IL 160810 A0 IL160810 A0 IL 160810A0
Authority
IL
Israel
Prior art keywords
substituted
group
unsubstituted
independently
aryl group
Prior art date
Application number
IL16081002A
Other languages
English (en)
Original Assignee
Synta Pharmaceuticals Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synta Pharmaceuticals Corp filed Critical Synta Pharmaceuticals Corp
Publication of IL160810A0 publication Critical patent/IL160810A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
IL16081002A 2001-09-13 2002-09-13 1-glyoxlylamide indolizines for treating cancer IL160810A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32202001P 2001-09-13 2001-09-13
PCT/US2002/029154 WO2003022846A1 (en) 2001-09-13 2002-09-13 1-glyoxlylamide indolizines for treating cancer

Publications (1)

Publication Number Publication Date
IL160810A0 true IL160810A0 (en) 2004-08-31

Family

ID=23253054

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16081002A IL160810A0 (en) 2001-09-13 2002-09-13 1-glyoxlylamide indolizines for treating cancer

Country Status (20)

Country Link
US (2) US6861436B2 (xx)
EP (1) EP1432709B8 (xx)
JP (1) JP2005504795A (xx)
KR (1) KR20040053125A (xx)
CN (1) CN1568324A (xx)
AT (1) ATE300542T1 (xx)
AU (1) AU2002333626B2 (xx)
BR (1) BR0212794A (xx)
CA (1) CA2459886A1 (xx)
DE (1) DE60205265T2 (xx)
ES (1) ES2245747T3 (xx)
HK (1) HK1063322A1 (xx)
IL (1) IL160810A0 (xx)
IS (1) IS7176A (xx)
MX (1) MXPA04002323A (xx)
NO (1) NO20041035L (xx)
NZ (1) NZ531700A (xx)
PT (1) PT1432709E (xx)
WO (1) WO2003022846A1 (xx)
ZA (1) ZA200401996B (xx)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040116462A1 (en) * 2002-12-12 2004-06-17 Mitsunori Ono Indolizine compounds
DE60205265T2 (de) * 2001-09-13 2006-03-30 Synta Pharmaceuticals Corporation, Lexington 1-glyoxylamidindolizine zur behandlung von krebs
EP1537105A2 (en) * 2002-09-13 2005-06-08 Synta Pharmaceuticals Corporation Synthesis of indolizines
DE10318611A1 (de) 2003-04-24 2004-11-11 Elbion Ag 4-, 6- oder 7-Hydroxyindole mit N-Oxidgruppen und deren Verwendung als Therapeutika
WO2005099824A1 (en) * 2004-03-30 2005-10-27 Synta Pharmaceuticals, Corp. 1-glyoxylamide indolizines for treating lung and ovarian cancer
GB0413605D0 (en) 2004-06-17 2004-07-21 Addex Pharmaceuticals Sa Novel compounds
WO2006073938A2 (en) * 2004-12-30 2006-07-13 East Carolina University Method for the synthesis of 3-substituted indolizine and benzoindolizine compounds
BRPI0609802A2 (pt) * 2005-05-20 2017-05-02 Alantos Pharmaceuticals Holding Inc composto, composição farmacêutica e uso de um composto
US20070155738A1 (en) * 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
EP2320906B1 (en) * 2008-08-14 2016-02-24 Beta Pharma Canada Inc. Heterocyclic amide derivatives as ep4 receptor antagonists
RU2624506C2 (ru) 2009-04-29 2017-07-04 АМАРИН КОРПОРЕЙШН ПиЭлСи Фармацевтические композиции, содержащие ера и сердечно-сосудистое средство, и способы их применения
AR077428A1 (es) * 2009-07-29 2011-08-24 Sanofi Aventis (aza) indolizinacarboxamidas ciclicas su preparacion y su uso como agentes farmaceuticos
CN113603694B (zh) * 2021-07-16 2022-07-22 浙江工业大学 一种1,2-二酮类化合物及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2287706A (en) * 1994-03-21 1995-09-27 Fujisawa Pharmaceutical Co Indolizine derivatives
FR2757166B1 (fr) * 1996-12-12 1999-01-29 Rhone Poulenc Rorer Sa Derives du pyrrole, leur preparation et les compositions pharmaceutiques qui les contiennent
WO1998047507A1 (en) * 1997-04-24 1998-10-29 Shionogi & Co., Ltd. Method for the treatment of stroke using n-heterocyclic glyoxylamide compounds
EP1085021A4 (en) 1998-05-21 2003-01-08 Shionogi & Co DERIVATIVES OF PYRROLO 1,2-B] PYRIDAZINE, WITH INHIBITOR EFFECT ON SPLA 2?
WO2000021563A1 (fr) 1998-10-14 2000-04-20 Shionogi & Co., Ltd. Moyens de traitement et de prevention contre les troubles ischemiques dus a la repercussion
US6461538B2 (en) * 1999-12-16 2002-10-08 Fuji Photo Film Co., Ltd. Production process for indolizine compounds and their use in organic light-emitting devices
US20040116462A1 (en) * 2002-12-12 2004-06-17 Mitsunori Ono Indolizine compounds
DE60205265T2 (de) * 2001-09-13 2006-03-30 Synta Pharmaceuticals Corporation, Lexington 1-glyoxylamidindolizine zur behandlung von krebs

Also Published As

Publication number Publication date
ATE300542T1 (de) 2005-08-15
KR20040053125A (ko) 2004-06-23
US20040214850A1 (en) 2004-10-28
EP1432709A1 (en) 2004-06-30
CA2459886A1 (en) 2003-03-20
EP1432709B8 (en) 2005-11-02
EP1432709B1 (en) 2005-07-27
AU2002333626B2 (en) 2006-06-29
WO2003022846A1 (en) 2003-03-20
NO20041035L (no) 2004-04-30
MXPA04002323A (es) 2005-04-08
ZA200401996B (en) 2005-05-31
US20030153759A1 (en) 2003-08-14
DE60205265T2 (de) 2006-03-30
ES2245747T3 (es) 2006-01-16
CN1568324A (zh) 2005-01-19
NZ531700A (en) 2006-10-27
BR0212794A (pt) 2004-10-05
IS7176A (is) 2004-03-11
PT1432709E (pt) 2005-10-31
HK1063322A1 (en) 2004-12-24
JP2005504795A (ja) 2005-02-17
DE60205265D1 (de) 2005-09-01
US6861436B2 (en) 2005-03-01

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